MA28363A1 - Antagonistes des recepteurs muscariniques de l'acetylcholine - Google Patents
Antagonistes des recepteurs muscariniques de l'acetylcholineInfo
- Publication number
- MA28363A1 MA28363A1 MA29273A MA29273A MA28363A1 MA 28363 A1 MA28363 A1 MA 28363A1 MA 29273 A MA29273 A MA 29273A MA 29273 A MA29273 A MA 29273A MA 28363 A1 MA28363 A1 MA 28363A1
- Authority
- MA
- Morocco
- Prior art keywords
- antagonists
- acetylcholine receptors
- muscarinic acetylcholine
- muscarinic
- receptors
- Prior art date
Links
- 102000014415 Muscarinic acetylcholine receptor Human genes 0.000 title 1
- 108050003473 Muscarinic acetylcholine receptor Proteins 0.000 title 1
- 239000005557 antagonist Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
- C07D451/06—Oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US53609204P | 2004-01-13 | 2004-01-13 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA28363A1 true MA28363A1 (fr) | 2006-12-01 |
Family
ID=34794385
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA29273A MA28363A1 (fr) | 2004-01-13 | 2006-08-15 | Antagonistes des recepteurs muscariniques de l'acetylcholine |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20080249127A1 (fr) |
| EP (1) | EP1711183A4 (fr) |
| JP (1) | JP2007518740A (fr) |
| KR (1) | KR20060129017A (fr) |
| CN (1) | CN1929844A (fr) |
| AR (1) | AR049464A1 (fr) |
| AU (1) | AU2005204935A1 (fr) |
| BR (1) | BRPI0506777A (fr) |
| CA (1) | CA2552880A1 (fr) |
| IL (1) | IL176775A0 (fr) |
| MA (1) | MA28363A1 (fr) |
| NO (1) | NO20063636L (fr) |
| PE (1) | PE20050898A1 (fr) |
| RU (1) | RU2006129289A (fr) |
| TW (1) | TW200534855A (fr) |
| WO (1) | WO2005067537A2 (fr) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20090253908A1 (en) * | 2004-03-11 | 2009-10-08 | Glaxo Group Limited | Novel m3 muscarinic acetylchoine receptor antagonists |
| PE20060259A1 (es) | 2004-04-27 | 2006-03-25 | Glaxo Group Ltd | Compuestos de quinuclidina como antagonistas del receptor de acetilcolina muscarinico |
| JP2007537261A (ja) * | 2004-05-13 | 2007-12-20 | グラクソ グループ リミテッド | ムスカリン性アセチルコリン受容体アンタゴニスト |
| EP1765339A4 (fr) * | 2004-06-30 | 2009-09-02 | Glaxo Group Ltd | Antagonistes du recepteur muscarinique d'acetylcholine |
| US7932247B2 (en) * | 2004-11-15 | 2011-04-26 | Glaxo Group Limited | M3 muscarinic acetylcholine receptor antagonists |
| JP2008537931A (ja) | 2005-03-10 | 2008-10-02 | セラヴァンス, インコーポレーテッド | ムスカリン性レセプターアンタゴニストとして有用なビフェニル化合物 |
| US20090012116A1 (en) * | 2005-07-11 | 2009-01-08 | Naresh Kumar | Muscarinic Receptor Antagonists |
| UY31637A1 (es) | 2008-02-06 | 2009-08-03 | Farmacoforos duales-antagonistas muscarinicos de pde4 | |
| UY31636A1 (es) | 2008-02-06 | 2009-08-03 | Farmacoforos duales-antagonistas muscarinicos de pde4 | |
| AR070564A1 (es) | 2008-02-06 | 2010-04-21 | Glaxo Group Ltd | Derivados de 1h-pirazolo[3,4-b]piridin-5-ilo,inhibidores de fosfodiesterasas pde4 y antagonistas de receptores muscarinicos de acetilcolina(machr), utiles en el tratamiento y/o profilaxis de enfermedades respiratorias y alergicas,y composiciones farmaceuticas que los comprenden |
| WO2010094643A1 (fr) | 2009-02-17 | 2010-08-26 | Glaxo Group Limited | Dérivés de quinoline et applications associées dans la rhinite et l'urticaire |
| AU2010242646A1 (en) * | 2009-04-30 | 2011-11-03 | Teijin Pharma Limited | Quaternary ammonium salt compound |
| WO2014023325A1 (fr) * | 2012-08-06 | 2014-02-13 | Fondazione Istituto Italiano Di Tecnologia | Inhibiteurs de faah et de cox multicibles et leurs utilisations thérapeutiques |
| KR101538846B1 (ko) * | 2013-07-30 | 2015-07-22 | 동아에스티 주식회사 | 신규한 바이페닐 유도체 및 그의 제조방법 |
| KR102239776B1 (ko) * | 2016-08-26 | 2021-04-13 | 동아에스티 주식회사 | (r)-(1-메틸피롤리딘-3-일)메틸(3'-클로로-4'-플루오로-[1,1'-비페닐]-2-일)카바메이트의 신규염 및 이의 결정형 |
| BR112019003949B1 (pt) | 2016-08-26 | 2023-12-12 | Dong-A St Co., Ltd | Sal de (r)-(1-metilpirrolidina-3-il)metil(3-cloro-4- fluoro-[1,1-bifenil] -2-il)carbamato inovador e uma forma cristalina dos mesmos |
| WO2019096226A1 (fr) | 2017-11-16 | 2019-05-23 | Chengdu Easton Biopharmaceuticals Co., Ltd. | Protéines de fusion vegfr/pdgfr pasylées et leur utilisation en thérapie |
| JP2021505569A (ja) * | 2017-12-04 | 2021-02-18 | フリードリヒ−アレクサンダー−ウニヴェルシテート エアランゲン−ニュルンベルク | M2よりもm3に対して選択性を有するフルオロフェニル置換ムスカリン受容体リガンド |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1140998B (it) * | 1980-06-18 | 1986-10-10 | Valeas Ind Chimica E Farmaceut | Sali di endo-8-metil-8-sin-alchil-8-azoniabiciclo aperta par. quadrata 3.2.1. chiusa par. quadrata-ottan-3-alchilcarbossilati, processo per la loro preparazione e composizioni terapeutiche che li contengono come principio attivo |
| EP0747355A4 (fr) * | 1994-02-10 | 1997-04-09 | Yamanouchi Pharma Co Ltd | Nouveau derive du carbamate et composition correspondante |
| US6846835B2 (en) * | 2000-07-11 | 2005-01-25 | Banyu Pharmaceutical Co., Ltd. | Ester derivatives |
| US7365167B2 (en) * | 2001-11-26 | 2008-04-29 | Cell Matrix, Inc. | Humanized collagen antibodies and related methods |
| MXPA04010966A (es) * | 2002-05-07 | 2005-01-25 | Neurosearch As | Derivados novedosos de biarilo diazabiciclico. |
| DE10255040A1 (de) * | 2002-11-26 | 2004-06-03 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Carbaminsäureester mit anticholinerger Wirksamkeit |
| US7041674B2 (en) * | 2002-11-26 | 2006-05-09 | Boehringer Ingelhiem Pharma Gmbh & Co. Kg | Carbamic acid esters with anticholinergic activity |
| EP1613307A4 (fr) * | 2003-04-07 | 2008-03-12 | Glaxo Group Ltd | Antagonistes du recepteur muscarinique m sb 3 /sb de l'acetylcholine |
-
2005
- 2005-01-11 TW TW094100746A patent/TW200534855A/zh unknown
- 2005-01-13 EP EP05711495A patent/EP1711183A4/fr not_active Withdrawn
- 2005-01-13 KR KR1020067016188A patent/KR20060129017A/ko not_active Withdrawn
- 2005-01-13 WO PCT/US2005/001333 patent/WO2005067537A2/fr not_active Ceased
- 2005-01-13 CN CNA2005800081262A patent/CN1929844A/zh active Pending
- 2005-01-13 BR BRPI0506777-4A patent/BRPI0506777A/pt not_active Application Discontinuation
- 2005-01-13 AR ARP050100118A patent/AR049464A1/es not_active Application Discontinuation
- 2005-01-13 US US10/585,830 patent/US20080249127A1/en not_active Abandoned
- 2005-01-13 CA CA002552880A patent/CA2552880A1/fr not_active Abandoned
- 2005-01-13 JP JP2006549649A patent/JP2007518740A/ja active Pending
- 2005-01-13 AU AU2005204935A patent/AU2005204935A1/en not_active Abandoned
- 2005-01-13 PE PE2005000059A patent/PE20050898A1/es not_active Application Discontinuation
- 2005-01-13 RU RU2006129289/04A patent/RU2006129289A/ru not_active Application Discontinuation
-
2006
- 2006-07-10 IL IL176775A patent/IL176775A0/en unknown
- 2006-08-11 NO NO20063636A patent/NO20063636L/no not_active Application Discontinuation
- 2006-08-15 MA MA29273A patent/MA28363A1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US20080249127A1 (en) | 2008-10-09 |
| CN1929844A (zh) | 2007-03-14 |
| AU2005204935A1 (en) | 2005-07-28 |
| EP1711183A2 (fr) | 2006-10-18 |
| RU2006129289A (ru) | 2008-02-20 |
| JP2007518740A (ja) | 2007-07-12 |
| WO2005067537A3 (fr) | 2006-05-18 |
| BRPI0506777A (pt) | 2007-05-22 |
| IL176775A0 (en) | 2006-10-31 |
| AR049464A1 (es) | 2006-08-09 |
| TW200534855A (en) | 2005-11-01 |
| PE20050898A1 (es) | 2005-11-06 |
| NO20063636L (no) | 2006-10-04 |
| EP1711183A4 (fr) | 2009-04-01 |
| KR20060129017A (ko) | 2006-12-14 |
| WO2005067537A2 (fr) | 2005-07-28 |
| CA2552880A1 (fr) | 2005-07-28 |
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