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SV2009003288A - Derivados de 2, 3-dihidroimidazo [1,2-c] quinazolina sustituidos de utilidad en el tratamiento de trastornos hiperproliferativos y enfermedades asociadas con la angiogenesis - Google Patents

Derivados de 2, 3-dihidroimidazo [1,2-c] quinazolina sustituidos de utilidad en el tratamiento de trastornos hiperproliferativos y enfermedades asociadas con la angiogenesis

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Publication number
SV2009003288A
SV2009003288A SV2009003288A SV2009003288A SV2009003288A SV 2009003288 A SV2009003288 A SV 2009003288A SV 2009003288 A SV2009003288 A SV 2009003288A SV 2009003288 A SV2009003288 A SV 2009003288A SV 2009003288 A SV2009003288 A SV 2009003288A
Authority
SV
El Salvador
Prior art keywords
treatment
dihydroimidazo
angiogenesis
hyperproliferative disorders
derivatives
Prior art date
Application number
SV2009003288A
Other languages
English (en)
Inventor
Martin F Hentemann
Jill Wood
William Scott
Martin Michels
Ann-Marie Campbell
R Bruce Rowley
Aniko Redman
Ann-Marie Bullion
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39492563&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SV2009003288(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of SV2009003288A publication Critical patent/SV2009003288A/es

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    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
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    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
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    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
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    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • AHUMAN NECESSITIES
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • CCHEMISTRY; METALLURGY
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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings

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Abstract

NUEVOS COMPUESTOS DE 2,3-DIHIDROIMIDAZO [1,2-C]QUINAZOLINA, CON COMPOSICIONES FARMACÉUTICAS QUE CONTIENEN A DICHOS COMPUESTOS Y CON EL USO DE DICHOS COMPUESTOS O COMPOSICIONES EN LA INHIBICIÓN Y EL TRATAMIENTO DE ENFERMEDADES ASOCIADAS CON LA ACTIVIDAD DE LA FOSFOTIDILINOSITOL-3-QUINASA (PI3K), EN PARTICULAR EN EL TRATAMIENTO DE TRASTORNOS HIPERPROLIFERATIVOS Y/O DE ANGIOGENESIS, COMO AGENTE ÚNICO O EN COMBINACIÓN CON OTROS INGREDIENTES ACTIVOS
SV2009003288A 2006-12-05 2009-06-05 Derivados de 2, 3-dihidroimidazo [1,2-c] quinazolina sustituidos de utilidad en el tratamiento de trastornos hiperproliferativos y enfermedades asociadas con la angiogenesis SV2009003288A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US87309006P 2006-12-05 2006-12-05

Publications (1)

Publication Number Publication Date
SV2009003288A true SV2009003288A (es) 2009-10-02

Family

ID=39492563

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2009003288A SV2009003288A (es) 2006-12-05 2009-06-05 Derivados de 2, 3-dihidroimidazo [1,2-c] quinazolina sustituidos de utilidad en el tratamiento de trastornos hiperproliferativos y enfermedades asociadas con la angiogenesis

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US (3) USRE46856E1 (es)
EP (1) EP2096919B1 (es)
JP (1) JP5326092B2 (es)
KR (1) KR101501785B1 (es)
CN (4) CN101631464B (es)
AR (1) AR064106A1 (es)
AU (1) AU2007328008B2 (es)
BR (1) BRPI0720178B8 (es)
CA (1) CA2671614C (es)
CL (1) CL2007003508A1 (es)
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CR (1) CR10838A (es)
CU (1) CU23796B7 (es)
DK (1) DK2096919T3 (es)
DO (1) DOP2009000135A (es)
EA (1) EA018839B1 (es)
EC (1) ECSP099387A (es)
ES (1) ES2572189T3 (es)
GT (1) GT200900154A (es)
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PA (1) PA8759601A1 (es)
PE (1) PE20081444A1 (es)
PL (1) PL2096919T3 (es)
RS (1) RS56045B1 (es)
SG (1) SG177170A1 (es)
SI (1) SI2096919T1 (es)
SV (1) SV2009003288A (es)
TN (1) TN2009000137A1 (es)
TW (1) TWI406662B (es)
UA (1) UA96965C2 (es)
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