SE8300945D0 - Mellanprodukter for framstellning av 4-substituerade imidazo (1,2-a)kinoxaliner - Google Patents

Mellanprodukter for framstellning av 4-substituerade imidazo (1,2-a)kinoxaliner

Info

Publication number: SE8300945D0
Authority: SE; Sweden
Prior art keywords: kinoxalines; intermediates; preparation; substituted imidazo; nitrogen
Prior art date: 1977-01-07

Application number

SE8300945A

Other languages

English (en)

Other versions

SE8300945L (sv

SE460477B (sv

Inventor

P L Warner

Jr E J Luber

Original Assignee

Bristol Myers Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-01-07

Filing date

1983-02-21

Publication date

1983-02-21

1983-02-21 Application filed by Bristol Myers Co filed Critical Bristol Myers Co

1983-02-21 Publication of SE8300945L publication Critical patent/SE8300945L/sv

1983-02-21 Publication of SE8300945D0 publication Critical patent/SE8300945D0/sv

1989-10-16 Publication of SE460477B publication Critical patent/SE460477B/sv

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Immunology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Transplantation (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

SE8300945A 1977-01-07 1983-02-21 1-(2-acylaminofenyl)imidazoler till anvaendning sommellanprodukter SE460477B (sv)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US75764077A	1977-01-07	1977-01-07

Publications (3)

Publication Number	Publication Date
SE8300945L SE8300945L (sv)	1983-02-21
SE8300945D0 true SE8300945D0 (sv)	1983-02-21
SE460477B SE460477B (sv)	1989-10-16

Family

ID=25048641

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
SE7800138A SE436359B (sv)	1977-01-07	1978-01-05	Analogiforfarande for framstellning av 4-substituerade imidazo/1,2-a/kinoxaliner
SE8300945A SE460477B (sv)	1977-01-07	1983-02-21	1-(2-acylaminofenyl)imidazoler till anvaendning sommellanprodukter

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
SE7800138A SE436359B (sv)	1977-01-07	1978-01-05	Analogiforfarande for framstellning av 4-substituerade imidazo/1,2-a/kinoxaliner

Country Status (19)

Country	Link
US (1)	US4160097A (sv)
JP (2)	JPS5387398A (sv)
AU (1)	AU521807B2 (sv)
BE (1)	BE862608A (sv)
CA (1)	CA1149385A (sv)
CH (2)	CH636102A5 (sv)
CS (1)	CS200232B2 (sv)
DE (2)	DE2800480A1 (sv)
DK (1)	DK157024C (sv)
FI (1)	FI64374C (sv)
FR (1)	FR2376858A1 (sv)
GB (2)	GB1579498A (sv)
GR (1)	GR73168B (sv)
IE (1)	IE46191B1 (sv)
LU (1)	LU78813A1 (sv)
NL (1)	NL7800114A (sv)
SE (2)	SE436359B (sv)
YU (1)	YU44663B (sv)
ZA (1)	ZA7827B (sv)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SE439308B (sv) *	1978-08-02	1985-06-10	Roussel Uclaf	Imidazo(1,2-a)kinoxaliner och farmaceutiska kompositioner derav
JPS5569567A (en) *	1978-11-21	1980-05-26	Eisai Co Ltd	Novel imidazole compound, and antidepressant containing the same
IT1209431B (it) *	1980-11-28	1989-07-16	Angeli Inst Spa	Imidazolilfenil amidine, processi per la loro preparazione e loro impiego farmaceutico, ed intermedi di preparazione.
DE3830054A1 (de) *	1988-09-03	1990-03-15	Boehringer Mannheim Gmbh	Phenylamide - verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel
JPH0349309U (sv) *	1989-09-21	1991-05-14
US6235740B1 (en)	1997-08-25	2001-05-22	Bristol-Myers Squibb Co.	Imidazoquinoxaline protein tyrosine kinase inhibitors
US6635626B1 (en)	1997-08-25	2003-10-21	Bristol-Myers Squibb Co.	Imidazoquinoxaline protein tyrosine kinase inhibitors
US6451796B1 (en)	1997-11-11	2002-09-17	Ono Pharmaceutical Co., Ltd.	Fused pyrazine compounds
WO1999045009A1 (en) *	1998-03-04	1999-09-10	Bristol-Myers Squibb Company	Heterocyclo-substituted imidazopyrazine protein tyrosine kinase inhibitors
US6869956B2 (en) *	2000-10-03	2005-03-22	Bristol-Myers Squibb Company	Methods of treating inflammatory and immune diseases using inhibitors of IκB kinase (IKK)
HUP0302925A3 (en)	2000-10-03	2004-10-28	Bristol Myers Squibb Co	Amino-substituted tetracyclic compouds useful as anti-inflammatory agents and pharmaceutical compositions comprising same
JP2004529088A (ja) *	2001-02-01	2004-09-24	ブリストル−マイヤーズ　スクイブ　カンパニー	ＩｋＢキナーゼ（ＩＫＫ）のインヒビターを用いる炎症性および免疫疾患の処置法
WO2008039794A1 (en) *	2006-09-25	2008-04-03	Arete Therapeutics, Inc.	Soluble epoxide hydrolase inhibitors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3541109A (en) *	1968-06-25	1970-11-17	Du Pont	1-substituted imidazoles useful in acth reserve assay
US4011236A (en) *	1968-09-09	1977-03-08	Merck & Co., Inc.	N-(benzimidazol-2-yl)arylcarboxamides as ultraviolet (uv) light absorbers
GB1347493A (en) *	1971-02-11	1974-02-27	Aspro Nicholas Ltd	Benzazine derivatives
US3994893A (en)	1975-11-03	1976-11-30	E. R. Squibb & Sons, Inc.	4-Amino derivatives of pyrozolo[1,5-a]quinoxaline-3-carboxylic acid and esters

1977
- 1977-12-08 US US05/858,515 patent/US4160097A/en not_active Expired - Lifetime
- 1977-12-23 GR GR55051A patent/GR73168B/el unknown
- 1977-12-28 JP JP15758177A patent/JPS5387398A/ja active Granted
- 1977-12-28 CA CA000293972A patent/CA1149385A/en not_active Expired
1978
- 1978-01-03 BE BE184085A patent/BE862608A/xx not_active IP Right Cessation
- 1978-01-04 DK DK004278A patent/DK157024C/da not_active IP Right Cessation
- 1978-01-04 ZA ZA00780027A patent/ZA7827B/xx unknown
- 1978-01-04 NL NL7800114A patent/NL7800114A/xx not_active Application Discontinuation
- 1978-01-04 FI FI780023A patent/FI64374C/fi not_active IP Right Cessation
- 1978-01-05 DE DE19782800480 patent/DE2800480A1/de active Granted
- 1978-01-05 SE SE7800138A patent/SE436359B/sv not_active IP Right Cessation
- 1978-01-05 LU LU78813A patent/LU78813A1/xx unknown
- 1978-01-05 DE DE2858766A patent/DE2858766C2/de not_active Expired - Fee Related
- 1978-01-06 YU YU21/78A patent/YU44663B/xx unknown
- 1978-01-06 CH CH15278A patent/CH636102A5/fr not_active IP Right Cessation
- 1978-01-06 IE IE37/78A patent/IE46191B1/en unknown
- 1978-01-06 GB GB492/78A patent/GB1579498A/en not_active Expired
- 1978-01-06 GB GB13335/79A patent/GB1579499A/en not_active Expired
- 1978-01-06 FR FR7800308A patent/FR2376858A1/fr active Granted
- 1978-01-09 CS CS78169A patent/CS200232B2/cs unknown
- 1978-01-11 AU AU32331/78A patent/AU521807B2/en not_active Expired
1983
- 1983-01-18 CH CH27483A patent/CH640229A5/fr not_active IP Right Cessation
- 1983-02-21 SE SE8300945A patent/SE460477B/sv not_active IP Right Cessation
1986
- 1986-01-17 JP JP61006590A patent/JPS61171470A/ja active Granted

Also Published As

Publication number	Publication date
CH636102A5 (fr)	1983-05-13
FI780023A7 (fi)	1978-07-08
SE8300945L (sv)	1983-02-21
AU521807B2 (en)	1982-04-29
CA1149385A (en)	1983-07-05
FI64374C (fi)	1983-11-10
FR2376858A1 (fr)	1978-08-04
GR73168B (sv)	1984-02-14
GB1579499A (en)	1980-11-19
US4160097A (en)	1979-07-03
CS200232B2 (en)	1980-08-29
CH640229A5 (fr)	1983-12-30
DK157024B (da)	1989-10-30
JPS5387398A (en)	1978-08-01
IE780037L (en)	1978-07-07
YU44663B (en)	1990-12-31
DE2800480A1 (de)	1978-07-13
BE862608A (fr)	1978-07-03
SE7800138L (sv)	1978-07-08
DE2858766C2 (sv)	1990-04-05
LU78813A1 (fr)	1978-09-18
DK157024C (da)	1990-04-02
DE2800480C2 (sv)	1990-04-12
JPS6259110B2 (sv)	1987-12-09
NL7800114A (nl)	1978-07-11
FI64374B (fi)	1983-07-29
FR2376858B1 (sv)	1980-10-24
GB1579498A (en)	1980-11-19
SE460477B (sv)	1989-10-16
IE46191B1 (en)	1983-03-23
YU2178A (en)	1990-04-30
JPH0130825B2 (sv)	1989-06-22
ZA7827B (en)	1979-01-31
SE436359B (sv)	1984-12-03
DK4278A (da)	1978-07-08
AU3233178A (en)	1979-07-19
JPS61171470A (ja)	1986-08-02

Publication	Publication Date	Title
SE8300945D0 (sv)	1983-02-21	Mellanprodukter for framstellning av 4-substituerade imidazo (1,2-a)kinoxaliner
FI852974L (fi)	1986-02-04	Nya n-hydroxylgruppen skyddande grupper och framstaellningsfoerfarande foer 3-acylamino-1-hydroxi-2-azetidinoner.
FI833918A0 (fi)	1983-10-26	-karboliner, foerfarande foer deras framstaellning och dessa innehaollande farmaceutiska preparat
DE3678797D1 (de)	1991-05-23	Neue 3-oxadiazol- und 3-carbonsaeure-beta-carbolinderivate, ihre herstellung und ihre verwendung als arzneimittel.
SE8002293L (sv)	1980-09-27	Nya antisekretoriska foreningar och deras anvendningsomrade
ES8101530A1 (es)	1980-12-16	Un procedimiento para la preparacion de alcoholes beta-gama-dihidro-poliprenilicos.
SE7910072L (sv)	1980-06-08	Pyrrolo- eller pyrido(2,1-c)(1,4)tiaziner eller -tiazepiner
JPS5750989A (en)	1982-03-25	Imidazole compound
AU588065B2 (en)	1989-09-07	Substituted diazaoxaspirodecanes, preparation thereof and use thereof as stabilizers for polymers
ES545009A0 (es)	1986-07-16	Procedimiento de preparacion de nuevas fenil-naftiridinas.
SE8306740D0 (sv)	1983-12-06	2-thiacephems and (5r) penems derivatives
DE3264928D1 (en)	1985-08-29	Process for producing brominated 1,3-dioxolen-2-ones
ES8307236A1 (es)	1983-02-01	Un procedimiento para la preparacion de ranitidina.
SE8803765L (sv)	1989-04-22	Nya isopolypeptider samt foerfarande foer framstaellning av desamma
ES8604940A1 (es)	1986-03-01	Procedimiento para la obtencion del 2-(2,4-difluorofenil)- 1,3-bis(1h-1,2,4-triazol-1-il)-propan-2-ol.
FI831521A0 (fi)	1983-05-03	Nytt foerfarande foer framstaellning av derivat av cyklopropankarboxylsyra och nya mellanprodukter
DK146389C (da)	1984-03-05	Analogifremgangsmaade til fremstilling af imidazo(1,2-a)imidazolforbindelser eller syreadditionssalte deraf
FI821583L (fi)	1982-11-08	Nya 1-pyrrolintiolaktimetrar och foerfarande foer deras framstaellning
DK452984A (da)	1985-03-23	Fremgangsmaade til fremstilling af quinolin-4-oner
MX156076A (es)	1988-06-29	Procedimiento para preparar esteres fluorofenoxibencilicos
ES8301991A1 (es)	1982-12-16	Procedimiento para la preparacion de 7-(2,6-dibromo-4-metil-fenil)-2,3-dihidro-imidazo 1,2-a, imidazoles.
GR76302B (sv)	1984-08-04
ES441437A1 (es)	1977-07-01	Procedimiento para la preparacion de crotonanilidas susti- tuidas.
DK452684D0 (da)	1984-09-21	Fremgangsmaade til fremstilling af quinolin-4-oner
ES8205774A1 (es)	1982-08-16	Procedimiento para la obtencion de 2(1h)-piridinonas

Legal Events

Date	Code	Title	Description
1995-01-31	NUG	Patent has lapsed	Ref document number: 8300945-6 Effective date: 19920806 Format of ref document f/p: F

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