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PE20120325A1 - Aminopirimidinas sustituidas con arilo como agentes fungicidas - Google Patents

Aminopirimidinas sustituidas con arilo como agentes fungicidas

Info

Publication number
PE20120325A1
PE20120325A1 PE2011001972A PE2011001972A PE20120325A1 PE 20120325 A1 PE20120325 A1 PE 20120325A1 PE 2011001972 A PE2011001972 A PE 2011001972A PE 2011001972 A PE2011001972 A PE 2011001972A PE 20120325 A1 PE20120325 A1 PE 20120325A1
Authority
PE
Peru
Prior art keywords
aminopyrimidines
aryl
substituted
fungicide
compounds
Prior art date
Application number
PE2011001972A
Other languages
English (en)
Inventor
George Davis
William Lo
James Renga
Francis Tisdell
Maurice Yap
David Young
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of PE20120325A1 publication Critical patent/PE20120325A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/30—Halogen atoms or nitro radicals

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

SE REFIERE A COMPUESTOS DERIVADOS DE AMINOPIRIMIDINAS DE FORMULA (1) DONDE X1 ES N O C-R3; X2 ES N O C-R4 CON LA CONDICION DE QUE X1 Y X2 NO SEAN AMBOS N; R1 A R7 SON CADA UNO H, CN, CHO, F, ALQUILO(C1-C4), ALCOXI(C1-C4), ENTRE OTROS, OPCIONALMENTE SUSTITUIDOS CON F, OH, CN, NO2, ENTRE OTROS; Q ES ARILO O HETEROCICLO OPCIONALMENTE SUSTITUIDO CON R1 A R7. SON COMPUESTOS PREFERIDOS LOS DE FORMULA (i), (ii), ENTRE OTROS. TAMBIEN SE REFIERE A UNA COMPOSICION FUNGICIDA QUE ADEMAS PUEDE CONTENER UN INSECTICIDA, HERBICIDA O FUNGICIDA. DICHOS COMPUESTOS SON UTILES PARA CONTROLAR HONGOS PATOGENOS EN PLANTAS
PE2011001972A 2009-05-19 2010-05-03 Aminopirimidinas sustituidas con arilo como agentes fungicidas PE20120325A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17940209P 2009-05-19 2009-05-19

Publications (1)

Publication Number Publication Date
PE20120325A1 true PE20120325A1 (es) 2012-04-12

Family

ID=42315653

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2011001972A PE20120325A1 (es) 2009-05-19 2010-05-03 Aminopirimidinas sustituidas con arilo como agentes fungicidas

Country Status (24)

Country Link
US (2) US8759356B2 (es)
EP (1) EP2432767B1 (es)
JP (1) JP2012527461A (es)
KR (1) KR20120016247A (es)
CN (1) CN102438993A (es)
AU (1) AU2010250017B2 (es)
BR (1) BRPI1011058A2 (es)
CA (1) CA2760911A1 (es)
CL (1) CL2011002922A1 (es)
CO (1) CO6460778A2 (es)
CR (1) CR20110589A (es)
DK (1) DK2432767T3 (es)
EC (1) ECSP11011467A (es)
ES (1) ES2417355T3 (es)
HN (1) HN2011003040A (es)
MX (1) MX2011012343A (es)
NZ (1) NZ596123A (es)
PE (1) PE20120325A1 (es)
PL (1) PL2432767T3 (es)
PT (1) PT2432767E (es)
RU (1) RU2011151603A (es)
SI (1) SI2432767T1 (es)
TW (1) TW201041512A (es)
WO (1) WO2010135070A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GEP20166432B (en) 2011-09-27 2016-02-10 Novartis Ag 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant idh
UY34632A (es) 2012-02-24 2013-05-31 Novartis Ag Compuestos de oxazolidin- 2- ona y usos de los mismos
US9296733B2 (en) 2012-11-12 2016-03-29 Novartis Ag Oxazolidin-2-one-pyrimidine derivative and use thereof for the treatment of conditions, diseases and disorders dependent upon PI3 kinases
WO2014141104A1 (en) 2013-03-14 2014-09-18 Novartis Ag 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant idh

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Also Published As

Publication number Publication date
HN2011003040A (es) 2013-10-22
US20140275123A1 (en) 2014-09-18
BRPI1011058A2 (pt) 2015-08-25
PL2432767T3 (pl) 2013-11-29
AU2010250017B2 (en) 2015-02-12
DK2432767T3 (da) 2013-09-30
WO2010135070A1 (en) 2010-11-25
CN102438993A (zh) 2012-05-02
AU2010250017A1 (en) 2011-11-24
US20100298143A1 (en) 2010-11-25
ECSP11011467A (es) 2011-12-30
RU2011151603A (ru) 2013-06-27
KR20120016247A (ko) 2012-02-23
ES2417355T3 (es) 2013-08-07
US8759356B2 (en) 2014-06-24
JP2012527461A (ja) 2012-11-08
CL2011002922A1 (es) 2012-04-13
SI2432767T1 (sl) 2013-10-30
EP2432767B1 (en) 2013-06-26
EP2432767A1 (en) 2012-03-28
CR20110589A (es) 2012-03-06
TW201041512A (en) 2010-12-01
MX2011012343A (es) 2011-12-14
NZ596123A (en) 2014-08-29
PT2432767E (pt) 2013-07-25
CO6460778A2 (es) 2012-06-15
CA2760911A1 (en) 2010-11-25

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