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AR043046A1 - Compuestos de amida de acido carboxilico con efecto antagonico de la hcm, medicamentos que contienen estos compuestos y procedimientos para su preparacion - Google Patents

Compuestos de amida de acido carboxilico con efecto antagonico de la hcm, medicamentos que contienen estos compuestos y procedimientos para su preparacion

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Publication number
AR043046A1
AR043046A1 ARP030103034A ARP030103034A AR043046A1 AR 043046 A1 AR043046 A1 AR 043046A1 AR P030103034 A ARP030103034 A AR P030103034A AR P030103034 A ARP030103034 A AR P030103034A AR 043046 A1 AR043046 A1 AR 043046A1
Authority
AR
Argentina
Prior art keywords
alkyl
group
phenyl
atoms
independently
Prior art date
Application number
ARP030103034A
Other languages
English (en)
Spanish (es)
Inventor
Dirk Stenkamp
Martin Lenter
Heike-Andrea Wieland
Rudolf Klaus Dr
Stephan Georg Mueller
Ralf R H Lotz
Kirsten Arndt
Lustenberger Philipp Dr
Thorsten Lehmann-Lintz
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of AR043046A1 publication Critical patent/AR043046A1/es

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    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
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    • C07C233/78—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
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    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/20—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
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PL375344A1 (en) 2005-11-28
BR0313790A (pt) 2005-07-12
WO2004024702A1 (de) 2004-03-25
PE20040974A1 (es) 2005-01-12
HRP20050179A2 (en) 2006-05-31
RS20050173A (sr) 2007-09-21
NO20050068L (no) 2005-03-04
EA200500301A1 (ru) 2006-02-24
JP2006507246A (ja) 2006-03-02
ECSP055615A (es) 2005-05-30
EP1534689A1 (de) 2005-06-01
ZA200500086B (en) 2006-07-26
CA2496563A1 (en) 2004-03-25
CN1678591A (zh) 2005-10-05
MXPA05002158A (es) 2005-05-23

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