AR077138A1 - Composiciones farmaceuticas utiles para tratar el vhc - Google Patents
Composiciones farmaceuticas utiles para tratar el vhcInfo
- Publication number
- AR077138A1 AR077138A1 ARP100102159A ARP100102159A AR077138A1 AR 077138 A1 AR077138 A1 AR 077138A1 AR P100102159 A ARP100102159 A AR P100102159A AR P100102159 A ARP100102159 A AR P100102159A AR 077138 A1 AR077138 A1 AR 077138A1
- Authority
- AR
- Argentina
- Prior art keywords
- compound
- composition
- pharmaceutical compositions
- compositions useful
- treat hcv
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 239000000203 mixture Substances 0.000 abstract 8
- 229940125904 compound 1 Drugs 0.000 abstract 5
- 229940125782 compound 2 Drugs 0.000 abstract 5
- 239000003814 drug Substances 0.000 abstract 1
- 208000015181 infectious disease Diseases 0.000 abstract 1
- 239000007788 liquid Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000008247 solid mixture Substances 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Virology (AREA)
- Oncology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Abstract
Reivindicacion 1: Una composicion que comprende el compuesto 1 y el compuesto 2, o sales o solvatos del compuesto 1 y del compuesto 2, en donde el compuesto 1 tiene la estructura que se muestra en la formula 1 y el compuesto 2 tiene la estructura que se muestra en la formula 2. Reivindicacion 2: La composicion de la reivindicacion 1 en donde el compuesto 1 está presente en una cantidad de 1 mg a 100 mg. Reivindicacion 4: La composicion de la reivindicacion 1 en donde el compuesto 2 está presente en una cantidad de 100 mg a 1200 mg. Reivindicacion 7: La composicion de la reivindicacion 1 en donde dicha composicion es una composicion solida. Reivindicacion 8: La composicion de la reivindicacion 1 en donde dicha composicion es una composicion líquida. Reivindicacion 18: El uso de la combinacion del compuesto 1 y del compuesto 2 en la fabricacion de un medicamento para el tratamiento de la infeccion por VHC en un ser humano.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US21964609P | 2009-06-23 | 2009-06-23 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR077138A1 true AR077138A1 (es) | 2011-08-03 |
Family
ID=42536374
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP100102159A AR077138A1 (es) | 2009-06-23 | 2010-06-18 | Composiciones farmaceuticas utiles para tratar el vhc |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20100324059A1 (es) |
| AR (1) | AR077138A1 (es) |
| TW (1) | TW201113279A (es) |
| UY (1) | UY32721A (es) |
| WO (1) | WO2010151487A1 (es) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20110075019A (ko) * | 2008-10-15 | 2011-07-05 | 인터뮨, 인크. | 치료용 항바이러스성 펩티드 |
| AR075584A1 (es) | 2009-02-27 | 2011-04-20 | Intermune Inc | COMPOSICIONES TERAPEUTICAS QUE COMPRENDEN beta-D-2'-DESOXI-2'-FLUORO-2'-C-METILCITIDINA Y UN DERIVADO DE ACIDO ISOINDOL CARBOXILICO Y SUS USOS. COMPUESTO. |
| CN102712644A (zh) * | 2009-09-28 | 2012-10-03 | 豪夫迈·罗氏有限公司 | 丙肝病毒复制的新型大环抑制剂 |
| WO2011041551A1 (en) * | 2009-10-01 | 2011-04-07 | Intermune, Inc. | Therapeutic antiviral peptides |
| WO2012009394A2 (en) * | 2010-07-16 | 2012-01-19 | Bristol-Myers Squibb Company | Methods to identify combinations of ns5a targeting compounds that act synergistically to inhibit hepatitis c virus replication |
| SG2014011647A (en) | 2011-10-21 | 2014-08-28 | Abbvie Inc | Methods for treating hcv comprising at least two direct acting antiviral agent, ribavirin but not interferon. |
| US8492386B2 (en) | 2011-10-21 | 2013-07-23 | Abbvie Inc. | Methods for treating HCV |
| SG2014011670A (en) | 2011-10-21 | 2014-10-30 | Abbvie Inc | Combination treatment (eg. with abt-072 or abt -333) of daas for use in treating hcv |
| US8466159B2 (en) | 2011-10-21 | 2013-06-18 | Abbvie Inc. | Methods for treating HCV |
| SG11201705069YA (en) | 2014-12-26 | 2017-07-28 | Univ Emory | N4-hydroxycytidine and derivatives and anti-viral uses related thereto |
| JP7129703B2 (ja) | 2016-04-28 | 2022-09-02 | エモリー ユニバーシティー | アルキン含有ヌクレオチド及びヌクレオシド治療組成物並びにそれらに関連した使用 |
| WO2019113462A1 (en) | 2017-12-07 | 2019-06-13 | Emory University | N4-hydroxycytidine and derivatives and anti-viral uses related thereto |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SV2003000617A (es) | 2000-08-31 | 2003-01-13 | Lilly Co Eli | Inhibidores de la proteasa peptidomimetica ref. x-14912m |
| US20070015553A1 (en) | 2005-07-12 | 2007-01-18 | Microsoft Corporation | Compact and durable clamshell smartphone |
| US20080008682A1 (en) * | 2006-07-07 | 2008-01-10 | Chong Lee S | Modulators of toll-like receptor 7 |
| ATE454384T1 (de) | 2006-07-07 | 2010-01-15 | Gilead Sciences Inc | Neue pyridazinverbindung und ihre verwendung |
| BRPI0813952A2 (pt) * | 2007-06-29 | 2017-05-09 | Gilead Sciences Inc | derivados de purina e seu emprego como moduladores e receptor 7 semelhante ao dobre de sino |
-
2010
- 2010-06-18 TW TW099119939A patent/TW201113279A/zh unknown
- 2010-06-18 AR ARP100102159A patent/AR077138A1/es unknown
- 2010-06-18 UY UY0001032721A patent/UY32721A/es not_active Application Discontinuation
- 2010-06-18 US US12/818,407 patent/US20100324059A1/en not_active Abandoned
- 2010-06-18 WO PCT/US2010/039134 patent/WO2010151487A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| UY32721A (es) | 2011-01-31 |
| WO2010151487A1 (en) | 2010-12-29 |
| US20100324059A1 (en) | 2010-12-23 |
| TW201113279A (en) | 2011-04-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |