DK4278A - 4-substituerede imidazo(1,2-a)quinoxaliner og mellemproduktersamt fremgangsmaade til fremstilling deraf - Google Patents

4-substituerede imidazo(1,2-a)quinoxaliner og mellemproduktersamt fremgangsmaade til fremstilling deraf

Info

Publication number: DK4278A
Authority: DK; Denmark
Prior art keywords: quinoxalines; manufacture; substituted imidazo; intermediate procedures; procedures
Prior art date: 1977-01-07

Application number

DK4278A

Other languages

English (en)

Other versions

DK157024C (da

DK157024B (da

Inventor

Jr P L Warner

Jr E J Luber

Original Assignee

Bristol Myers Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-01-07

Filing date

1978-01-04

Publication date

1978-07-08

1978-01-04 Application filed by Bristol Myers Co filed Critical Bristol Myers Co

1978-07-08 Publication of DK4278A publication Critical patent/DK4278A/da

1989-10-30 Publication of DK157024B publication Critical patent/DK157024B/da

1990-04-02 Application granted granted Critical

1990-04-02 Publication of DK157024C publication Critical patent/DK157024C/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Immunology (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Transplantation (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

DK004278A 1977-01-07 1978-01-04 Analogifremgangsmaade til fremstilling af 4-substituerede imidazooe1,2-aaaquinoxaliner samt 1-(2-acylaminophenyl)imidazoler til anvendelse som udgangsmaterialer ved fremgangsmaaden DK157024C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US75764077A	1977-01-07	1977-01-07
US75764077		1977-01-07

Publications (3)

Publication Number	Publication Date
DK4278A true DK4278A (da)	1978-07-08
DK157024B DK157024B (da)	1989-10-30
DK157024C DK157024C (da)	1990-04-02

Family

ID=25048641

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK004278A DK157024C (da)	1977-01-07	1978-01-04	Analogifremgangsmaade til fremstilling af 4-substituerede imidazooe1,2-aaaquinoxaliner samt 1-(2-acylaminophenyl)imidazoler til anvendelse som udgangsmaterialer ved fremgangsmaaden

Country Status (19)

Country	Link
US (1)	US4160097A (da)
JP (2)	JPS5387398A (da)
AU (1)	AU521807B2 (da)
BE (1)	BE862608A (da)
CA (1)	CA1149385A (da)
CH (2)	CH636102A5 (da)
CS (1)	CS200232B2 (da)
DE (2)	DE2858766C2 (da)
DK (1)	DK157024C (da)
FI (1)	FI64374C (da)
FR (1)	FR2376858A1 (da)
GB (2)	GB1579499A (da)
GR (1)	GR73168B (da)
IE (1)	IE46191B1 (da)
LU (1)	LU78813A1 (da)
NL (1)	NL7800114A (da)
SE (2)	SE436359B (da)
YU (1)	YU44663B (da)
ZA (1)	ZA7827B (da)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SE439308B (sv) *	1978-08-02	1985-06-10	Roussel Uclaf	Imidazo(1,2-a)kinoxaliner och farmaceutiska kompositioner derav
JPS5569567A (en) *	1978-11-21	1980-05-26	Eisai Co Ltd	Novel imidazole compound, and antidepressant containing the same
IT1209431B (it) *	1980-11-28	1989-07-16	Angeli Inst Spa	Imidazolilfenil amidine, processi per la loro preparazione e loro impiego farmaceutico, ed intermedi di preparazione.
DE3830054A1 (de) *	1988-09-03	1990-03-15	Boehringer Mannheim Gmbh	Phenylamide - verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel
JPH0349309U (da) *	1989-09-21	1991-05-14
US6235740B1 (en)	1997-08-25	2001-05-22	Bristol-Myers Squibb Co.	Imidazoquinoxaline protein tyrosine kinase inhibitors
US6635626B1 (en)	1997-08-25	2003-10-21	Bristol-Myers Squibb Co.	Imidazoquinoxaline protein tyrosine kinase inhibitors
US6451796B1 (en)	1997-11-11	2002-09-17	Ono Pharmaceutical Co., Ltd.	Fused pyrazine compounds
EP1066286B1 (en) *	1998-03-04	2009-04-29	Bristol-Myers Squibb Company	Heterocyclo-substituted imidazopyrazine protein tyrosine kinase inhibitors
CA2424303A1 (en)	2000-10-03	2002-04-11	Bristol-Myers Squibb Company	Amino-substituted tetracyclic compounds useful as anti-inflammatory agents and pharmaceutical compositions comprising same
US6869956B2 (en) *	2000-10-03	2005-03-22	Bristol-Myers Squibb Company	Methods of treating inflammatory and immune diseases using inhibitors of IκB kinase (IKK)
HUP0304045A3 (en) *	2001-02-01	2005-05-30	Bristol Myers Squibb Company P	Use of ikb-kinase inhibitors for treating of inflammatory and immune diseases and pharmaceutical compositions containing them
JP2010504362A (ja) *	2006-09-25	2010-02-12	アレテセラピューティクス，インコーポレイテッド	可溶性エポキシドヒドロラーゼ阻害剤

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3541109A (en) *	1968-06-25	1970-11-17	Du Pont	1-substituted imidazoles useful in acth reserve assay
US4011236A (en) *	1968-09-09	1977-03-08	Merck & Co., Inc.	N-(benzimidazol-2-yl)arylcarboxamides as ultraviolet (uv) light absorbers
GB1347493A (en) *	1971-02-11	1974-02-27	Aspro Nicholas Ltd	Benzazine derivatives
US3994893A (en)	1975-11-03	1976-11-30	E. R. Squibb & Sons, Inc.	4-Amino derivatives of pyrozolo[1,5-a]quinoxaline-3-carboxylic acid and esters

1977
- 1977-12-08 US US05/858,515 patent/US4160097A/en not_active Expired - Lifetime
- 1977-12-23 GR GR55051A patent/GR73168B/el unknown
- 1977-12-28 CA CA000293972A patent/CA1149385A/en not_active Expired
- 1977-12-28 JP JP15758177A patent/JPS5387398A/ja active Granted
1978
- 1978-01-03 BE BE184085A patent/BE862608A/xx not_active IP Right Cessation
- 1978-01-04 FI FI780023A patent/FI64374C/fi not_active IP Right Cessation
- 1978-01-04 DK DK004278A patent/DK157024C/da not_active IP Right Cessation
- 1978-01-04 ZA ZA00780027A patent/ZA7827B/xx unknown
- 1978-01-04 NL NL7800114A patent/NL7800114A/xx not_active Application Discontinuation
- 1978-01-05 DE DE2858766A patent/DE2858766C2/de not_active Expired - Fee Related
- 1978-01-05 LU LU78813A patent/LU78813A1/xx unknown
- 1978-01-05 DE DE19782800480 patent/DE2800480A1/de active Granted
- 1978-01-05 SE SE7800138A patent/SE436359B/sv not_active IP Right Cessation
- 1978-01-06 GB GB13335/79A patent/GB1579499A/en not_active Expired
- 1978-01-06 YU YU21/78A patent/YU44663B/xx unknown
- 1978-01-06 FR FR7800308A patent/FR2376858A1/fr active Granted
- 1978-01-06 GB GB492/78A patent/GB1579498A/en not_active Expired
- 1978-01-06 CH CH15278A patent/CH636102A5/fr not_active IP Right Cessation
- 1978-01-06 IE IE37/78A patent/IE46191B1/en unknown
- 1978-01-09 CS CS78169A patent/CS200232B2/cs unknown
- 1978-01-11 AU AU32331/78A patent/AU521807B2/en not_active Expired
1983
- 1983-01-18 CH CH27483A patent/CH640229A5/fr not_active IP Right Cessation
- 1983-02-21 SE SE8300945A patent/SE460477B/sv not_active IP Right Cessation
1986
- 1986-01-17 JP JP61006590A patent/JPS61171470A/ja active Granted

Also Published As

Publication number	Publication date
CH640229A5 (fr)	1983-12-30
DK157024C (da)	1990-04-02
CS200232B2 (en)	1980-08-29
SE460477B (sv)	1989-10-16
GB1579499A (en)	1980-11-19
GR73168B (da)	1984-02-14
IE780037L (en)	1978-07-07
JPH0130825B2 (da)	1989-06-22
DE2858766C2 (da)	1990-04-05
DE2800480A1 (de)	1978-07-13
CH636102A5 (fr)	1983-05-13
IE46191B1 (en)	1983-03-23
DK157024B (da)	1989-10-30
YU44663B (en)	1990-12-31
YU2178A (en)	1990-04-30
JPS5387398A (en)	1978-08-01
BE862608A (fr)	1978-07-03
SE436359B (sv)	1984-12-03
ZA7827B (en)	1979-01-31
LU78813A1 (fr)	1978-09-18
GB1579498A (en)	1980-11-19
SE7800138L (sv)	1978-07-08
JPS61171470A (ja)	1986-08-02
CA1149385A (en)	1983-07-05
FI780023A7 (fi)	1978-07-08
FI64374C (fi)	1983-11-10
FR2376858A1 (fr)	1978-08-04
US4160097A (en)	1979-07-03
SE8300945L (sv)	1983-02-21
JPS6259110B2 (da)	1987-12-09
AU3233178A (en)	1979-07-19
AU521807B2 (en)	1982-04-29
FI64374B (fi)	1983-07-29
FR2376858B1 (da)	1980-10-24
NL7800114A (nl)	1978-07-11
DE2800480C2 (da)	1990-04-12
SE8300945D0 (sv)	1983-02-21

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Legal Events

Date	Code	Title	Description
1992-09-28	PBP	Patent lapsed