MX2009009332A - Antagonista del receptor de mineralocorticoides para el tratamiento de endometriosis. - Google Patents
Antagonista del receptor de mineralocorticoides para el tratamiento de endometriosis.Info
- Publication number
- MX2009009332A MX2009009332A MX2009009332A MX2009009332A MX2009009332A MX 2009009332 A MX2009009332 A MX 2009009332A MX 2009009332 A MX2009009332 A MX 2009009332A MX 2009009332 A MX2009009332 A MX 2009009332A MX 2009009332 A MX2009009332 A MX 2009009332A
- Authority
- MX
- Mexico
- Prior art keywords
- endometriosis
- treatment
- mineralcorticoid receptor
- receptor antagonists
- present
- Prior art date
Links
- 201000009273 Endometriosis Diseases 0.000 title abstract 4
- 239000002395 mineralocorticoid Substances 0.000 title abstract 3
- 239000002464 receptor antagonist Substances 0.000 title abstract 3
- 229940044551 receptor antagonist Drugs 0.000 title abstract 3
- 239000003814 drug Substances 0.000 abstract 2
- 210000000988 bone and bone Anatomy 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 230000002349 favourable effect Effects 0.000 abstract 1
- 229940124597 therapeutic agent Drugs 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
- A61K31/585—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Oncology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Steroid Compounds (AREA)
Abstract
Es objeto de la presente invención el uso de antagonistas del receptor de mineralocorticoides para preparar un medicamento para el tratamiento de endometriosis. En especial, la presente invención se refiere a un agente terapéutico mejorado contra la endometriosis, que muestra un perfil de acción o de efectos colaterales más ventajoso que las terapias de tratamiento disponibles hasta ahora. Con un antagonista del receptor de mineralocorticoides se puede tratar la endometriosis de modo duradero, sin que se produzca, en este caso, una pérdida de la masa ósea.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102007011105A DE102007011105A1 (de) | 2007-03-02 | 2007-03-02 | Mineralcorticoid-Rezeptor-Antagonisten zur Behandlung von Endometriose |
| PCT/EP2008/052456 WO2008107373A1 (de) | 2007-03-02 | 2008-02-28 | Mineralcorticoid-rezeptor-antagonisten zur behandlung von endometriose |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2009009332A true MX2009009332A (es) | 2009-09-11 |
Family
ID=39431148
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2009009332A MX2009009332A (es) | 2007-03-02 | 2008-02-28 | Antagonista del receptor de mineralocorticoides para el tratamiento de endometriosis. |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20110003778A1 (es) |
| EP (1) | EP2131825A1 (es) |
| JP (1) | JP2010520178A (es) |
| KR (1) | KR20090119870A (es) |
| CN (1) | CN101621995A (es) |
| AR (1) | AR065585A1 (es) |
| AU (1) | AU2008223859A1 (es) |
| BR (1) | BRPI0808427A2 (es) |
| CA (1) | CA2679520A1 (es) |
| DE (1) | DE102007011105A1 (es) |
| IL (1) | IL200380A0 (es) |
| MX (1) | MX2009009332A (es) |
| RU (1) | RU2009136305A (es) |
| TW (1) | TW200900080A (es) |
| WO (1) | WO2008107373A1 (es) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI1003661A2 (pt) * | 2010-09-15 | 2013-01-08 | Libbs Farmaceutica Ltda | associaÇço farmacÊutica para tratar e/ou prevenir mioma e/ou endometriose, uso de resveratrol e progestogenio, composiÇço farmacÊutica para tratamento e/ou prevenÇço de mioma e/ou endometriose medicamento para tratamento e/ou prevenÇço de mioma e/ou endometrios, kit e mÉtodo para tratamento e/ou prevenÇço de mioma e/ou endometriose |
| EA201400537A1 (ru) | 2011-11-04 | 2014-10-30 | Байер Фарма Акциенгезельшафт | 18-МЕТИЛ-6,7-МЕТИЛЕН-3-ОКСО-17-ПРЕГН-4-ЕН-21,17β-КАРБОЛАКТОНЫ, ФАРМАЦЕВТИЧЕСКИЕ КОМПОЗИЦИИ, СОДЕРЖАЩИЕ УКАЗАННЫЕ СОЕДИНЕНИЯ, И ИХ ПРИМЕНЕНИЕ В ЛЕЧЕНИИ ЭНДОМЕТРИОЗА |
| TW201350122A (zh) * | 2012-04-23 | 2013-12-16 | Bayer Pharma AG | 18-甲基-15β,16β-亞甲基-19-降-20-螺氧-4-烯-3-酮的子宮內用途,包含18-甲基-15β,16β-亞甲基-19-降-20-螺氧-4-烯-3-酮的子宮內系統,及其於避孕及婦科治療之用途 |
| UA115576C2 (uk) | 2012-12-06 | 2017-11-27 | Байєр Фарма Акцієнгезелльшафт | Похідні бензимідазолу як антагоністи ер4 |
| WO2014115449A1 (ja) * | 2013-01-22 | 2014-07-31 | シャープ株式会社 | 液晶表示装置 |
| TW201607943A (zh) | 2013-12-19 | 2016-03-01 | 拜耳製藥公司 | 作為ep4配體之新穎苯并咪唑衍生物 |
| CN117959293B (zh) * | 2024-01-18 | 2025-05-13 | 香港大学深圳医院 | 非奈利酮在制备治疗和/或预防卵巢功能障碍疾病药物中的应用 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4042004A1 (de) * | 1990-12-22 | 1992-06-25 | Schering Ag | 14(beta)-h-, 14- u. 15-en-11(beta)-aryl-4-estrene |
| DE4042005A1 (de) * | 1990-12-22 | 1992-06-25 | Schering Ag | D-homo-(16-en)-11(beta)-aryl-4-estrene |
| SK287192B6 (sk) | 1999-08-31 | 2010-02-08 | Bayer Schering Pharma Aktiengesellschaft | Mezoprogestíny (modulátory receptora pre progesterón) na liečenie a prevenciu benígnych gynekologických ochorení závislých od hormónov |
| RS52149B (sr) * | 2000-01-18 | 2012-08-31 | Bayer Schering Pharma Aktiengesellschaft | Farmaceutska kombinacija mikronizovanog drospirenona i estrogena za terapiju zamene hormona |
| EP1535618A1 (en) * | 2003-11-26 | 2005-06-01 | Schering Aktiengesellschaft | Pharmaceutical preparation for continuous hormonal treatment over a period of longer than 21-28 days comprising two estrogen and/or progestin compositions |
| MY151322A (en) * | 2004-04-30 | 2014-05-15 | Bayer Ip Gmbh | Management of breakthrough bleeding in extended hormonal contraceptive regimens |
| FR2886151B1 (fr) * | 2005-05-31 | 2007-09-07 | Mayoly Spindler Soc Par Action | Utilisation de la colchicine pour la preparation d'un medicament destine a la prevention et/ou au traitement de l'endometriose |
-
2007
- 2007-03-02 DE DE102007011105A patent/DE102007011105A1/de not_active Withdrawn
-
2008
- 2008-02-28 JP JP2009551220A patent/JP2010520178A/ja active Pending
- 2008-02-28 KR KR1020097018145A patent/KR20090119870A/ko not_active Ceased
- 2008-02-28 CN CN200880006913A patent/CN101621995A/zh active Pending
- 2008-02-28 AU AU2008223859A patent/AU2008223859A1/en not_active Abandoned
- 2008-02-28 CA CA002679520A patent/CA2679520A1/en not_active Abandoned
- 2008-02-28 RU RU2009136305/15A patent/RU2009136305A/ru not_active Application Discontinuation
- 2008-02-28 EP EP08717238A patent/EP2131825A1/de not_active Withdrawn
- 2008-02-28 US US12/529,447 patent/US20110003778A1/en not_active Abandoned
- 2008-02-28 BR BRPI0808427-0A patent/BRPI0808427A2/pt not_active IP Right Cessation
- 2008-02-28 MX MX2009009332A patent/MX2009009332A/es active IP Right Grant
- 2008-02-28 WO PCT/EP2008/052456 patent/WO2008107373A1/de not_active Ceased
- 2008-02-29 TW TW097107235A patent/TW200900080A/zh unknown
- 2008-03-03 AR ARP080100887A patent/AR065585A1/es unknown
-
2009
- 2009-08-13 IL IL200380A patent/IL200380A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN101621995A (zh) | 2010-01-06 |
| DE102007011105A1 (de) | 2008-09-04 |
| AR065585A1 (es) | 2009-06-17 |
| EP2131825A1 (de) | 2009-12-16 |
| AU2008223859A1 (en) | 2008-09-12 |
| IL200380A0 (en) | 2010-04-29 |
| TW200900080A (en) | 2009-01-01 |
| JP2010520178A (ja) | 2010-06-10 |
| KR20090119870A (ko) | 2009-11-20 |
| US20110003778A1 (en) | 2011-01-06 |
| RU2009136305A (ru) | 2011-04-10 |
| CA2679520A1 (en) | 2008-09-12 |
| BRPI0808427A2 (pt) | 2014-07-22 |
| WO2008107373A1 (de) | 2008-09-12 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant or registration | ||
| GB | Transfer or rights | ||
| HC | Change of company name or juridical status |