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UY30431A1 - Suspensiones acuosas de tmc278 - Google Patents

Suspensiones acuosas de tmc278

Info

Publication number
UY30431A1
UY30431A1 UY30431A UY30431A UY30431A1 UY 30431 A1 UY30431 A1 UY 30431A1 UY 30431 A UY30431 A UY 30431A UY 30431 A UY30431 A UY 30431A UY 30431 A1 UY30431 A1 UY 30431A1
Authority
UY
Uruguay
Prior art keywords
tmc278
pharmaceutical compositions
suspensions
waterproof
waterproof suspensions
Prior art date
Application number
UY30431A
Other languages
English (en)
Inventor
Peter Jozef Maria V Remoortere
Marc Carel Jozef Francois
Laurent Bruno Schueller
Willy Alber Maria Carlo Dries
Derivados De Benzoxazol Estruc
Original Assignee
Tibotec Pharm Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38833797&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY30431(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Tibotec Pharm Ltd filed Critical Tibotec Pharm Ltd
Publication of UY30431A1 publication Critical patent/UY30431A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Dermatology (AREA)
  • Inorganic Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Dispersion Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La presente invencion comprende composiciones farmacéuticas para la administracion por inyeccion intramuscular o subcutánea, que comprende micro o nanopartículas del compuesto NNRTI TMC278, suspendido en un portador acuoso farmacéuticamente aceptable, y el uso de dichas composiciones farmacéuticas en el tratamiento y la prevencion de infeccion por VIH.
UY30431A 2006-06-23 2007-06-22 Suspensiones acuosas de tmc278 UY30431A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP06115938 2006-06-23

Publications (1)

Publication Number Publication Date
UY30431A1 true UY30431A1 (es) 2008-01-31

Family

ID=38833797

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30431A UY30431A1 (es) 2006-06-23 2007-06-22 Suspensiones acuosas de tmc278

Country Status (33)

Country Link
US (4) US20090176813A1 (es)
EP (2) EP2040671B1 (es)
JP (1) JP5292288B2 (es)
KR (1) KR101406879B1 (es)
CN (1) CN101478950B (es)
AP (1) AP2618A (es)
AR (1) AR061620A1 (es)
AU (1) AU2007262941B2 (es)
BR (2) BRPI0713334B1 (es)
CA (1) CA2654115C (es)
CL (1) CL2007001847A1 (es)
CY (1) CY1120564T1 (es)
DK (2) DK2040671T3 (es)
EA (1) EA021700B1 (es)
ES (2) ES2989051T3 (es)
FI (1) FI3366278T3 (es)
HR (2) HRP20241265T3 (es)
HU (2) HUE038797T2 (es)
IL (1) IL195491A (es)
JO (1) JOP20200160A1 (es)
LT (2) LT2040671T (es)
MX (1) MX2009000158A (es)
NZ (1) NZ573291A (es)
PE (1) PE20080210A1 (es)
PL (2) PL3366278T3 (es)
PT (2) PT3366278T (es)
RS (2) RS65990B1 (es)
SG (1) SG173315A1 (es)
SI (2) SI3366278T1 (es)
TW (1) TWI413521B (es)
UA (1) UA97641C2 (es)
UY (1) UY30431A1 (es)
WO (1) WO2007147882A2 (es)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY169670A (en) 2003-09-03 2019-05-08 Tibotec Pharm Ltd Combinations of a pyrimidine containing nnrti with rt inhibitors
TWI457136B (zh) * 2005-04-04 2014-10-21 Tibotec Pharm Ltd Hiv-感染之預防
JP5754005B2 (ja) 2006-01-20 2015-07-22 ヤンセン・アールアンドデイ・アイルランド Tcm278を用いるhiv−感染症の長期間処置
TWI494133B (zh) 2007-03-14 2015-08-01 Tibotec Pharm Ltd 重組用粉末
EP2306980A2 (en) * 2008-06-30 2011-04-13 Tibotec Pharmaceuticals Powders for reconstitution
ES2607107T3 (es) * 2008-12-24 2017-03-29 Janssen Sciences Ireland Uc Dispositivos implantables para tratar el VIH
TWI577377B (zh) 2010-09-16 2017-04-11 Viiv醫療保健公司 醫藥組合物
HRP20201241T1 (hr) * 2011-04-15 2020-11-27 Janssen Pharmaceutica N.V. Nanosuspenzije lijeka osušene zamrzavanjem
JO3387B1 (ar) 2011-12-16 2019-03-13 Glaxosmithkline Llc مشتقات بيتولين
HK1209638A1 (en) 2012-12-14 2016-04-08 Glaxosmithkline Llc Pharmaceutical compositions
BR112017006005A2 (pt) 2014-09-26 2017-12-19 Glaxosmithkline Ip No 2 Ltd composição farmacêutica, e, método de prevenção ou tratamento de uma infecção por hiv.
US10369129B2 (en) * 2016-05-31 2019-08-06 Taimed Biologics, Inc. Long acting pharmaceutical composition of protease inhibitor
TWI678203B (zh) * 2016-05-31 2019-12-01 中裕新藥股份有限公司 蛋白酶抑制劑之長效醫藥組合物
CN109475563A (zh) * 2016-05-31 2019-03-15 中裕新药股份有限公司 蛋白酶抑制剂的长效医药组合物
CN110191704A (zh) 2016-10-24 2019-08-30 爱尔兰詹森科学公司 可分散组合物
AU2018298855B2 (en) * 2017-07-14 2024-07-18 Janssen Pharmaceutica Nv Long-acting formulations
CN113440529B (zh) * 2020-03-25 2023-11-14 江苏恒瑞医药股份有限公司 一种可注射的药物组合物及其制备方法
MX2023000439A (es) 2020-07-09 2023-02-09 Janssen Pharmaceutica Nv Formulaciones a largo plazo.
JP2023532981A (ja) 2020-07-09 2023-08-01 ヤンセン ファーマシューティカ エヌ.ベー. 長時間作用型配合物
JP2023532982A (ja) 2020-07-09 2023-08-01 ヤンセン ファーマシューティカ エヌ.ベー. 長時間作用型配合物
KR20230110763A (ko) * 2020-11-17 2023-07-25 얀센 사이언시즈 아일랜드 언리미티드 컴퍼니 질환 또는 장애의 치료 또는 예방
TW202233192A (zh) 2020-11-17 2022-09-01 愛爾蘭商健生科學愛爾蘭無限公司 Hiv感染之治療或預防
KR20240095514A (ko) 2021-11-17 2024-06-25 얀센 사이언시즈 아일랜드 언리미티드 컴퍼니 용해도 평가
CN119403543A (zh) 2022-04-22 2025-02-07 爱尔兰詹森科学公司 液体组合物
CN119403545A (zh) 2022-04-22 2025-02-07 爱尔兰詹森科学公司 冷冻干燥的组合物
TW202408526A (zh) 2022-05-17 2024-03-01 愛爾蘭商健生科學愛爾蘭無限公司 治療或預防hiv感染(一)
TW202408527A (zh) 2022-05-17 2024-03-01 愛爾蘭商健生科學愛爾蘭無限公司 治療或預防hiv感染(二)
CA3268292A1 (en) 2022-09-28 2024-04-04 Janssen Pharmaceutica Nv LONG-ACTING FORMULAS
WO2024068693A1 (en) 2022-09-28 2024-04-04 Janssen Pharmaceutica Nv Long-acting formulations
WO2025054693A1 (pt) * 2023-09-14 2025-03-20 Instituto Hercílio Randon Premix funcional de nanopartículas, processo para sua obtenção, processo para modificação de propriedades de materiais e material com propriedades modificadas

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TWI457136B (zh) * 2005-04-04 2014-10-21 Tibotec Pharm Ltd Hiv-感染之預防
JP5754005B2 (ja) * 2006-01-20 2015-07-22 ヤンセン・アールアンドデイ・アイルランド Tcm278を用いるhiv−感染症の長期間処置

Also Published As

Publication number Publication date
HRP20241265T3 (hr) 2024-12-06
US11389447B2 (en) 2022-07-19
CA2654115A1 (en) 2007-12-27
DK2040671T3 (en) 2018-05-07
BRPI0713334A2 (pt) 2012-03-06
HRP20180629T1 (hr) 2018-06-01
RS65990B1 (sr) 2024-10-31
JP5292288B2 (ja) 2013-09-18
HUE038797T2 (hu) 2018-11-28
SI3366278T1 (sl) 2024-12-31
WO2007147882A3 (en) 2008-06-19
ES2989051T3 (es) 2024-11-25
RS57111B1 (sr) 2018-06-29
JOP20200160A1 (ar) 2022-10-30
ES2662068T3 (es) 2018-04-05
PL2040671T3 (pl) 2018-08-31
DK3366278T3 (da) 2024-09-23
MX2009000158A (es) 2009-01-23
TWI413521B (zh) 2013-11-01
IL195491A0 (en) 2009-09-01
KR101406879B1 (ko) 2014-06-13
WO2007147882A2 (en) 2007-12-27
EA021700B1 (ru) 2015-08-31
TW200817008A (en) 2008-04-16
UA97641C2 (en) 2012-03-12
HUE068406T2 (hu) 2024-12-28
EP2040671A2 (en) 2009-04-01
BR122020011487B1 (pt) 2024-02-20
US20150010637A1 (en) 2015-01-08
CN101478950B (zh) 2013-02-06
LT3366278T (lt) 2024-11-11
AR061620A1 (es) 2008-09-10
JP2009541271A (ja) 2009-11-26
EP3366278B1 (en) 2024-08-07
EP3366278A1 (en) 2018-08-29
EA200970047A1 (ru) 2009-04-28
CA2654115C (en) 2015-12-22
LT2040671T (lt) 2018-05-10
CY1120564T1 (el) 2019-07-10
AP2618A (en) 2013-03-18
CN101478950A (zh) 2009-07-08
AP2008004682A0 (en) 2008-12-31
PL3366278T3 (pl) 2024-10-28
CL2007001847A1 (es) 2008-02-08
US20220273653A1 (en) 2022-09-01
KR20090023703A (ko) 2009-03-05
IL195491A (en) 2014-11-30
FI3366278T3 (fi) 2024-09-25
NZ573291A (en) 2011-11-25
PE20080210A1 (es) 2008-04-11
AU2007262941B2 (en) 2013-11-21
PT3366278T (pt) 2024-10-21
SG173315A1 (en) 2011-08-29
BRPI0713334A8 (pt) 2018-01-02
BRPI0713334B1 (pt) 2024-02-20
AU2007262941A1 (en) 2007-12-27
PT2040671T (pt) 2018-03-14
SI2040671T1 (en) 2018-05-31
US20090176813A1 (en) 2009-07-09
US20160089369A1 (en) 2016-03-31
EP2040671B1 (en) 2018-01-24

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