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SMT201600321B - Composizione iniettabile a rilascio graduale antipsicotica - Google Patents

Composizione iniettabile a rilascio graduale antipsicotica

Info

Publication number
SMT201600321B
SMT201600321B SM201600321T SM201600321T SMT201600321B SM T201600321 B SMT201600321 B SM T201600321B SM 201600321 T SM201600321 T SM 201600321T SM 201600321 T SM201600321 T SM 201600321T SM T201600321 B SMT201600321 B SM T201600321B
Authority
SM
San Marino
Prior art keywords
antipsicotica
injectable composition
gradual release
gradual
release
Prior art date
Application number
SM201600321T
Other languages
English (en)
Inventor
Ochoa María Teresa Gomez
Aduriz Ibon Gutierro
Original Assignee
Laboratorios Farmacéuticos Rovi S A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43301889&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SMT201600321(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Laboratorios Farmacéuticos Rovi S A filed Critical Laboratorios Farmacéuticos Rovi S A
Publication of SMT201600321B publication Critical patent/SMT201600321B/it

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0024Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Dermatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Inorganic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Infusion, Injection, And Reservoir Apparatuses (AREA)
SM201600321T 2010-05-31 2016-09-15 Composizione iniettabile a rilascio graduale antipsicotica SMT201600321B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP10382154.2A EP2394664B1 (en) 2010-05-31 2010-05-31 Antipsychotic injectable depot composition

Publications (1)

Publication Number Publication Date
SMT201600321B true SMT201600321B (it) 2016-11-10

Family

ID=43301889

Family Applications (2)

Application Number Title Priority Date Filing Date
SM201600321T SMT201600321B (it) 2010-05-31 2016-09-15 Composizione iniettabile a rilascio graduale antipsicotica
SM201600320T SMT201600320B (it) 2010-05-31 2016-09-15 Composizione a deposito iniettabile antipsicotica

Family Applications After (1)

Application Number Title Priority Date Filing Date
SM201600320T SMT201600320B (it) 2010-05-31 2016-09-15 Composizione a deposito iniettabile antipsicotica

Country Status (33)

Country Link
US (2) US10085936B2 (it)
EP (2) EP2394664B1 (it)
JP (1) JP5882993B2 (it)
KR (1) KR101784330B1 (it)
CN (1) CN103002917B (it)
AP (1) AP3524A (it)
AU (1) AU2011260318B2 (it)
BR (1) BR112012030686B1 (it)
CA (1) CA2800111C (it)
CL (1) CL2012003350A1 (it)
CY (2) CY1117964T1 (it)
DK (2) DK2394664T3 (it)
EA (1) EA024155B1 (it)
ES (2) ES2589106T3 (it)
HR (2) HRP20161049T1 (it)
HU (2) HUE029895T2 (it)
IL (1) IL223129A (it)
LT (2) LT2394664T (it)
MA (1) MA34296B1 (it)
ME (1) ME02501B (it)
MX (1) MX338373B (it)
MY (1) MY161930A (it)
NZ (1) NZ604342A (it)
PH (1) PH12012502338B1 (it)
PL (2) PL2394664T3 (it)
PT (2) PT2394664T (it)
RS (1) RS55190B1 (it)
SG (1) SG185775A1 (it)
SI (2) SI2394664T1 (it)
SM (2) SMT201600321B (it)
UA (1) UA108885C2 (it)
WO (1) WO2011151355A1 (it)
ZA (1) ZA201209346B (it)

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US8852638B2 (en) 2005-09-30 2014-10-07 Durect Corporation Sustained release small molecule drug formulation
JP2010531807A (ja) 2007-05-25 2010-09-30 トルマー セラピューティクス, インコーポレイテッド リスペリドン化合物の徐放送達製剤
US10335366B2 (en) 2010-05-31 2019-07-02 Laboratorios Farmacéuticos Rovi, S.A. Risperidone or paliperidone implant formulation
US10285936B2 (en) 2010-05-31 2019-05-14 Laboratorios Farmacéuticos Rovi, S.A. Injectable composition with aromatase inhibitor
US10350159B2 (en) * 2010-05-31 2019-07-16 Laboratories Farmacéuticos Rovi, S.A. Paliperidone implant formulation
US10881605B2 (en) 2010-05-31 2021-01-05 Laboratorios Farmaceuticos Rovi, S.A. Methods for the preparation of injectable depot compositions
US10463607B2 (en) 2010-05-31 2019-11-05 Laboratorios Farmaceutics Rofi S.A. Antipsychotic Injectable Depot Composition
PT2394663T (pt) 2010-05-31 2021-11-26 Farm Rovi Lab Sa Composições para implantes biodegradáveis injectáveis
HUE029895T2 (en) 2010-05-31 2017-04-28 Farm Rovi Lab Sa Antipsychotic injectable depot composition
ES2456917T3 (es) * 2011-05-31 2014-04-24 Laboratorios Farmacéuticos Rovi, S.A. Formulación de implante de paliperidona
PT2529756T (pt) * 2011-05-31 2021-07-28 Farm Rovi Lab Sa Formulação de implante de risperidona e/ou paliperidona
US20140308352A1 (en) 2013-03-11 2014-10-16 Zogenix Inc. Compositions and methods involving polymer, solvent, and high viscosity liquid carrier material
CN105163719B (zh) 2013-03-11 2019-03-08 度瑞公司 包含高粘度液体载体的可注射控制释放组合物
WO2016199170A2 (en) * 2015-06-10 2016-12-15 Cipla Limited Paliperidone palmitate particles and compositions thereof
WO2018172850A1 (en) 2017-03-20 2018-09-27 Teva Pharmaceuticals International Gmbh Sustained release olanzapine formulaitons
CN109589304A (zh) * 2017-10-01 2019-04-09 万特制药(海南)有限公司 利培酮口服溶液及其制备方法
PE20210047A1 (es) 2018-06-12 2021-01-08 Farm Rovi Lab Sa Composicion inyectable
CN110420212A (zh) * 2019-08-19 2019-11-08 韩自勤 一种用于治疗精神分裂症组合物及其制备方法
US12318387B2 (en) 2021-07-16 2025-06-03 Laboratorios Farmaceuticos Rovi, S.A. Method of treating acute exacerbation of schizophrenia with long-acting injectable depot composition
TW202313047A (zh) 2021-09-21 2023-04-01 西班牙商禾霏藥品實驗室有限公司 抗精神病可注射儲積型組合物
WO2023233051A1 (es) 2022-05-18 2023-12-07 Laboratorios Farmacéuticos Rovi, S.A. Composiciones inyectables de liberación prolongada para su uso en el tratamiento con risperidona junto a inhibidores de la enzima cyp2d6

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DE50112157D1 (de) * 2000-01-11 2007-04-19 Roland Bodmeier Kit zur implantation enthaltend eine trägerphase und ein lösungsmittel
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JP2010531807A (ja) * 2007-05-25 2010-09-30 トルマー セラピューティクス, インコーポレイテッド リスペリドン化合物の徐放送達製剤
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RU2504360C2 (ru) * 2008-08-12 2014-01-20 Новартис Аг Фармацевтические композиции
US10335366B2 (en) 2010-05-31 2019-07-02 Laboratorios Farmacéuticos Rovi, S.A. Risperidone or paliperidone implant formulation
US10285936B2 (en) 2010-05-31 2019-05-14 Laboratorios Farmacéuticos Rovi, S.A. Injectable composition with aromatase inhibitor
US10350159B2 (en) 2010-05-31 2019-07-16 Laboratories Farmacéuticos Rovi, S.A. Paliperidone implant formulation
PT2394663T (pt) 2010-05-31 2021-11-26 Farm Rovi Lab Sa Composições para implantes biodegradáveis injectáveis
HUE029895T2 (en) 2010-05-31 2017-04-28 Farm Rovi Lab Sa Antipsychotic injectable depot composition
PT2529756T (pt) 2011-05-31 2021-07-28 Farm Rovi Lab Sa Formulação de implante de risperidona e/ou paliperidona
ES2456917T3 (es) 2011-05-31 2014-04-24 Laboratorios Farmacéuticos Rovi, S.A. Formulación de implante de paliperidona

Also Published As

Publication number Publication date
CL2012003350A1 (es) 2013-10-18
CN103002917A (zh) 2013-03-27
BR112012030686A2 (pt) 2020-08-25
AP2012006626A0 (en) 2012-12-31
BR112012030686B1 (pt) 2022-11-01
WO2011151355A1 (en) 2011-12-08
AU2011260318A1 (en) 2013-01-10
EP2394664B1 (en) 2016-06-01
RS55190B1 (sr) 2017-01-31
HRP20161100T1 (hr) 2016-11-04
MX2012013937A (es) 2013-02-11
DK2575890T3 (en) 2016-09-12
US10182982B2 (en) 2019-01-22
CA2800111A1 (en) 2011-12-08
US10085936B2 (en) 2018-10-02
PH12012502338B1 (en) 2018-08-31
ES2589106T3 (es) 2016-11-10
LT2575890T (lt) 2016-09-26
KR101784330B1 (ko) 2017-10-11
MA34296B1 (fr) 2013-06-01
PT2575890T (pt) 2016-09-06
CY1117964T1 (el) 2017-05-17
EA024155B1 (ru) 2016-08-31
SMT201600320B (it) 2016-11-10
AP3524A (en) 2016-01-11
PH12012502338A1 (en) 2013-02-11
SI2575890T1 (sl) 2016-10-28
CA2800111C (en) 2018-05-22
US20180221272A1 (en) 2018-08-09
ES2592527T3 (es) 2016-11-30
IL223129A (en) 2016-02-29
PL2575890T3 (pl) 2016-12-30
ZA201209346B (en) 2013-08-28
PT2394664T (pt) 2016-09-06
CY1117969T1 (el) 2017-05-17
AU2011260318B2 (en) 2014-11-27
EP2394664A1 (en) 2011-12-14
EP2575890B1 (en) 2016-06-01
JP2013528612A (ja) 2013-07-11
JP5882993B2 (ja) 2016-03-09
DK2394664T3 (en) 2016-09-12
PL2394664T3 (pl) 2016-12-30
US20130171202A1 (en) 2013-07-04
IL223129A0 (en) 2013-02-03
HRP20161049T1 (hr) 2016-12-30
ME02501B (me) 2017-02-20
EP2575890A1 (en) 2013-04-10
CN103002917B (zh) 2016-04-27
LT2394664T (lt) 2016-09-26
NZ604342A (en) 2014-11-28
HUE029056T2 (en) 2017-02-28
EA201201569A1 (ru) 2013-04-30
SI2394664T1 (sl) 2016-10-28
SG185775A1 (en) 2013-01-30
KR20130118742A (ko) 2013-10-30
MX338373B (es) 2016-04-13
UA108885C2 (uk) 2015-06-25
MY161930A (en) 2017-05-15
HUE029895T2 (en) 2017-04-28

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