MX2009000152A - Derivados de azaindol con una combinacion de agonismo parcial del receptor nicotinico acetilcolina e inhibicion de la reabsorcion de dopamina. - Google Patents

Derivados de azaindol con una combinacion de agonismo parcial del receptor nicotinico acetilcolina e inhibicion de la reabsorcion de dopamina.

Info

Publication number: MX2009000152A
Authority: MX; Mexico
Prior art keywords: pyrrolo; pyridine; pyrrolidin; proviso; compound
Prior art date: 2006-07-06

Application number

MX2009000152A

Other languages

English (en)

Spanish (es)

Inventor

Cornelis G Kruse

Axel Stoit

Hein K A C Coolen

Neut Martina A W Van Der

Original Assignee

Solvay Pharm Bv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-07-06

Filing date

2007-07-05

Publication date

2009-03-25

2007-07-05 Application filed by Solvay Pharm Bv filed Critical Solvay Pharm Bv

2007-07-05 Priority claimed from PCT/EP2007/056792 external-priority patent/WO2008003736A1/en

2009-03-25 Publication of MX2009000152A publication Critical patent/MX2009000152A/es

Links

102000019315 Nicotinic acetylcholine receptors Human genes 0.000 title abstract description 26
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230000036961 partial effect Effects 0.000 title abstract description 8
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125000005334 azaindolyl group Chemical class N1N=C(C2=CC=CC=C12)* 0.000 title abstract description 4
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238000002424 x-ray crystallography Methods 0.000 description 1

Landscapes

Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

MX2009000152A 2006-07-06 2007-07-05 Derivados de azaindol con una combinacion de agonismo parcial del receptor nicotinico acetilcolina e inhibicion de la reabsorcion de dopamina. MX2009000152A (es)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP06116690		2006-07-06
PCT/EP2007/056792 WO2008003736A1 (en)	2006-07-06	2007-07-05	Azaindole derivatives with a combination of partial nicotinic acetylcholine receptor agonism and dopamine reuptake inhibition

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CN (1)	CN101484454A (zh)
AR (1)	AR061808A1 (zh)
MX (1)	MX2009000152A (zh)
SA (1)	SA07280361B1 (zh)
TW (1)	TW200819448A (zh)
UA (1)	UA97374C2 (zh)

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GB201320905D0 (en)	2013-11-27	2014-01-08	Takeda Pharmaceutical	Therapeutic compounds
CN111171019A (zh) *	2018-11-13	2020-05-19	上海轶诺药业有限公司	一类五元并六元杂环化合物及其作为蛋白受体激酶抑制剂的用途

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- 2007-07-03 AR ARP070102976 patent/AR061808A1/es not_active Application Discontinuation
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UA97374C2 (ru)	2012-02-10
TW200819448A (en)	2008-05-01
CN101484454A (zh)	2009-07-15
SA07280361B1 (ar)	2011-05-04
AR061808A1 (es)	2008-09-24

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MX2009000152A (es)	2009-03-25	Derivados de azaindol con una combinacion de agonismo parcial del receptor nicotinico acetilcolina e inhibicion de la reabsorcion de dopamina.
TW202345794A (zh)	2023-12-01	依莫帕米結合蛋白抑制劑及其用途
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