MXPA03010134A - Derivados de ciclohexan-1-4-diamina sustituidos. - Google Patents
Derivados de ciclohexan-1-4-diamina sustituidos.Info
- Publication number
- MXPA03010134A MXPA03010134A MXPA03010134A MXPA03010134A MXPA03010134A MX PA03010134 A MXPA03010134 A MX PA03010134A MX PA03010134 A MXPA03010134 A MX PA03010134A MX PA03010134 A MXPA03010134 A MX PA03010134A MX PA03010134 A MXPA03010134 A MX PA03010134A
- Authority
- MX
- Mexico
- Prior art keywords
- substituted cyclohexane
- diamine derivatives
- diamine
- cyclohexane
- medicaments
- Prior art date
Links
- VKIRRGRTJUUZHS-UHFFFAOYSA-N cyclohexane-1,4-diamine Chemical class NC1CCC(N)CC1 VKIRRGRTJUUZHS-UHFFFAOYSA-N 0.000 title abstract 3
- 239000003814 drug Substances 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C211/00—Compounds containing amino groups bound to a carbon skeleton
- C07C211/33—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings
- C07C211/34—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of a saturated carbon skeleton
- C07C211/36—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of a saturated carbon skeleton containing at least two amino groups bound to the carbon skeleton
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- A—HUMAN NECESSITIES
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/132—Amines having two or more amino groups, e.g. spermidine, putrescine
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- A—HUMAN NECESSITIES
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- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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- A—HUMAN NECESSITIES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
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- Health & Medical Sciences (AREA)
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- Pharmacology & Pharmacy (AREA)
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- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
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- Engineering & Computer Science (AREA)
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- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
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- Pain & Pain Management (AREA)
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- Psychiatry (AREA)
- Heart & Thoracic Surgery (AREA)
- Immunology (AREA)
- Endocrinology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Diabetes (AREA)
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- Gynecology & Obstetrics (AREA)
- Hospice & Palliative Care (AREA)
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- Nutrition Science (AREA)
- Anesthesiology (AREA)
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- Obesity (AREA)
- Dermatology (AREA)
Abstract
La invencion se refiere a derivados de ciclohexan-1,4-diamina derivados, procedimientos para su preparacion, medicamentos conteniendo estos compuestos y el uso de derivados de ciclohexan-1,4-diamina sustituidos para la preparacion de medicamentos.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10123163A DE10123163A1 (de) | 2001-05-09 | 2001-05-09 | Substituierte Cyclohexan-1,4-diaminderivate |
| PCT/EP2002/005051 WO2002090317A1 (de) | 2001-05-09 | 2002-05-08 | Substituierte cyclohexan-1,4-diaminderivate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA03010134A true MXPA03010134A (es) | 2004-03-10 |
Family
ID=7684562
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA03010201A MXPA03010201A (es) | 2001-05-09 | 2002-05-08 | Derivados de 2-piridin-ciclohexan-1,4-diamina sustituidos. |
| MXPA03010134A MXPA03010134A (es) | 2001-05-09 | 2002-05-08 | Derivados de ciclohexan-1-4-diamina sustituidos. |
| MXPA03010195A MXPA03010195A (es) | 2001-05-09 | 2002-05-09 | Derivados de ciclohexan-1,4-diamina sustituidos con actividad antiarreica y analgesica periferica. |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA03010201A MXPA03010201A (es) | 2001-05-09 | 2002-05-08 | Derivados de 2-piridin-ciclohexan-1,4-diamina sustituidos. |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA03010195A MXPA03010195A (es) | 2001-05-09 | 2002-05-09 | Derivados de ciclohexan-1,4-diamina sustituidos con actividad antiarreica y analgesica periferica. |
Country Status (30)
| Country | Link |
|---|---|
| US (3) | US20040229872A1 (es) |
| EP (3) | EP1385825B1 (es) |
| JP (3) | JP2004533439A (es) |
| KR (2) | KR100895778B1 (es) |
| CN (2) | CN1533374B (es) |
| AR (1) | AR035883A1 (es) |
| AT (2) | ATE359260T1 (es) |
| AU (3) | AU2002341195B2 (es) |
| BR (2) | BR0209580A (es) |
| CA (3) | CA2446463C (es) |
| CO (2) | CO5700725A2 (es) |
| CY (2) | CY1106468T1 (es) |
| CZ (2) | CZ20032995A3 (es) |
| DE (3) | DE10123163A1 (es) |
| DK (2) | DK1385825T3 (es) |
| EC (2) | ECSP034830A (es) |
| ES (2) | ES2291486T3 (es) |
| HU (3) | HU228253B1 (es) |
| IL (4) | IL158782A0 (es) |
| MX (3) | MXPA03010201A (es) |
| NO (2) | NO328600B1 (es) |
| NZ (2) | NZ529334A (es) |
| PE (1) | PE20021094A1 (es) |
| PL (3) | PL212887B1 (es) |
| PT (2) | PT1385825E (es) |
| RU (2) | RU2321579C2 (es) |
| SI (2) | SI1385825T1 (es) |
| SK (2) | SK287319B6 (es) |
| WO (3) | WO2002090330A1 (es) |
| ZA (2) | ZA200309522B (es) |
Families Citing this family (48)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10252665A1 (de) | 2002-11-11 | 2004-06-03 | Grünenthal GmbH | 4-Aminomethyl-1-aryl-cyclohexylamin-Derivate |
| DE10252650A1 (de) * | 2002-11-11 | 2004-05-27 | Grünenthal GmbH | Cyclohexyl-Harnstoff-Derivate |
| AU2003296564A1 (en) | 2002-11-12 | 2004-06-03 | Grunenthal Gmbh | 4-hydroxymethyl-1-aryl-cyclohexylamine derivatives |
| EA200500846A1 (ru) | 2002-11-19 | 2005-12-29 | Ачиллион Фармасьютикалз, Инк. | Замещенные арилтиомочевины и родственные соединения; ингибиторы вирусной репликации |
| US7354988B2 (en) | 2003-08-12 | 2008-04-08 | General Electric Company | Electrically conductive compositions and method of manufacture thereof |
| US7026432B2 (en) | 2003-08-12 | 2006-04-11 | General Electric Company | Electrically conductive compositions and method of manufacture thereof |
| US7378409B2 (en) | 2003-08-21 | 2008-05-27 | Bristol-Myers Squibb Company | Substituted cycloalkylamine derivatives as modulators of chemokine receptor activity |
| US7309727B2 (en) | 2003-09-29 | 2007-12-18 | General Electric Company | Conductive thermoplastic compositions, methods of manufacture and articles derived from such compositions |
| DE10360793A1 (de) * | 2003-12-23 | 2005-07-28 | Grünenthal GmbH | Spirocyclische Cyclohexan-Derivate |
| DE10360792A1 (de) * | 2003-12-23 | 2005-07-28 | Grünenthal GmbH | Spirocyclische Cyclohexan-Derivate |
| DE102004023506A1 (de) | 2004-05-10 | 2005-12-01 | Grünenthal GmbH | Kettenverlängerte substituierte Cyclohexyl-1,4-diamin-Derivate |
| DE102004023635A1 (de) | 2004-05-10 | 2006-04-13 | Grünenthal GmbH | Heteroarylsubstituierte Cyclohexyl-1,4-diamin-Derivate |
| DE102004023632A1 (de) * | 2004-05-10 | 2005-12-08 | Grünenthal GmbH | Substituierte Cyclohexylcarbonsäure-Derivate |
| DE102004023501A1 (de) | 2004-05-10 | 2005-12-01 | Grünenthal GmbH | Oxosubstituierte Cyclohexyl-1,4-diamin-Derivate |
| DE102004023507A1 (de) * | 2004-05-10 | 2005-12-01 | Grünenthal GmbH | Substituierte Cyclohexylessigsäure-Derivate |
| DE102004023522A1 (de) | 2004-05-10 | 2005-12-01 | Grünenthal GmbH | Substituierte Cyclohexyl-1,4-diamin-Derivate |
| DE102004023508A1 (de) | 2004-05-10 | 2005-12-08 | Grünenthal GmbH | Säurederivate substituierter Cyclohexyl-1,4-diamine |
| TW200600492A (en) * | 2004-05-18 | 2006-01-01 | Achillion Pharmaceuticals Inc | Substituted aryl acylthioureas and related compounds; inhibitors of viral replication |
| US7462656B2 (en) | 2005-02-15 | 2008-12-09 | Sabic Innovative Plastics Ip B.V. | Electrically conductive compositions and method of manufacture thereof |
| DE102005061428A1 (de) | 2005-12-22 | 2007-08-16 | Grünenthal GmbH | Substituierte Cyclohexylmethyl-Derivate |
| DE102006033114A1 (de) | 2006-07-18 | 2008-01-24 | Grünenthal GmbH | Spirocyclische Azaindol-Derivate |
| DE102006033109A1 (de) * | 2006-07-18 | 2008-01-31 | Grünenthal GmbH | Substituierte Heteroaryl-Derivate |
| DE102006035787A1 (de) | 2006-07-28 | 2008-03-13 | Tesa Ag | Verfahren zum Stanzen von bei Raumtemperatur nicht tackigen hitzeaktivierbaren Klebmassen |
| WO2008089307A2 (en) * | 2007-01-18 | 2008-07-24 | Lexicon Pharmaceuticals, Inc. | Delta 5 desaturase inhibitors for the treatment of pain, inflammation and cancer |
| MX2009013676A (es) * | 2007-06-15 | 2010-06-01 | Mission Pharma Co | Metodos y composiciones para inhibir el factor de edema y la adenilil ciclasa. |
| US20090215725A1 (en) * | 2008-02-26 | 2009-08-27 | Grunenthal Gmbh | Substituted 4-aminocyclohexane derivatives |
| AR071067A1 (es) | 2008-03-27 | 2010-05-26 | Gruenenthal Chemie | Ciclohexildiaminas sustituidas |
| PT2260042E (pt) | 2008-03-27 | 2011-12-06 | Gruenenthal Gmbh | Derivados de ciclo-hexano espirocíclicos substituídos |
| CA2719739A1 (en) | 2008-03-27 | 2009-10-01 | Sven Frormann | Hydroxymethylcyclohexylamines |
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