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PE20070319A1 - Formulaciones farmaceuticas de liberacion inmediata y con una carga de droga elevada de (4-ciclofenil) [4-(4-piridilmetil) ftalazin-1- ilo] no micronizado, y sus sales - Google Patents

Formulaciones farmaceuticas de liberacion inmediata y con una carga de droga elevada de (4-ciclofenil) [4-(4-piridilmetil) ftalazin-1- ilo] no micronizado, y sus sales

Info

Publication number
PE20070319A1
PE20070319A1 PE2006000619A PE2006000619A PE20070319A1 PE 20070319 A1 PE20070319 A1 PE 20070319A1 PE 2006000619 A PE2006000619 A PE 2006000619A PE 2006000619 A PE2006000619 A PE 2006000619A PE 20070319 A1 PE20070319 A1 PE 20070319A1
Authority
PE
Peru
Prior art keywords
ilo
micronized
composition
ftalazin
cyclophenyl
Prior art date
Application number
PE2006000619A
Other languages
English (en)
Inventor
Kai Jurgens
Thomas Backensfeld
Adrian Funke
Kai Thode
Thorsten Wagner
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of PE20070319A1 publication Critical patent/PE20070319A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50Pyridazines; Hydrogenated pyridazines
    • A61K31/502Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with carbocyclic ring systems, e.g. cinnoline, phthalazine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

SE REFIERE A UNA COMPOSICION FARMACEUTICA SOLIDA QUE COMPRENDE A) UNA SAL DE (4-CLOROFENIL)[4-(4-PIRIDIL-METIL)-FTALAZIN-1-ILO] NO MICRONIZADO TAL COMO HIDROGENO SUCCINATO DE (4-CLOROFENIL)[4-(4-PIRIDIL-METIL)-FTALAZIN-1-IL]AMONIO QUE SE ENCUENTRA EN UNA CANTIDAD DE 50% A 95% EN PESO DE LA COMPOSICION Y SE LIBERA DE DICHA COMPOSICION EN 30 MINUTOS; Y B) EXCIPIENTES TALES COMO i) RELLENOS TAL COMO SACAROSA, SORBITOL, MANITOL, ENTRE OTROS; ii) AGLUTINANTES TAL COMO GLUCOSA, ACACIA, GELATINA, ENTRE OTROS; iii) AGENTES TENSIOACTIVOS TAL COMO LECITINA, ESTEARATO DE POLIOXIETILEN, LAURIL SULFATO DE SODIO, ENTRE OTROS; iv) DESINTEGRANTES TAL COMO CROSCARMELOSA SODICA, POVIDONA RETICULADA, GLICOLATO DE ALMIDON DE SODIO, ENTRE OTROS; Y v) DESLIZANTES Y LUBRICANTES TAL COMO ESTEARATO DE MAGNESIO, ESTEARATO DE CINC, ENTRE OTROS. SE REFIERE TAMBIEN A UN PROCESO DE PREPARACION. DICHA COMPOSICION ES UTIL PARA EL TRATAMIENTO DEL CANCER
PE2006000619A 2005-06-07 2006-06-06 Formulaciones farmaceuticas de liberacion inmediata y con una carga de droga elevada de (4-ciclofenil) [4-(4-piridilmetil) ftalazin-1- ilo] no micronizado, y sus sales PE20070319A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP05090166A EP1731153A1 (en) 2005-06-07 2005-06-07 Immediate-release and high-drug-load pharmaceutical formulations of non-micronised (4-chlorophenyl)¬4-(4-pyridylmethyl)phthalazin-1-yl| and salts thereof

Publications (1)

Publication Number Publication Date
PE20070319A1 true PE20070319A1 (es) 2007-04-12

Family

ID=34938467

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2006000619A PE20070319A1 (es) 2005-06-07 2006-06-06 Formulaciones farmaceuticas de liberacion inmediata y con una carga de droga elevada de (4-ciclofenil) [4-(4-piridilmetil) ftalazin-1- ilo] no micronizado, y sus sales

Country Status (21)

Country Link
EP (2) EP1731153A1 (es)
JP (1) JP2008542420A (es)
KR (1) KR20080031005A (es)
CN (1) CN101242840A (es)
AR (1) AR053889A1 (es)
AU (1) AU2006256852A1 (es)
BR (1) BRPI0613393A2 (es)
CA (1) CA2610975A1 (es)
CR (1) CR9563A (es)
DO (1) DOP2006000127A (es)
EC (1) ECSP078038A (es)
GT (1) GT200600242A (es)
IL (1) IL187905A0 (es)
MX (1) MX2007015494A (es)
NO (1) NO20080065L (es)
PE (1) PE20070319A1 (es)
RU (1) RU2007147951A (es)
TW (1) TW200716115A (es)
UY (1) UY29582A1 (es)
WO (1) WO2006131393A1 (es)
ZA (1) ZA200800112B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1958616A1 (en) * 2007-02-13 2008-08-20 Bayer Schering Pharma Aktiengesellschaft Pharmaceutical formulations of 1-[4-chloroanilino]-4-[4-pyridylmethyl] phthalazine or salts thereof
TW201618783A (zh) 2014-08-07 2016-06-01 艾森塔製藥公司 以布魯頓(Bruton)氏酪胺酸激酶(BTK)佔據和BTK再合成速率為基礎之治療癌症、免疫和自體免疫疾病及發炎性疾病之方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CO4950519A1 (es) * 1997-02-13 2000-09-01 Novartis Ag Ftalazinas, preparaciones farmaceuticas que las comprenden y proceso para su preparacion

Also Published As

Publication number Publication date
EP1888072A1 (en) 2008-02-20
ECSP078038A (es) 2008-01-23
CN101242840A (zh) 2008-08-13
IL187905A0 (en) 2008-03-20
WO2006131393A1 (en) 2006-12-14
MX2007015494A (es) 2008-02-22
KR20080031005A (ko) 2008-04-07
EP1731153A1 (en) 2006-12-13
CA2610975A1 (en) 2006-12-14
DOP2006000127A (es) 2006-12-15
AU2006256852A8 (en) 2006-12-14
JP2008542420A (ja) 2008-11-27
RU2007147951A (ru) 2009-07-20
AR053889A1 (es) 2007-05-23
CR9563A (es) 2008-02-20
TW200716115A (en) 2007-05-01
ZA200800112B (en) 2010-06-30
BRPI0613393A2 (pt) 2011-01-11
UY29582A1 (es) 2007-01-31
GT200600242A (es) 2007-02-09
NO20080065L (no) 2008-03-06
AU2006256852A1 (en) 2006-12-14

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