AR087276A1 - Composiciones y metodos para tratar policitemia vera y trombocitemia esencial - Google Patents
Composiciones y metodos para tratar policitemia vera y trombocitemia esencialInfo
- Publication number
- AR087276A1 AR087276A1 ARP120102656A ARP120102656A AR087276A1 AR 087276 A1 AR087276 A1 AR 087276A1 AR P120102656 A ARP120102656 A AR P120102656A AR P120102656 A ARP120102656 A AR P120102656A AR 087276 A1 AR087276 A1 AR 087276A1
- Authority
- AR
- Argentina
- Prior art keywords
- methods
- compositions
- vera
- essential
- thrombocitemia
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 2
- 208000032027 Essential Thrombocythemia Diseases 0.000 abstract 2
- 208000017733 acquired polycythemia vera Diseases 0.000 abstract 2
- 208000037244 polycythemia vera Diseases 0.000 abstract 2
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 2
- -1 2-pyrrolidin-1-ylethoxy Chemical group 0.000 abstract 1
- KHBQMWCZKVMBLN-UHFFFAOYSA-N Benzenesulfonamide Chemical compound NS(=O)(=O)C1=CC=CC=C1 KHBQMWCZKVMBLN-UHFFFAOYSA-N 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Composiciones y métodos para tratar policitemia vera (PV) y/o trombocitemia esencial (ET) en un sujeto. Los métodos comprenden administrar al sujeto una cantidad eficaz de compuesto que es N-terc-butil-3-[(5-metil-2-{[4-(2-pirrolidin-1-iletoxi)fenil]amino}pirimidin-4-il)amino]bencenosulfonamida o una sal farmacéuticamente aceptable o un hidrato de éste.
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161510406P | 2011-07-21 | 2011-07-21 | |
| US201161510409P | 2011-07-21 | 2011-07-21 | |
| FR1251748 | 2012-02-27 | ||
| FR1251749 | 2012-02-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR087276A1 true AR087276A1 (es) | 2014-03-12 |
Family
ID=47558514
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP120102656A AR087276A1 (es) | 2011-07-21 | 2012-07-20 | Composiciones y metodos para tratar policitemia vera y trombocitemia esencial |
Country Status (3)
| Country | Link |
|---|---|
| AR (1) | AR087276A1 (es) |
| TW (1) | TW201316989A (es) |
| WO (1) | WO2013013195A1 (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2816957A1 (en) | 2010-11-07 | 2012-05-10 | Targegen, Inc. | Compositions and methods for treating myelofibrosis |
| FR3092581A1 (fr) * | 2019-02-12 | 2020-08-14 | Impact Biomedicines, Inc | Formes cristallines d'un inhibiteur de jak2 |
| JP2022519885A (ja) * | 2019-02-12 | 2022-03-25 | インパクト バイオメディシンズ インコーポレイテッド | Jak2阻害剤の結晶形態 |
| CA3188245A1 (en) * | 2020-08-04 | 2022-02-10 | Adrian SENDEROWICZ | 2-((4s)-6-(4-chlorophenyl)-1-methyl-4h-benzo[c]isoxazolo[4,5-e]azepin-4-yl)acetamide for treating thrombocythemia |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2470534A4 (en) * | 2009-08-24 | 2013-02-27 | Merck Sharp & Dohme | JAK INHIBITION FOR BLOCKING TOXICITY ASSOCIATED WITH RNA INTERFERENCE |
-
2012
- 2012-07-20 TW TW101126365A patent/TW201316989A/zh unknown
- 2012-07-20 AR ARP120102656A patent/AR087276A1/es not_active Application Discontinuation
- 2012-07-20 WO PCT/US2012/047704 patent/WO2013013195A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| TW201316989A (zh) | 2013-05-01 |
| WO2013013195A1 (en) | 2013-01-24 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ECSP13012658A (es) | Composiciones y métodos para el tratamiento de la mielofibrosis | |
| BR112014016805A8 (pt) | compostos terapeuticamente ativos e seus métodos de uso | |
| EA201490194A1 (ru) | Комбинированная терапия, включающая ингибитор cdk4/6 и ингибитор pi3k для применения в лечении рака | |
| MX2016004580A (es) | Uso de un inhibidor de pcsk9 para tratar la hiperlipidemia. | |
| EA201201680A1 (ru) | Морфолинопиримидины и их применение в терапии | |
| MX2021008610A (es) | Tratamiento del cancer usando combinaciones de inhibidores de erk y raf. | |
| GT201400009A (es) | 4-imidazopiridazin-1-il-benzamidas y 4-imidazotriazin-1-il-benzamidas como inhibidores de btk | |
| BR112013025386A2 (pt) | combinação de um composto, composto de fórmula ia ou um sal farmaceuticamente aceitável do mesmo, método para tratamento de uma doença ou afecção modulada por mutação braf v600e e altos níveis de pakt em um mamífero e uso | |
| GT201300266A (es) | Derivados de pirrolotriazinona como inhibidores de pi3k | |
| EA201391285A1 (ru) | Производные тетрагидрохинолина, полезные в качестве ингибиторов бромодомена | |
| EA201390803A1 (ru) | Ингибиторы бромодомена и их применение | |
| CL2013001093A1 (es) | Compuestos triciclicos inhibidores de la quinasa pi3 (pi3k); composicion farmaceutica que los comprende; metodo para tratar el cancer; y su uso para el tratamiento del cancer . | |
| CL2016000241A1 (es) | Formulación de inhibidores de la syk. | |
| IN2014DN10386A (es) | ||
| ECSP13013011A (es) | Triazolopiridinas | |
| MX2016015434A (es) | Combinaciones farmaceuticas para tratar cancer. | |
| UA108711C2 (uk) | Сполуки триазолопіридину як інгібітори фосфодіестерази pde10a | |
| DOP2013000131A (es) | Composiciones y métodos para tratar el cáncer usando un inhibidor de pi3k y un inhibidor de mek | |
| AR087276A1 (es) | Composiciones y metodos para tratar policitemia vera y trombocitemia esencial | |
| CL2013003556A1 (es) | Compuestos derivados de ftalazinona-pirrolo[3,2-d]pirimidin-carboxamida, inhibidoers de fosfodiesterasa tipo 4 y tipo 5; composcin farmaceutica que o comprende, combinacion fija, no fija y kit, uso del compuesto en la preparacion de un medicamento para trata enfermedaes de las vias respiratorias | |
| MX2013014398A (es) | Derivados de sulfonamida heterociclicos. | |
| BR112015005392A2 (pt) | formulação de comprimido de um inibidor de fosfatidilinositol 3-cinase | |
| AR081024A1 (es) | Asociacion de los inhibidores de la xantina oxidasa y la metformina y su uso | |
| DOP2014000221A (es) | Métodos para tratar el cáncer usando inhibidor de pi3k e inhibidor de mek | |
| BR112015025033A2 (pt) | prodrogas de inibidores da pde-5 do tipo pirimidina bicíclico substituídas |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |