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LT4676B - 1-(3-aminoindazol-5-il)-3-fenilmetil-cikliniai karbamidai, naudojami kaip živ proteazės inhibitoriai - Google Patents

1-(3-aminoindazol-5-il)-3-fenilmetil-cikliniai karbamidai, naudojami kaip živ proteazės inhibitoriai Download PDF

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Publication number
LT4676B
LT4676B LT99-044A LT99044A LT4676B LT 4676 B LT4676 B LT 4676B LT 99044 A LT99044 A LT 99044A LT 4676 B LT4676 B LT 4676B
Authority
LT
Lithuania
Prior art keywords
compound
formula
hiv
combination
reverse transcriptase
Prior art date
Application number
LT99-044A
Other languages
English (en)
Lithuanian (lt)
Other versions
LT99044A (en
Inventor
James David Rodgers
Robert Frank Kaltenbach Iii
Original Assignee
Dupont Pharmaceuticals Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dupont Pharmaceuticals Company filed Critical Dupont Pharmaceuticals Company
Publication of LT99044A publication Critical patent/LT99044A/xx
Publication of LT4676B publication Critical patent/LT4676B/lt

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
LT99-044A 1996-11-08 1999-05-03 1-(3-aminoindazol-5-il)-3-fenilmetil-cikliniai karbamidai, naudojami kaip živ proteazės inhibitoriai LT4676B (lt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US74710496A 1996-11-08 1996-11-08

Publications (2)

Publication Number Publication Date
LT99044A LT99044A (en) 2000-02-25
LT4676B true LT4676B (lt) 2000-07-25

Family

ID=25003672

Family Applications (1)

Application Number Title Priority Date Filing Date
LT99-044A LT4676B (lt) 1996-11-08 1999-05-03 1-(3-aminoindazol-5-il)-3-fenilmetil-cikliniai karbamidai, naudojami kaip živ proteazės inhibitoriai

Country Status (4)

Country Link
AR (1) AR011008A1 (es)
HR (1) HRP970586A2 (es)
LT (1) LT4676B (es)
ZA (1) ZA979867B (es)

Non-Patent Citations (5)

* Cited by examiner, † Cited by third party
Title
H. MITSUYA ET AL.: "Stratagies for antiviral therapy", NATURE, 1987, pages 775
J. WELLINK, A. VAN KAMMEN: "Proteases involved in the processing of viral polyproteins. Brief review", ARCH VIROL., 1988, pages 1 - 26
KATOH I ET AL.: "Murine leukemia virus maturation: protease region required for conversion from "immature" to "mature" core form and for virus infectivity", VIROLOGY, 1985, pages 280, XP023058656, DOI: doi:10.1016/0042-6822(85)90161-8
S. CRAWFORD, S. P. GOFF: "A deletion mutation in the 5 part of the pol gene of Moloney murine leukemia virus blocks proteolytic processing of the gag and pol polyproteins", J VIROL., 1985, pages 899, XP000651443
S. ERICKSON-VIITANEN ET AL.: "Cleavage of HIV-1 gag Polyprotein Synthesized In Vitro: Sequential Cleavage by the Viral Protease", AIDS RESEARCH AND HUMAN RETROVIRUSES, 1989, pages 577

Also Published As

Publication number Publication date
LT99044A (en) 2000-02-25
HRP970586A2 (en) 1998-08-31
ZA979867B (en) 1999-05-03
AR011008A1 (es) 2000-08-02

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Effective date: 20011104