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LU90100I2 - Valsartan et ses dérivés pharmaceutiquement acceptables - Google Patents

Valsartan et ses dérivés pharmaceutiquement acceptables

Info

Publication number
LU90100I2
LU90100I2 LU90100C LU90100C LU90100I2 LU 90100 I2 LU90100 I2 LU 90100I2 LU 90100 C LU90100 C LU 90100C LU 90100 C LU90100 C LU 90100C LU 90100 I2 LU90100 I2 LU 90100I2
Authority
LU
Luxembourg
Prior art keywords
hydrocarbon
carboxy
cycloaliphatic
aliphatic hydrocarbon
optionally
Prior art date
Application number
LU90100C
Other languages
English (en)
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25684817&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU90100(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of LU90100I2 publication Critical patent/LU90100I2/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/38—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to acyclic carbon atoms and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/45—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/53—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring
    • C07C233/54—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of a saturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04—Five-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Magnetic Record Carriers (AREA)
  • Pyrrole Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Peptides Or Proteins (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Pyridine Compounds (AREA)
LU90100C 1990-02-19 1997-07-16 Valsartan et ses dérivés pharmaceutiquement acceptables LU90100I2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH51890 1990-02-19
CH223490 1990-07-05

Publications (1)

Publication Number Publication Date
LU90100I2 true LU90100I2 (fr) 1997-09-25

Family

ID=25684817

Family Applications (4)

Application Number Title Priority Date Filing Date
LU90100C LU90100I2 (fr) 1990-02-19 1997-07-16 Valsartan et ses dérivés pharmaceutiquement acceptables
LU90362C LU90362I2 (fr) 1990-02-19 1999-03-09 Valsartan en combinaison avec le hydrochlorothiazide (CO-DIOVAN)
LU91347C LU91347I2 (fr) 1990-02-19 2007-07-13 Valsartan et amlodipine, et leurs sels pharmaceutiquement acceptables
LU91676C LU91676I2 (fr) 1990-02-19 2010-04-07 "Valsartan, amlodipine et hydrochlorothiazide et leur sel pharmaceutiquement acceptable - EXFORGIE HCT"

Family Applications After (3)

Application Number Title Priority Date Filing Date
LU90362C LU90362I2 (fr) 1990-02-19 1999-03-09 Valsartan en combinaison avec le hydrochlorothiazide (CO-DIOVAN)
LU91347C LU91347I2 (fr) 1990-02-19 2007-07-13 Valsartan et amlodipine, et leurs sels pharmaceutiquement acceptables
LU91676C LU91676I2 (fr) 1990-02-19 2010-04-07 "Valsartan, amlodipine et hydrochlorothiazide et leur sel pharmaceutiquement acceptable - EXFORGIE HCT"

Country Status (26)

Country Link
US (2) US5399578A (fr)
EP (1) EP0443983B1 (fr)
JP (1) JP2749458B2 (fr)
KR (1) KR0171409B1 (fr)
AT (1) ATE134624T1 (fr)
AU (1) AU644844B2 (fr)
CA (2) CA2036427C (fr)
CY (2) CY1978A (fr)
DE (4) DE59107440D1 (fr)
DK (1) DK0443983T3 (fr)
ES (1) ES2084801T3 (fr)
FI (2) FI980787A7 (fr)
GR (1) GR3019155T3 (fr)
HK (1) HK219996A (fr)
HU (2) HU220073B (fr)
IE (1) IE71155B1 (fr)
IL (1) IL97219A (fr)
LU (4) LU90100I2 (fr)
LV (1) LV5773B4 (fr)
NL (3) NL970001I2 (fr)
NO (5) NO304023B1 (fr)
NZ (1) NZ237126A (fr)
PH (1) PH30484A (fr)
PT (1) PT96799B (fr)
SA (1) SA93140130A (fr)
UY (1) UY23835A1 (fr)

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* Cited by examiner, † Cited by third party
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