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PE20071244A1 - Formas farmaceuticas en forma de pelicula para usar en la cavidad bucal (obleas) - Google Patents

Formas farmaceuticas en forma de pelicula para usar en la cavidad bucal (obleas)

Info

Publication number
PE20071244A1
PE20071244A1 PE2007000071A PE2007000071A PE20071244A1 PE 20071244 A1 PE20071244 A1 PE 20071244A1 PE 2007000071 A PE2007000071 A PE 2007000071A PE 2007000071 A PE2007000071 A PE 2007000071A PE 20071244 A1 PE20071244 A1 PE 20071244A1
Authority
PE
Peru
Prior art keywords
beta
weight
cyclodextrin
wafers
proportion
Prior art date
Application number
PE2007000071A
Other languages
English (en)
Inventor
Hans-Peter Podhaisky
Stefan Bracht
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of PE20071244A1 publication Critical patent/PE20071244A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/40Cyclodextrins; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26Androgens
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30Oestrogens
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/34Gestagens

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Nutrition Science (AREA)
  • Molecular Biology (AREA)
  • Physiology (AREA)
  • Reproductive Health (AREA)
  • Inorganic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

SE REFIERE A UNA FORMA FARMACEUTICA EN FORMA DE PELICULA (OBLEA) DE APLICACION BUCAL QUE CONSISTE EN UN SISTEMA QUE COMPRENDE a) UN FARMACO LIPOFILICO TAL COMO UNA HORMONA ESTEROIDE DEL GRUPO DE LOS ANDROGENOS, GESTAGENOS Y LOS ESTROGENOS EN UNA PROPORCION DE 0,1- 5% EN PESO; b) UNA PROPORCION DE 30 A 70% EN PESO DE UNA CICLODEXTINA TAL COMO BETA O GAMMA CICLODEXTRINA O UN DERIVADO TAL COMO HP-BETA-CICLODEXTRINA O SULFOBUTILETER-BETA-CICLODEXTRINA; Y c) UN FORMADOR DE PELICULAS QUE SE DESCOMPONE EN MEDIO ACUOSO SELECCIONADO DEL GRUPO QUE CONTIENE EUDRAGITS, ALCOHOLES POLIVINILICOS Y CELULOSAS, EN UNA PROPORCION DE 0,01-0,1% EN PESO. TAMBIEN SE REFIERE UN PROCEDIMIENTO DE PREPARACION. DICHA OBLEA PRESENTA BUENAS PROPIEDADES MUCOHADESIVAS, Y EL FARMACO PERMANECE TOTALMENTE DISUELTO DE MANERA QUE LA PELICULA SECA PERMITA UNA TRANSMICION DE LUZ VISIBLE DE IGUAL A MAS DEL 50%
PE2007000071A 2006-01-24 2007-01-23 Formas farmaceuticas en forma de pelicula para usar en la cavidad bucal (obleas) PE20071244A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102006003512A DE102006003512A1 (de) 2006-01-24 2006-01-24 Plättchenförmige Arzneimittel zur transbukkalen Applikation von Arzneistoffen

Publications (1)

Publication Number Publication Date
PE20071244A1 true PE20071244A1 (es) 2008-02-24

Family

ID=37930392

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2007000071A PE20071244A1 (es) 2006-01-24 2007-01-23 Formas farmaceuticas en forma de pelicula para usar en la cavidad bucal (obleas)

Country Status (13)

Country Link
US (1) US20070292479A1 (es)
EP (1) EP1978927A1 (es)
JP (1) JP2009523837A (es)
KR (1) KR20080091156A (es)
CN (1) CN101374500A (es)
AR (1) AR059174A1 (es)
CA (1) CA2637300A1 (es)
DE (1) DE102006003512A1 (es)
DO (1) DOP2007000017A (es)
PE (1) PE20071244A1 (es)
TW (1) TW200808382A (es)
UY (1) UY30109A1 (es)
WO (1) WO2007085498A1 (es)

Families Citing this family (26)

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Publication number Priority date Publication date Assignee Title
US8821915B2 (en) 2002-08-09 2014-09-02 Veroscience, Llc Therapeutic process for the treatment of the metabolic syndrome and associated metabolic disorders
US20100035886A1 (en) 2007-06-21 2010-02-11 Veroscience, Llc Parenteral formulations of dopamine agonists
US8741918B2 (en) * 2007-06-21 2014-06-03 Veroscience Llc Parenteral formulations of dopamine agonists
MX2010008940A (es) * 2008-02-13 2010-10-05 Bayer Schering Pharma Ag Sistemas de administracion de drogas que contienen estradiol.
EP2252261A2 (en) * 2008-02-13 2010-11-24 Bayer Schering Pharma Aktiengesellschaft Drug delivery system with stabilising effect
US9265779B2 (en) 2008-05-13 2016-02-23 Lts Lohmann Therapie-Systeme Ag Method of using a film-shaped preparation comprising oily substances for oral administration
DE102008023345B4 (de) * 2008-05-13 2014-12-04 Lts Lohmann Therapie-Systeme Ag Filmförmige Zubereitung mit öligen Substanzen zur oralen Verabreichung
TW201008569A (en) * 2008-08-08 2010-03-01 Bayer Schering Pharma Ag Progestin-containing drug delivery system
US20120282340A1 (en) * 2008-11-21 2012-11-08 Bayer Schering Pharma Aktiengesellschaft Drug delivery system
US9352025B2 (en) 2009-06-05 2016-05-31 Veroscience Llc Combination of dopamine agonists plus first phase insulin secretagogues for the treatment of metabolic disorders
UY32836A (es) * 2009-08-12 2011-03-31 Bayer Schering Pharma Ag Partículas estabilizadas que comprenden 5-metil-(6s)-tetrahidrofolato
WO2011020610A1 (en) 2009-08-19 2011-02-24 Bayer Schering Pharma Aktiengesellschaft Drug delivery systems (wafer) for pediatric use
CN101919803A (zh) * 2010-07-16 2010-12-22 钟术光 一种控释制剂
CN101985044B (zh) * 2010-07-16 2013-10-23 钟术光 一种掩味的药物涂层组合物
IT1401354B1 (it) 2010-08-02 2013-07-18 Quaglia Sistemi per il rilascio controllato a base di polimeri bioadesivi loro processo di produzione e impieghi clinici
CN102440979A (zh) * 2010-09-30 2012-05-09 迪特克(济源)绿色生物科技有限公司 一种纤维素衍生物复合膜及其制备方法
US20140271867A1 (en) * 2013-03-15 2014-09-18 Monosol Rx, Llc Film delivery system for active ingredients
US20130115266A1 (en) * 2011-11-04 2013-05-09 Bestsweet, Inc. Edible wafer-type product for delivery of nutraceuticals and pharmaceuticals
WO2014078576A2 (en) * 2012-11-14 2014-05-22 Abon Pharmaceuticals, Llc Oral transmucosal drug delivery system
WO2014144366A1 (en) * 2013-03-15 2014-09-18 Monosol Rx, Llc. Steroid hormone delivery systems and methods of preparing the same
EA201792206A1 (ru) * 2015-04-03 2018-02-28 Сантен Фармасьютикал Ко., Лтд. Терапевтическое средство для лечения синдрома сухого глаза, содержащее в качестве активного ингредиента нандролон или его сложный эфир или метенолон или его сложный эфир
WO2017151042A1 (en) * 2016-03-02 2017-09-08 Marvel Pharma Consulting Pharmaceutical compositions for on demand anticoagulant therapy
RU2699808C2 (ru) * 2017-12-05 2019-09-11 Общество с ограниченной ответственностью "Эндокринные технологии" Биоразлагаемая система трансмукозальной доставки дротаверина
DE102018002066A1 (de) 2018-03-14 2019-09-19 Irina Gentsinger Orale filmförmige Darreichungsform
RU2729659C1 (ru) * 2019-05-29 2020-08-11 Общество с ограниченной ответственностью "Эндокринные технологии" Лекарственная форма для высвобождения дротаверина в полости рта
CN116077416B (zh) * 2021-11-05 2024-12-06 深圳埃格林医药有限公司 一种包含孕激素的口服制剂及制备方法和应用

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US4596795A (en) * 1984-04-25 1986-06-24 The United States Of America As Represented By The Secretary, Dept. Of Health & Human Services Administration of sex hormones in the form of hydrophilic cyclodextrin derivatives
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Also Published As

Publication number Publication date
DE102006003512A1 (de) 2007-08-02
DOP2007000017A (es) 2007-09-15
AR059174A1 (es) 2008-03-12
CN101374500A (zh) 2009-02-25
US20070292479A1 (en) 2007-12-20
KR20080091156A (ko) 2008-10-09
EP1978927A1 (de) 2008-10-15
CA2637300A1 (en) 2007-08-02
WO2007085498A1 (de) 2007-08-02
JP2009523837A (ja) 2009-06-25
UY30109A1 (es) 2007-08-31
TW200808382A (en) 2008-02-16

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