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AR058019A1 - Proceso de preparacion de un derivado de pirrolopirimidina - Google Patents

Proceso de preparacion de un derivado de pirrolopirimidina

Info

Publication number
AR058019A1
AR058019A1 ARP060103390A ARP060103390A AR058019A1 AR 058019 A1 AR058019 A1 AR 058019A1 AR P060103390 A ARP060103390 A AR P060103390A AR P060103390 A ARP060103390 A AR P060103390A AR 058019 A1 AR058019 A1 AR 058019A1
Authority
AR
Argentina
Prior art keywords
pirrolopirimidine
derivative
preparation process
phenyl
ethyl
Prior art date
Application number
ARP060103390A
Other languages
English (en)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of AR058019A1 publication Critical patent/AR058019A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Reivindicacion 1: Un método para la preparacion de {6-[4-(4-etil-piperazin-1-ilmetil)-fenil-7H-pirrolo-[2,3-d]-pirimidin-4-il]-(R-1-fenil-etil)amina, que tiene la formula (1), la cual comprende reducir la fraccion de amida del compuesto de la formula (2).
ARP060103390A 2005-08-05 2006-08-03 Proceso de preparacion de un derivado de pirrolopirimidina AR058019A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US70607105P 2005-08-05 2005-08-05

Publications (1)

Publication Number Publication Date
AR058019A1 true AR058019A1 (es) 2008-01-23

Family

ID=37198768

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP060103390A AR058019A1 (es) 2005-08-05 2006-08-03 Proceso de preparacion de un derivado de pirrolopirimidina

Country Status (15)

Country Link
US (1) US20080227980A1 (es)
EP (1) EP1919917A2 (es)
JP (1) JP2009503034A (es)
KR (1) KR20080040695A (es)
CN (1) CN101238130A (es)
AR (1) AR058019A1 (es)
AU (1) AU2006277997A1 (es)
BR (1) BRPI0614710A2 (es)
CA (1) CA2617720A1 (es)
GT (1) GT200600349A (es)
MX (1) MX2008001611A (es)
PE (1) PE20070415A1 (es)
RU (1) RU2008108089A (es)
TW (1) TW200726770A (es)
WO (1) WO2007017468A2 (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7955473B2 (en) 2004-12-22 2011-06-07 Akzo Nobel N.V. Process for the production of paper
US20060254464A1 (en) 2005-05-16 2006-11-16 Akzo Nobel N.V. Process for the production of paper
US8273216B2 (en) 2005-12-30 2012-09-25 Akzo Nobel N.V. Process for the production of paper
RU2008134314A (ru) * 2006-01-23 2010-02-27 Новартис АГ (CH) Твердые формы производного пирролопиримидина и их применение в качестве противоопухолевых агентов
WO2010150921A1 (ja) 2009-06-26 2010-12-29 帝人ファーマ株式会社 高血圧症または正常高値血圧症の治療薬
KR20120125332A (ko) 2010-02-01 2012-11-14 바스프 에스이 동물 해충을 퇴치하기 위한 치환된 케톤계 이속사졸린 화합물 및 유도체
AR083646A1 (es) 2010-10-01 2013-03-13 Basf Se Compuestos de imina, composiciones veterinarias y agricolas que los contienen y su uso en el control de plagas de invertebrados
BR112013007056A2 (pt) 2010-10-01 2019-09-24 Basf Se compostos de imina
CN110498812B (zh) * 2018-05-17 2021-08-24 上海医药工业研究院 一种艾拉普林的中间体化合物的制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CZ1598A3 (cs) * 1995-07-06 1998-04-15 Novartis Ag Pyrrolopyrimidiny a způsoby jejich přípravy
GB0119249D0 (en) * 2001-08-07 2001-10-03 Novartis Ag Organic compounds

Also Published As

Publication number Publication date
BRPI0614710A2 (pt) 2011-04-12
JP2009503034A (ja) 2009-01-29
WO2007017468A3 (en) 2007-05-03
KR20080040695A (ko) 2008-05-08
CA2617720A1 (en) 2007-02-15
GT200600349A (es) 2007-02-28
PE20070415A1 (es) 2007-05-29
WO2007017468A2 (en) 2007-02-15
RU2008108089A (ru) 2009-09-10
US20080227980A1 (en) 2008-09-18
TW200726770A (en) 2007-07-16
MX2008001611A (es) 2008-02-19
AU2006277997A1 (en) 2007-02-15
EP1919917A2 (en) 2008-05-14
CN101238130A (zh) 2008-08-06

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