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TW201316989A - 用於治療真性多血症及原發性血小板過多症之組合物及方法 - Google Patents

用於治療真性多血症及原發性血小板過多症之組合物及方法 Download PDF

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Publication number
TW201316989A
TW201316989A TW101126365A TW101126365A TW201316989A TW 201316989 A TW201316989 A TW 201316989A TW 101126365 A TW101126365 A TW 101126365A TW 101126365 A TW101126365 A TW 101126365A TW 201316989 A TW201316989 A TW 201316989A
Authority
TW
Taiwan
Prior art keywords
compound
individual
amino
butyl
phenyl
Prior art date
Application number
TW101126365A
Other languages
English (en)
Chinese (zh)
Inventor
Pamela Cohen
Frank Neumann
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of TW201316989A publication Critical patent/TW201316989A/zh

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
TW101126365A 2011-07-21 2012-07-20 用於治療真性多血症及原發性血小板過多症之組合物及方法 TW201316989A (zh)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201161510406P 2011-07-21 2011-07-21
US201161510409P 2011-07-21 2011-07-21
FR1251748 2012-02-27
FR1251749 2012-02-27

Publications (1)

Publication Number Publication Date
TW201316989A true TW201316989A (zh) 2013-05-01

Family

ID=47558514

Family Applications (1)

Application Number Title Priority Date Filing Date
TW101126365A TW201316989A (zh) 2011-07-21 2012-07-20 用於治療真性多血症及原發性血小板過多症之組合物及方法

Country Status (3)

Country Link
AR (1) AR087276A1 (es)
TW (1) TW201316989A (es)
WO (1) WO2013013195A1 (es)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116367839A (zh) * 2020-08-04 2023-06-30 星座制药公司 2-((4s)-6-(4-氯苯基)-1-甲基-4h-苯并[c]异恶唑并[4,5-e]氮杂卓-4-基)乙酰胺用于治疗血小板增多症

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2012060847A1 (en) 2010-11-07 2012-05-10 Targegen, Inc. Compositions and methods for treating myelofibrosis
FR3092581A1 (fr) * 2019-02-12 2020-08-14 Impact Biomedicines, Inc Formes cristallines d'un inhibiteur de jak2
CN113840604B (zh) * 2019-02-12 2025-04-25 生物医学影响公司 Jak2抑制剂的结晶形式

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011025685A1 (en) * 2009-08-24 2011-03-03 Merck Sharp & Dohme Corp. Jak inhibition blocks rna interference associated toxicities

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116367839A (zh) * 2020-08-04 2023-06-30 星座制药公司 2-((4s)-6-(4-氯苯基)-1-甲基-4h-苯并[c]异恶唑并[4,5-e]氮杂卓-4-基)乙酰胺用于治疗血小板增多症

Also Published As

Publication number Publication date
AR087276A1 (es) 2014-03-12
WO2013013195A1 (en) 2013-01-24

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