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PE20030323A1 - Composicion farmaceutica - Google Patents

Composicion farmaceutica

Info

Publication number
PE20030323A1
PE20030323A1 PE2002000832A PE2002000832A PE20030323A1 PE 20030323 A1 PE20030323 A1 PE 20030323A1 PE 2002000832 A PE2002000832 A PE 2002000832A PE 2002000832 A PE2002000832 A PE 2002000832A PE 20030323 A1 PE20030323 A1 PE 20030323A1
Authority
PE
Peru
Prior art keywords
tablet
pharmaceutical composition
fluoroanilyline
cyclooxygenase
polyvinylpyrrolidone
Prior art date
Application number
PE2002000832A
Other languages
English (en)
Inventor
Anees Abdulquadar Karnachi
Simon David Bateman
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of PE20030323A1 publication Critical patent/PE20030323A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

PARA TRATAR UN TRANSTORNO O UNA CONDICION DEPENDIENTES DE CICLOOXIGENASA-2, CARACTERIZADA PORQUE COMPRENDE: A)UNA TABLETA DE LIBERACION INMEDIATA DE 400 mg DE ACIDO 5-METIL-2-(2´-CLORO-6´-FLUOROANILINO) FENILACETICO O UNA SAL DEL MISMO FARMACEUTICAMENTE ACEPTABLE COMO AGENTE ACTIVO QUE ESTA PRESENTE EN LA TABLETA ENTRE 60% Y 70%, EN PESO; Y, B)6,6% DE POLIVINILPIRROLIDONA; C)4,3% DE CROSCARAMELOSA SODICA; D)0,5% DE ESTEARATO DE MAGNESIO; Y, E)23,56% DE CELULOSA MICROCRISTALINA. DONDE, LA TABLETA NO COMPRENDE SUFICIENTES COMPONENTES INSOLUBLES EN AGUA O POLIMERICOS QUE IMPARTAN A LA COMPOSICION CARACTERISTICAS DE LIBERACION PROLONGADA
PE2002000832A 2001-08-31 2002-08-29 Composicion farmaceutica PE20030323A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US31638901P 2001-08-31 2001-08-31

Publications (1)

Publication Number Publication Date
PE20030323A1 true PE20030323A1 (es) 2003-05-12

Family

ID=23228840

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2002000832A PE20030323A1 (es) 2001-08-31 2002-08-29 Composicion farmaceutica

Country Status (29)

Country Link
US (2) US20030114527A1 (es)
EP (1) EP1425005B1 (es)
JP (1) JP4636796B2 (es)
KR (1) KR100895551B1 (es)
CN (1) CN100406008C (es)
AR (1) AR036312A1 (es)
AT (1) ATE324883T1 (es)
AU (1) AU2002331094B2 (es)
BR (1) BR0212155A (es)
CA (1) CA2456604C (es)
CO (1) CO5560554A2 (es)
CY (1) CY1106137T1 (es)
DE (1) DE60211183T2 (es)
DK (1) DK1425005T3 (es)
EC (1) ECSP044986A (es)
ES (1) ES2263813T3 (es)
HU (1) HUP0401429A2 (es)
IL (1) IL160375A0 (es)
MX (1) MXPA04001933A (es)
MY (1) MY137516A (es)
NO (1) NO20040860L (es)
NZ (1) NZ531342A (es)
PE (1) PE20030323A1 (es)
PL (1) PL367464A1 (es)
PT (1) PT1425005E (es)
RU (1) RU2329801C2 (es)
SI (1) SI1425005T1 (es)
WO (1) WO2003020261A1 (es)
ZA (1) ZA200400877B (es)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR030630A1 (es) * 2000-09-11 2003-08-27 Novartis Ag Composiciones farmaceuticas
GB0201520D0 (en) * 2002-01-23 2002-03-13 Novartis Ag Pharmaceutical uses
PL370907A1 (en) * 2002-03-07 2005-05-30 Novartis Ag Pharmaceutical compositions
US8148414B2 (en) 2008-08-19 2012-04-03 Xenoport, Inc. Prodrugs of methyl hydrogen fumarate, pharmaceutical compositions thereof, and methods of use
US10787701B2 (en) 2010-04-05 2020-09-29 Prognosys Biosciences, Inc. Spatially encoded biological assays
US20140093563A1 (en) * 2011-06-13 2014-04-03 Ranbaxy Laboratories Limited Febuxostat compositions
PL2851075T3 (pl) 2012-05-14 2022-02-21 Shionogi & Co., Ltd. Preparat zawierający pochodną 6,7-nienasyconego-7-karbamoilomorfinanu
WO2014031844A1 (en) 2012-08-22 2014-02-27 Xenoport, Inc. Methods of administering monomethyl fumarate and prodrugs thereof having reduced side effects
AU2013305684B2 (en) 2012-08-22 2016-11-24 Xenoport, Inc. Oral dosage forms of methyl hydrogen fumarate and prodrugs thereof
EA018867B1 (ru) * 2012-11-01 2013-11-29 Лаборатория Тютор С.А.С.И.Ф.И.А. Способ получения фармацевтической композиции и продукт способа
US10179118B2 (en) 2013-03-24 2019-01-15 Arbor Pharmaceuticals, Llc Pharmaceutical compositions of dimethyl fumarate
US9302977B2 (en) 2013-06-07 2016-04-05 Xenoport, Inc. Method of making monomethyl fumarate
US9421182B2 (en) 2013-06-21 2016-08-23 Xenoport, Inc. Cocrystals of dimethyl fumarate
EP3041467A1 (en) 2013-09-06 2016-07-13 XenoPort, Inc. Crystalline forms of (n,n-diethylcarbamoyl)methyl methyl (2e)but-2-ene-1,4-dioate, methods of synthesis and use
RU2712267C2 (ru) * 2014-01-10 2020-01-28 Джонсон энд Джонсон Консьюмер Инк. Способ изготовления таблеток с использованием радиочастотного излучения и частиц с поглощающим покрытием
US9999672B2 (en) 2014-03-24 2018-06-19 Xenoport, Inc. Pharmaceutical compositions of fumaric acid esters
EP3162362A1 (de) * 2015-10-30 2017-05-03 Dr. Falk Pharma Gmbh Optimierte mesalazinhaltige hochdosistablette
US10493026B2 (en) 2017-03-20 2019-12-03 Johnson & Johnson Consumer Inc. Process for making tablet using radiofrequency and lossy coated particles
WO2025043076A1 (en) 2023-08-24 2025-02-27 10X Genomics, Inc. Methods, kits, and compositions for spatial detection of genetic variants

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH08511009A (ja) * 1993-06-08 1996-11-19 チバ−ガイギー アクチェンゲゼルシャフト ジクロフェナックを含有する経口固体剤形の製造方法
IL126899A (en) * 1996-05-17 2004-03-28 Merck & Co Inc Preparations for once-daily treatment of diseases mediated by cyclooxygenase-2
CO4960662A1 (es) * 1997-08-28 2000-09-25 Novartis Ag Ciertos acidos 5-alquil-2-arilaminofenilaceticos y sus derivados
SA99191255B1 (ar) * 1998-11-30 2006-11-25 جي دي سيرل اند كو مركبات سيليكوكسيب celecoxib
AR030630A1 (es) * 2000-09-11 2003-08-27 Novartis Ag Composiciones farmaceuticas

Also Published As

Publication number Publication date
IL160375A0 (en) 2004-07-25
MXPA04001933A (es) 2004-06-15
CO5560554A2 (es) 2005-09-30
CY1106137T1 (el) 2011-06-08
MY137516A (en) 2009-02-27
NO20040860L (no) 2004-04-22
DE60211183D1 (de) 2006-06-08
US20070231382A1 (en) 2007-10-04
ZA200400877B (en) 2004-11-01
HUP0401429A2 (hu) 2004-11-29
KR20040031019A (ko) 2004-04-09
RU2329801C2 (ru) 2008-07-27
CA2456604C (en) 2011-02-08
ES2263813T3 (es) 2006-12-16
AU2002331094B2 (en) 2006-08-31
EP1425005B1 (en) 2006-05-03
WO2003020261A1 (en) 2003-03-13
PL367464A1 (en) 2005-02-21
CN100406008C (zh) 2008-07-30
JP2005520785A (ja) 2005-07-14
US20030114527A1 (en) 2003-06-19
DE60211183T2 (de) 2007-02-01
EP1425005A1 (en) 2004-06-09
NZ531342A (en) 2005-09-30
BR0212155A (pt) 2004-07-13
DK1425005T3 (da) 2006-09-04
CN1728993A (zh) 2006-02-01
PT1425005E (pt) 2006-09-29
KR100895551B1 (ko) 2009-04-29
JP4636796B2 (ja) 2011-02-23
HK1087336A1 (zh) 2006-10-13
ECSP044986A (es) 2004-04-28
ATE324883T1 (de) 2006-06-15
SI1425005T1 (sl) 2006-12-31
RU2004109920A (ru) 2005-04-20
AR036312A1 (es) 2004-08-25
CA2456604A1 (en) 2003-03-13

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