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MX2018003261A - Coterapia que comprende canagliflozina y fentermina para el tratamiento de la obesidad y de los trastornos relacionados con la obesidad. - Google Patents

Coterapia que comprende canagliflozina y fentermina para el tratamiento de la obesidad y de los trastornos relacionados con la obesidad.

Info

Publication number
MX2018003261A
MX2018003261A MX2018003261A MX2018003261A MX2018003261A MX 2018003261 A MX2018003261 A MX 2018003261A MX 2018003261 A MX2018003261 A MX 2018003261A MX 2018003261 A MX2018003261 A MX 2018003261A MX 2018003261 A MX2018003261 A MX 2018003261A
Authority
MX
Mexico
Prior art keywords
obesity
treat
delay
prevent
therapy
Prior art date
Application number
MX2018003261A
Other languages
English (en)
Other versions
MX383002B (es
Inventor
R Rosenthal Norman
C Polidori David
K Ways Douglas
P Stein Peter
Rothenberg Paul
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of MX2018003261A publication Critical patent/MX2018003261A/es
Publication of MX383002B publication Critical patent/MX383002B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Child & Adolescent Psychology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención está dirigida al uso de una coterapia que comprende administrar canagliflozina y fentermina para el tratamiento de la obesidad y de trastornos relacionados con la obesidad; más particularmente, la presente invención está dirigida a una coterapia para tratar la obesidad, para promover la pérdida de peso y/o para suprimir el apetito; para tratar, retrasar, ralentizar el avance y/o prevenir trastornos metabólicos (que incluyen, por ejemplo, la diabetes mellitus tipo 2); para tratar, retrasar, ralentizar el avance y/o prevenir trastornos renales o de hígado graso (que incluyen, por ejemplo, EHNA, HGNA, etc.); para tratar, retrasar, ralentizar el avance y/o prevenir trastornos del sueño (que incluyen, por ejemplo, apnea del sueño); para proporcionar protección cardiovascular; para tratar, retrasar, ralentizar el avance y/o prevenir eventos cardiovasculares (que incluyen eventos cardíacos adversos mayores (ECAM), tales como infarto de miocardio, angina inestable, muerte cardiovascular, revascularización, accidente cerebrovascular fatal o no fatal, arteriopatía periférica, eventos aórticos, hospitalización por insuficiencia cardíaca congestiva, etc.); y/o para extender o prolongar la longevidad.
MX2018003261A 2015-09-15 2016-09-13 Coterapia que comprende canagliflozina y fentermina para el tratamiento de la obesidad y de los trastornos relacionados con la obesidad. MX383002B (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201562218842P 2015-09-15 2015-09-15
US201662306110P 2016-03-10 2016-03-10
US15/262,038 US20170071970A1 (en) 2015-09-15 2016-09-12 Co-therapy comprising canagliflozin and phentermine for the treatment of obesity and obesity related disorders
PCT/US2016/051435 WO2017048670A1 (en) 2015-09-15 2016-09-13 Co-therapy comprising canagliflozin and phentermine for the treatment of obesity and obesity related disorders

Publications (2)

Publication Number Publication Date
MX2018003261A true MX2018003261A (es) 2018-05-17
MX383002B MX383002B (es) 2025-03-04

Family

ID=58236464

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2018003261A MX383002B (es) 2015-09-15 2016-09-13 Coterapia que comprende canagliflozina y fentermina para el tratamiento de la obesidad y de los trastornos relacionados con la obesidad.

Country Status (18)

Country Link
US (3) US20170071970A1 (es)
EP (1) EP3349740B1 (es)
JP (1) JP2018527374A (es)
KR (1) KR20180051560A (es)
CN (1) CN108024977A (es)
AU (1) AU2016322537B2 (es)
CA (1) CA2998730A1 (es)
CO (1) CO2018002708A2 (es)
EA (1) EA201890738A1 (es)
ES (1) ES2873117T3 (es)
HK (1) HK1248124A1 (es)
IL (1) IL257876A (es)
MX (1) MX383002B (es)
PH (1) PH12018500501A1 (es)
TW (1) TW201722413A (es)
UA (1) UA122974C2 (es)
WO (1) WO2017048670A1 (es)
ZA (1) ZA201802448B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI835735B (zh) * 2017-06-12 2024-03-21 比利時商健生藥品公司 減少或預防第ii型糖尿病患者中心血管事件之方法
CN110038009B (zh) * 2019-05-13 2021-01-08 浙江大学 卡格列净在制备抗肿瘤药物中的应用
TW202535454A (zh) * 2020-02-18 2025-09-16 丹麥商諾佛 儂迪克股份有限公司 醫藥配方
CN112716940A (zh) * 2021-02-18 2021-04-30 苏州大学 卡格列净在制备治疗与stat6蛋白相关疾病的药物中的应用
CN113812378B (zh) * 2021-09-29 2023-02-03 湖北天勤生物技术研究院有限公司 一种食蟹猴肥胖症模型的建立方法及其应用
CN113893349B (zh) * 2021-12-13 2022-07-22 北京大学第三医院（北京大学第三临床医学院） 达格列净及其类似物在制备防治雄性生殖功能障碍的药物中的用途

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