AR065585A1 - Antagonistas del receptor de mineralocorticoides para el tratamiento de endometriosis uso - Google Patents
Antagonistas del receptor de mineralocorticoides para el tratamiento de endometriosis usoInfo
- Publication number
- AR065585A1 AR065585A1 ARP080100887A ARP080100887A AR065585A1 AR 065585 A1 AR065585 A1 AR 065585A1 AR P080100887 A ARP080100887 A AR P080100887A AR P080100887 A ARP080100887 A AR P080100887A AR 065585 A1 AR065585 A1 AR 065585A1
- Authority
- AR
- Argentina
- Prior art keywords
- endometriosis
- treatment
- antagonists
- estrogen
- receptor antagonists
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
- A61K31/585—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Oncology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Steroid Compounds (AREA)
Abstract
Uso de antagonistas del receptor de mineralocorticoides para preparar un medicamento para el tratamiento de endometriosis. En especial, la presente se refiere a un agente terapéutico mejorado contra la endometriosis, que muestra un perfil de acciono de efectos colaterales más ventajoso que las terapias de tratamiento disponibles hasta ahora. Con un antagonista del receptor de mineralocorticoides se puede tratar la endometriosis de modo duradero, sin que se produzca, en este caso, una pérdidade la masa osea. Reivindicacion 4: Uso de espironolactona de acuerdo con la reivindicacion 1, 2 o 3. Reivindicacion 8: Uso de antagonistas del receptor de mineralocorticoides de acuerdo con una de las reivindicaciones 1 a 7 junto con al menos uncompuesto del grupo de los gestágenos, los SERM (Selective Estrogen Receptor Modulators), los SPRM (Selective Progesterone Receptor Modulators), combinaciones de gestágenos y estrogenos, antagonistas del receptor de progesterona, antagonistas delreceptor de estrogenos, glucocorticoides, ligandos específicos del isotipo del receptor de estrogenos (ligandos ER-beta), androgenos, antiandrogenos y los SARM (Selective Androgen Receptor Modulators). Reivindicacion 14: Uso de etinilestradiolcomo estrogeno de acuerdo con la reivindicacion 13.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102007011105A DE102007011105A1 (de) | 2007-03-02 | 2007-03-02 | Mineralcorticoid-Rezeptor-Antagonisten zur Behandlung von Endometriose |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR065585A1 true AR065585A1 (es) | 2009-06-17 |
Family
ID=39431148
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP080100887A AR065585A1 (es) | 2007-03-02 | 2008-03-03 | Antagonistas del receptor de mineralocorticoides para el tratamiento de endometriosis uso |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20110003778A1 (es) |
| EP (1) | EP2131825A1 (es) |
| JP (1) | JP2010520178A (es) |
| KR (1) | KR20090119870A (es) |
| CN (1) | CN101621995A (es) |
| AR (1) | AR065585A1 (es) |
| AU (1) | AU2008223859A1 (es) |
| BR (1) | BRPI0808427A2 (es) |
| CA (1) | CA2679520A1 (es) |
| DE (1) | DE102007011105A1 (es) |
| IL (1) | IL200380A0 (es) |
| MX (1) | MX2009009332A (es) |
| RU (1) | RU2009136305A (es) |
| TW (1) | TW200900080A (es) |
| WO (1) | WO2008107373A1 (es) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI1003661A2 (pt) * | 2010-09-15 | 2013-01-08 | Libbs Farmaceutica Ltda | associaÇço farmacÊutica para tratar e/ou prevenir mioma e/ou endometriose, uso de resveratrol e progestogenio, composiÇço farmacÊutica para tratamento e/ou prevenÇço de mioma e/ou endometriose medicamento para tratamento e/ou prevenÇço de mioma e/ou endometrios, kit e mÉtodo para tratamento e/ou prevenÇço de mioma e/ou endometriose |
| CN103957921A (zh) | 2011-11-04 | 2014-07-30 | 拜耳医药股份有限公司 | 18-甲基-6,7-亚甲基-3-氧代-17-孕甾-4-烯-21,17β-碳内酯、包含所述化合物的药物制剂及其在治疗子宫内膜异位症中的用途 |
| TW201350122A (zh) * | 2012-04-23 | 2013-12-16 | Bayer Pharma AG | 18-甲基-15β,16β-亞甲基-19-降-20-螺氧-4-烯-3-酮的子宮內用途,包含18-甲基-15β,16β-亞甲基-19-降-20-螺氧-4-烯-3-酮的子宮內系統,及其於避孕及婦科治療之用途 |
| UA115576C2 (uk) | 2012-12-06 | 2017-11-27 | Байєр Фарма Акцієнгезелльшафт | Похідні бензимідазолу як антагоністи ер4 |
| WO2014115449A1 (ja) * | 2013-01-22 | 2014-07-31 | シャープ株式会社 | 液晶表示装置 |
| TW201607943A (zh) | 2013-12-19 | 2016-03-01 | 拜耳製藥公司 | 作為ep4配體之新穎苯并咪唑衍生物 |
| CN117959293B (zh) * | 2024-01-18 | 2025-05-13 | 香港大学深圳医院 | 非奈利酮在制备治疗和/或预防卵巢功能障碍疾病药物中的应用 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4042004A1 (de) * | 1990-12-22 | 1992-06-25 | Schering Ag | 14(beta)-h-, 14- u. 15-en-11(beta)-aryl-4-estrene |
| DE4042005A1 (de) * | 1990-12-22 | 1992-06-25 | Schering Ag | D-homo-(16-en)-11(beta)-aryl-4-estrene |
| PT1229906E (pt) | 1999-08-31 | 2008-01-18 | Bayer Schering Pharma Ag | Mesoprogestinas para o tratamento e prevenção de distúrbios ginecológicos hormonodependentes benignos |
| SI1611892T1 (sl) | 2000-01-18 | 2010-01-29 | Bayer Schering Pharma Ag | Farmacevtski sestavki, ki obsegajo drospirenon |
| EP1535618A1 (en) * | 2003-11-26 | 2005-06-01 | Schering Aktiengesellschaft | Pharmaceutical preparation for continuous hormonal treatment over a period of longer than 21-28 days comprising two estrogen and/or progestin compositions |
| MY151322A (en) * | 2004-04-30 | 2014-05-15 | Bayer Ip Gmbh | Management of breakthrough bleeding in extended hormonal contraceptive regimens |
| FR2886151B1 (fr) * | 2005-05-31 | 2007-09-07 | Mayoly Spindler Soc Par Action | Utilisation de la colchicine pour la preparation d'un medicament destine a la prevention et/ou au traitement de l'endometriose |
-
2007
- 2007-03-02 DE DE102007011105A patent/DE102007011105A1/de not_active Withdrawn
-
2008
- 2008-02-28 KR KR1020097018145A patent/KR20090119870A/ko not_active Ceased
- 2008-02-28 CN CN200880006913A patent/CN101621995A/zh active Pending
- 2008-02-28 US US12/529,447 patent/US20110003778A1/en not_active Abandoned
- 2008-02-28 WO PCT/EP2008/052456 patent/WO2008107373A1/de not_active Ceased
- 2008-02-28 BR BRPI0808427-0A patent/BRPI0808427A2/pt not_active IP Right Cessation
- 2008-02-28 MX MX2009009332A patent/MX2009009332A/es active IP Right Grant
- 2008-02-28 EP EP08717238A patent/EP2131825A1/de not_active Withdrawn
- 2008-02-28 RU RU2009136305/15A patent/RU2009136305A/ru not_active Application Discontinuation
- 2008-02-28 JP JP2009551220A patent/JP2010520178A/ja active Pending
- 2008-02-28 CA CA002679520A patent/CA2679520A1/en not_active Abandoned
- 2008-02-28 AU AU2008223859A patent/AU2008223859A1/en not_active Abandoned
- 2008-02-29 TW TW097107235A patent/TW200900080A/zh unknown
- 2008-03-03 AR ARP080100887A patent/AR065585A1/es unknown
-
2009
- 2009-08-13 IL IL200380A patent/IL200380A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| RU2009136305A (ru) | 2011-04-10 |
| JP2010520178A (ja) | 2010-06-10 |
| KR20090119870A (ko) | 2009-11-20 |
| TW200900080A (en) | 2009-01-01 |
| US20110003778A1 (en) | 2011-01-06 |
| BRPI0808427A2 (pt) | 2014-07-22 |
| CN101621995A (zh) | 2010-01-06 |
| DE102007011105A1 (de) | 2008-09-04 |
| AU2008223859A1 (en) | 2008-09-12 |
| CA2679520A1 (en) | 2008-09-12 |
| EP2131825A1 (de) | 2009-12-16 |
| MX2009009332A (es) | 2009-09-11 |
| IL200380A0 (en) | 2010-04-29 |
| WO2008107373A1 (de) | 2008-09-12 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AR065585A1 (es) | Antagonistas del receptor de mineralocorticoides para el tratamiento de endometriosis uso | |
| BR112012014059A2 (pt) | gel transdérmico de progestina / estradiol. | |
| BR112014031910A2 (pt) | formulações e terapias naturais de combinação para reposição hormonal | |
| AR082998A1 (es) | Asociacion farmaceutica para tratar y/o prevenir mioma y/o endometriosis, uso de resveratrol y progestogeno, composicion farmaceutica para tratamiento y/o prevencion de mioma y/o endometriosis, medicamento para tratamiento y/o prevencion de mioma y/o endometriosis, kit y metodo para tratamiento y/o prevencion de mioma y/o endometriosis | |
| WO2013078422A3 (en) | Natural combination hormone replacement formulations and therapies | |
| IL149448A0 (en) | New topical estrogen-progestogen compositions with a systemic effect | |
| ECSP077131A (es) | Regímenes y los juegos de anticonceptivos del antagonista del receptor de progesterona | |
| CL2008001721A1 (es) | Compuestos derivados de 17-beta-ciano-18 alfa-homo-19-nor-androst-4-eno; que presentan actividad gestagena y antimineralcorticoide; composicion farmaceutica; y uso en el tratamiento de trastornos pre-peri-y posmenopausicos y trastornos premenstruales. | |
| TW200605882A (en) | Progesterone receptor modulators comprising pyrrole-oxindole derivatives and uses thereof | |
| MX347890B (es) | Neuroproteccion y reparacion de melina usando progestina. | |
| SI2148681T1 (sl) | Selektivni modulatorji progesterona v zdravljenju maternične krvavitve | |
| PE20211588A1 (es) | Compuestos y sus usos para aliviar sintomas asociados a la menopausia | |
| CR8529A (es) | Nueva forma cristalina v de la agomelatina, su procedimiento de preparacion y las composiciones farmaceuticas que la contiene | |
| CL2009001011A1 (es) | Uso del compuesto 21-metoxi-17a-acetoxi-11ß-(4-n,n-dimetilaminofenil)-19-norpregna-4,9-dien-3,20-diona (cdb-4124) para tratar el cancer de mama; y uso de la combinacion de cdb-4124 con un inhibidor de aromatasa. | |
| MX2016014281A (es) | Formulaciones y terapias de reemplazo de combinación de hormonas naturales. | |
| EP3462875A4 (en) | COMPOSITIONS AND METHODS WITH THE ANDERSTENONE, TESTOSTERONE, PROGESTERONE AND ESTROGEN PHEROMONIC COMPOUNDS | |
| AR080544A1 (es) | Mezclador de cemento oseo | |
| Nowak et al. | Potential operators associated with Jacobi and Fourier–Bessel expansions | |
| CL2008000999A1 (es) | Composicion farmaceutica que comprende drospirenona y 17beta estradiol; kit farmaceutico que comprende a dicha composicion, util para terapia hormonal y contracepcion en mujeres. | |
| HK1204287A1 (en) | Transdermal hormone delivery | |
| AR096464A1 (es) | Extracto de curcuma mangga val et. zipp. como un tratamiento para superar problemas prostáticos | |
| ECSP109872A (es) | Estratrienos 8-beta-sustituidos como estrógenos de acción selectiva | |
| AR070302A1 (es) | Composicion farmaceutica de un sistema de liberacion vaginal de esteroides | |
| UA99259C2 (ru) | Лечение ожирения антагонистами мускаринового рецептора м1 | |
| CL2003001545A1 (es) | Compuestos derivados de 7,9-difluoro-5h-cromeno-[3,4-f]quinolina de formula i, moduladores selectivos del receptor de progesterona; composicion farmaceutica; y su uso en el tratamiento de sangrado uterino disfuncional, dismenorrea, endometriosis, lei |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |