UA92765C2 - Фармацевтическое средство для лечения уретеролитиаза - Google Patents
Фармацевтическое средство для лечения уретеролитиазаInfo
- Publication number
- UA92765C2 UA92765C2 UAA200808421A UAA200808421A UA92765C2 UA 92765 C2 UA92765 C2 UA 92765C2 UA A200808421 A UAA200808421 A UA A200808421A UA A200808421 A UAA200808421 A UA A200808421A UA 92765 C2 UA92765 C2 UA 92765C2
- Authority
- UA
- Ukraine
- Prior art keywords
- ureterolithiasis
- cyano
- substituent
- carbamoyl
- substituted
- Prior art date
Links
- 201000011086 ureterolithiasis Diseases 0.000 title abstract 3
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 3
- 125000004093 cyano group Chemical class *C#N 0.000 abstract 3
- 125000001424 substituent group Chemical group 0.000 abstract 3
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 210000000626 ureter Anatomy 0.000 abstract 2
- 230000001133 acceleration Effects 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
- 230000008602 contraction Effects 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000002768 hydroxyalkyl group Chemical group 0.000 abstract 1
- 125000003387 indolinyl group Chemical class N1(CCC2=CC=CC=C12)* 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 230000003389 potentiating effect Effects 0.000 abstract 1
- 125000005400 pyridylcarbonyl group Chemical group N1=C(C=CC=C1)C(=O)* 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/04—Drugs for disorders of the urinary system for urolithiasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Urology & Nephrology (AREA)
- Epidemiology (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
Abstract
Данное изобретение относится к фармацевтическим композициям, которые используются для облегчения боли, вызываемой камнями в мочеточниках, как средство, способствующее выделению камней мочеточников или т.п.Заявлена фармацевтическая композиция для лечения уретеролитиаза, которая включает как активный ингредиент производное индолина, представленное общей формулой (И), или его соль. В указанной формуле R представляет собой насыщенную или ненасыщенную алифатическую ацильную группу, которая может иметь заместитель; гидроксиалкилгруппу; алифатическую ацилоксиалкилгруппу; низшую алкилгруппу, которая содержит как заместитель низшую алкоксигруппу, карбо
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2005339188 | 2005-11-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA92765C2 true UA92765C2 (ru) | 2010-12-10 |
Family
ID=38067199
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200808421A UA92765C2 (ru) | 2005-11-24 | 2006-11-22 | Фармацевтическое средство для лечения уретеролитиаза |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US20090163571A1 (ru) |
| EP (1) | EP1956001A4 (ru) |
| JP (1) | JP4865724B2 (ru) |
| KR (1) | KR101232425B1 (ru) |
| CN (1) | CN101336230B (ru) |
| BR (1) | BRPI0618996A2 (ru) |
| CA (1) | CA2628476C (ru) |
| EA (1) | EA016008B1 (ru) |
| NO (1) | NO20082816L (ru) |
| TW (1) | TW200803843A (ru) |
| UA (1) | UA92765C2 (ru) |
| WO (1) | WO2007060974A1 (ru) |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2132254T3 (es) * | 1992-09-14 | 1999-08-16 | Forssmann Wolf Georg Prof Dr | Nueva utilizacion de inhibidores de la fosfodiesterasa iv. |
| EP0600675B1 (en) * | 1992-12-02 | 1998-07-08 | Kissei Pharmaceutical Co., Ltd. | Indoline compounds for the treatment of dysuria |
| JP4324266B2 (ja) * | 1999-02-26 | 2009-09-02 | キッセイ薬品工業株式会社 | α1Aアドレナリン受容体の変異体、当該変異体を用いた測定方法及び前立腺肥大に伴う排尿困難症治療剤 |
| KR100554813B1 (ko) * | 2001-01-02 | 2006-02-22 | 에프. 호프만-라 로슈 아게 | 알파 1에이/비 아드레날린성 수용체 길항제로서의퀴나졸론 유도체 |
| JP2001288115A (ja) * | 2001-02-07 | 2001-10-16 | Yamanouchi Pharmaceut Co Ltd | 下部尿路症治療剤 |
| US20040072551A1 (en) * | 2002-10-10 | 2004-04-15 | Sanford John Richard | Communication device with front-end integration |
-
2006
- 2006-11-22 UA UAA200808421A patent/UA92765C2/ru unknown
- 2006-11-22 CA CA2628476A patent/CA2628476C/en not_active Expired - Fee Related
- 2006-11-22 WO PCT/JP2006/323280 patent/WO2007060974A1/ja not_active Ceased
- 2006-11-22 KR KR1020087015259A patent/KR101232425B1/ko not_active Expired - Fee Related
- 2006-11-22 EP EP06823507A patent/EP1956001A4/en not_active Withdrawn
- 2006-11-22 CN CN2006800517242A patent/CN101336230B/zh not_active Expired - Fee Related
- 2006-11-22 BR BRPI0618996-2A patent/BRPI0618996A2/pt not_active IP Right Cessation
- 2006-11-22 JP JP2007546458A patent/JP4865724B2/ja not_active Expired - Fee Related
- 2006-11-22 US US12/093,230 patent/US20090163571A1/en not_active Abandoned
- 2006-11-22 EA EA200801420A patent/EA016008B1/ru not_active IP Right Cessation
- 2006-11-23 TW TW095143355A patent/TW200803843A/zh not_active IP Right Cessation
-
2008
- 2008-06-24 NO NO20082816A patent/NO20082816L/no not_active Application Discontinuation
-
2011
- 2011-04-13 US US13/086,040 patent/US20110230538A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| KR20080071603A (ko) | 2008-08-04 |
| CN101336230B (zh) | 2011-11-23 |
| JPWO2007060974A1 (ja) | 2009-05-07 |
| EA200801420A1 (ru) | 2009-02-27 |
| TW200803843A (en) | 2008-01-16 |
| BRPI0618996A2 (pt) | 2011-09-20 |
| HK1125634A1 (en) | 2009-08-14 |
| WO2007060974A1 (ja) | 2007-05-31 |
| JP4865724B2 (ja) | 2012-02-01 |
| CA2628476C (en) | 2013-10-15 |
| TWI379680B (ru) | 2012-12-21 |
| EA016008B1 (ru) | 2012-01-30 |
| EP1956001A4 (en) | 2012-12-26 |
| US20110230538A1 (en) | 2011-09-22 |
| US20090163571A1 (en) | 2009-06-25 |
| CA2628476A1 (en) | 2007-05-31 |
| EP1956001A1 (en) | 2008-08-13 |
| KR101232425B1 (ko) | 2013-02-12 |
| NO20082816L (no) | 2008-08-13 |
| CN101336230A (zh) | 2008-12-31 |
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