UA84737C2 - Производные имидазолина с антагонистической активностью относительно cb1 - Google Patents
Производные имидазолина с антагонистической активностью относительно cb1Info
- Publication number
- UA84737C2 UA84737C2 UAA200610009A UAA200610009A UA84737C2 UA 84737 C2 UA84737 C2 UA 84737C2 UA A200610009 A UAA200610009 A UA A200610009A UA A200610009 A UAA200610009 A UA A200610009A UA 84737 C2 UA84737 C2 UA 84737C2
- Authority
- UA
- Ukraine
- Prior art keywords
- imidazoline derivatives
- antagonistic activity
- compounds
- preparation
- methods
- Prior art date
Links
- 229940083254 peripheral vasodilators imidazoline derivative Drugs 0.000 title abstract 4
- 150000002462 imidazolines Chemical class 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000000543 intermediate Substances 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 abstract 2
- 238000002360 preparation method Methods 0.000 abstract 2
- -1 1,2,4-tri-substituted imidazoline Chemical class 0.000 abstract 1
- 208000012902 Nervous system disease Diseases 0.000 abstract 1
- 208000025966 Neurological disease Diseases 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 208000020016 psychiatric disease Diseases 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP04100656 | 2004-02-19 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA84737C2 true UA84737C2 (ru) | 2008-11-25 |
Family
ID=34928876
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200610009A UA84737C2 (ru) | 2004-02-19 | 2005-02-16 | Производные имидазолина с антагонистической активностью относительно cb1 |
Country Status (7)
| Country | Link |
|---|---|
| CN (1) | CN101076520B (zh) |
| AR (1) | AR047613A1 (zh) |
| BR (1) | BRPI0507269A (zh) |
| SA (1) | SA05260008B1 (zh) |
| TW (1) | TWI335321B (zh) |
| UA (1) | UA84737C2 (zh) |
| ZA (1) | ZA200606123B (zh) |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI231757B (en) * | 2001-09-21 | 2005-05-01 | Solvay Pharm Bv | 1H-Imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1-antagonistic activity |
| ES2272809T3 (es) * | 2001-09-21 | 2007-05-01 | Solvay Pharm Bv | Nuevos derivados de 4,5-dihidro-1h-pirazol con actividad antagonista de cb1. |
| AR038966A1 (es) * | 2002-03-18 | 2005-02-02 | Solvay Pharm Bv | Derivados de tiazol que tienen actividad antagonista, agonista o agonista parcial de cb1 |
| US6878735B2 (en) * | 2002-05-31 | 2005-04-12 | Board Of Trustees Of Michigan State University | Multi-substituted imidazolines and method of use thereof |
-
2005
- 2005-02-14 TW TW94104182A patent/TWI335321B/zh not_active IP Right Cessation
- 2005-02-14 AR ARP050100514 patent/AR047613A1/es not_active Application Discontinuation
- 2005-02-16 SA SA05260008A patent/SA05260008B1/ar unknown
- 2005-02-16 BR BRPI0507269-7A patent/BRPI0507269A/pt not_active IP Right Cessation
- 2005-02-16 CN CN2005800033771A patent/CN101076520B/zh not_active Expired - Fee Related
- 2005-02-16 UA UAA200610009A patent/UA84737C2/ru unknown
-
2006
- 2006-07-24 ZA ZA200606123A patent/ZA200606123B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AR047613A1 (es) | 2006-01-25 |
| CN101076520B (zh) | 2011-06-01 |
| SA05260008A (ar) | 2005-12-03 |
| TWI335321B (en) | 2011-01-01 |
| CN101076520A (zh) | 2007-11-21 |
| BRPI0507269A (pt) | 2007-06-26 |
| ZA200606123B (en) | 2007-11-28 |
| SA05260008B1 (ar) | 2007-10-29 |
| TW200530191A (en) | 2005-09-16 |
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