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IS8487A - Nefholssamsetning af rótigótíni - Google Patents

Nefholssamsetning af rótigótíni

Info

Publication number
IS8487A
IS8487A IS8487A IS8487A IS8487A IS 8487 A IS8487 A IS 8487A IS 8487 A IS8487 A IS 8487A IS 8487 A IS8487 A IS 8487A IS 8487 A IS8487 A IS 8487A
Authority
IS
Iceland
Prior art keywords
rotigotine
nasal composition
cyclodextrin
alpha
viscosity
Prior art date
Application number
IS8487A
Other languages
English (en)
Other versions
IS2310B (is
Inventor
Krämer Robert
Original Assignee
Schwarz Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schwarz Pharma Ag filed Critical Schwarz Pharma Ag
Publication of IS8487A publication Critical patent/IS8487A/is
Publication of IS2310B publication Critical patent/IS2310B/is

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IS8487A 2003-12-23 2006-05-26 Nefholssamsetning úr rótigótíni IS2310B (is)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP03029680A EP1547592A1 (en) 2003-12-23 2003-12-23 Intranasal formulation of rotigotine
PCT/EP2004/014626 WO2005063236A1 (en) 2003-12-23 2004-12-22 Intranasal formulation of rotigotine

Publications (2)

Publication Number Publication Date
IS8487A true IS8487A (is) 2006-05-26
IS2310B IS2310B (is) 2007-11-15

Family

ID=34530709

Family Applications (1)

Application Number Title Priority Date Filing Date
IS8487A IS2310B (is) 2003-12-23 2006-05-26 Nefholssamsetning úr rótigótíni

Country Status (27)

Country Link
US (1) US7683040B2 (is)
EP (2) EP1547592A1 (is)
JP (1) JP4430067B2 (is)
KR (1) KR100718760B1 (is)
CN (1) CN100374112C (is)
AT (1) ATE326961T1 (is)
AU (1) AU2004308641B2 (is)
BR (1) BRPI0407845A (is)
CA (1) CA2516400C (is)
CY (1) CY1105131T1 (is)
DE (1) DE602004000982T2 (is)
DK (1) DK1605932T3 (is)
EA (1) EA008005B1 (is)
ES (1) ES2262122T3 (is)
HR (1) HRP20060240T3 (is)
IL (1) IL170297A (is)
IS (1) IS2310B (is)
MX (1) MXPA05008909A (is)
NO (1) NO20054018L (is)
NZ (1) NZ541875A (is)
PL (1) PL1605932T3 (is)
PT (1) PT1605932E (is)
RS (1) RS50534B (is)
SI (1) SI1605932T1 (is)
UA (1) UA79196C2 (is)
WO (1) WO2005063236A1 (is)
ZA (1) ZA200506550B (is)

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DE10041478A1 (de) 2000-08-24 2002-03-14 Sanol Arznei Schwarz Gmbh Neue pharmazeutische Zusammensetzung
DE10041479A1 (de) * 2000-08-24 2002-03-14 Sanol Arznei Schwarz Gmbh Neue pharmazeutische Zusammensetzung zur Verabreichung von N-0923
US20040048779A1 (en) * 2002-05-06 2004-03-11 Erwin Schollmayer Use of rotigotine for treating the restless leg syndrome
DE10234673B4 (de) * 2002-07-30 2007-08-16 Schwarz Pharma Ag Heißschmelz-TTS zur Verabreichung von Rotigotin und Verfahren zu seiner Herstellung sowie Verwendung von Rotigotin bei der Herstellung eines TTS im Heißschmelzverfahren
US8246979B2 (en) 2002-07-30 2012-08-21 Ucb Pharma Gmbh Transdermal delivery system for the administration of rotigotine
US8211462B2 (en) * 2002-07-30 2012-07-03 Ucb Pharma Gmbh Hot-melt TTS for administering rotigotine
US8246980B2 (en) 2002-07-30 2012-08-21 Ucb Pharma Gmbh Transdermal delivery system
SI1426049T1 (en) 2002-12-02 2005-08-31 Sanol Arznei Schwarz Gmbh Iontophoretic delivery of rotigotine for the treatment of Parkinson's disease
DE10261696A1 (de) 2002-12-30 2004-07-15 Schwarz Pharma Ag Vorrichtung zur transdermalen Verabreichung von Rotigotin-Base
DE10334188B4 (de) * 2003-07-26 2007-07-05 Schwarz Pharma Ag Verwendung von Rotigotin zur Behandlung von Depressionen
DE10359528A1 (de) * 2003-12-18 2005-07-28 Schwarz Pharma Ag (S)-2-N-Propylamino-5-hydroxytetralin als D3-agonistisches Therapeutikum
EP1547592A1 (en) 2003-12-23 2005-06-29 Schwarz Pharma Ag Intranasal formulation of rotigotine
DE10361258A1 (de) * 2003-12-24 2005-07-28 Schwarz Pharma Ag Verwendung von substituierten 2-Aminotetralinen zur vorbeugenden Behandlung von Morbus Parkinson
US20050197385A1 (en) * 2004-02-20 2005-09-08 Schwarz Pharma Ag Use of rotigotine for treatment or prevention of dopaminergic neuron loss
DE102004014841B4 (de) * 2004-03-24 2006-07-06 Schwarz Pharma Ag Verwendung von Rotigotin zur Behandlung und Prävention des Parkinson-Plus-Syndroms
TWI392670B (zh) * 2006-06-22 2013-04-11 Ucb Pharma Gmbh 經取代的２-胺基萘滿之於製造用於預防、減緩及／或治療各種類型疼痛之藥物上的用途
EP1987815A1 (en) * 2007-05-04 2008-11-05 Schwarz Pharma Ag Oronasopharyngeally deliverable pharmaceutical compositions of dopamine agonists for the prevention and/or treatment of restless limb disorders
AU2008328920B2 (en) 2007-11-28 2013-09-12 Ucb Pharma Gmbh Polymorphic form of Rotigotine
US8580801B2 (en) 2008-07-23 2013-11-12 Robert I. Henkin Phosphodiesterase inhibitor treatment
EP2281559A1 (en) 2009-06-26 2011-02-09 UCB Pharma GmbH Pharmaceutical composition comprising rotigotine salts (acid or Na), especially for iontophoresis
PT3257504T (pt) 2009-12-22 2024-09-03 Ucb Biopharma Sprl Polivinilpirrolidona para a estabilização de uma dispersão sólida da forma não cristalina de rotigotina
EP2559435A1 (en) 2011-08-19 2013-02-20 UCB Pharma GmbH Rotigotine in the treatment of hemispatial neglect, stroke and deficits following stroke
DE102012013439A1 (de) 2012-07-03 2014-01-23 Alfred E. Tiefenbacher (Gmbh & Co. Kg) Transdermales therapeutisches System umfassend Rotigotin und Kristallisationsinhibitor
WO2013075823A1 (en) 2011-11-22 2013-05-30 Alfred E. Tiefenbacher (Gmbh & Co. Kg) Transdermal therapeutic system comprising rotigotine and crystallization inhibitor
DE102012013421A1 (de) 2012-07-03 2014-01-09 Alfred E. Tiefenbacher (Gmbh & Co. Kg) Transdermales therapeutisches System (TTS) mit Rotigotin
CN103768043B (zh) * 2012-10-22 2015-12-09 苏州药明康德新药开发股份有限公司 采用羟丙基-β-环糊精配制四氢化萘类化合物均一稳定溶液的方法
TW201431570A (zh) 2012-11-22 2014-08-16 Ucb Pharma Gmbh 用於經皮投服羅替戈汀（Ｒｏｔｉｇｏｔｉｎｅ）之多天式貼片
CA2916183C (en) 2013-07-03 2022-03-29 Lts Lohmann Therapie-Systeme Ag Transdermal therapeutic system with electronic component
WO2015126944A1 (en) 2014-02-18 2015-08-27 Henkin Robert I Methods and compositions for diagnosing and treating loss and/or distortion of taste or smell
ES2924899T3 (es) 2014-05-20 2022-10-11 Lts Lohmann Therapie Systeme Ag Sistema de administración transdérmica que contiene rotigotina
CN106456567A (zh) 2014-05-20 2017-02-22 Lts勒曼治疗系统股份公司 在经皮递送系统中调节活性剂释放的方法
JP6599899B2 (ja) 2014-05-20 2019-10-30 エルテーエス ローマン テラピー−ジステーメ アーゲー 界面介在物を含む経皮送達システム
US9956201B2 (en) 2014-07-21 2018-05-01 Spriaso Llc Compositions comprising bioreversible derivatives of hydroxy N-substituted-2-aminotetralins, and related dosage forms
CN110917125B (zh) * 2020-01-02 2022-08-12 安徽中医药大学 一种罗替戈汀鼻用胶束温敏凝胶的制备方法
JP2025502075A (ja) * 2022-01-06 2025-01-24 シラノ セラピューティクス， インコーポレイテッド パーキンソン病治療剤の改善された鼻投与
CN120053353A (zh) * 2024-05-31 2025-05-30 纳索菲德(上海)制药技术有限公司 一种巴氯芬鼻脑递释组合物

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KR20070045254A (ko) 2004-08-02 2007-05-02 슈바르츠 파르마 악티엔게젤샤프트 인돌리진 카르복사미드 및 그 아자 및 디아자유도체
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Also Published As

Publication number Publication date
DE602004000982T2 (de) 2007-05-10
US7683040B2 (en) 2010-03-23
ZA200506550B (en) 2006-05-31
AU2004308641B2 (en) 2006-10-26
MXPA05008909A (es) 2005-10-05
EA008005B1 (ru) 2007-02-27
EP1605932B1 (en) 2006-05-24
IS2310B (is) 2007-11-15
PL1605932T3 (pl) 2006-09-29
KR100718760B1 (ko) 2007-05-15
UA79196C2 (en) 2007-05-25
JP4430067B2 (ja) 2010-03-10
IL170297A (en) 2010-06-30
NZ541875A (en) 2008-08-29
DE602004000982D1 (de) 2006-06-29
RS50534B (sr) 2010-05-07
JP2006526004A (ja) 2006-11-16
HRP20060240T3 (hr) 2007-05-31
SI1605932T1 (sl) 2006-08-31
CN1777422A (zh) 2006-05-24
ES2262122T3 (es) 2006-11-16
NO20054018L (no) 2005-08-30
ATE326961T1 (de) 2006-06-15
EP1547592A1 (en) 2005-06-29
CA2516400A1 (en) 2005-07-14
DK1605932T3 (da) 2006-09-18
CA2516400C (en) 2009-10-27
WO2005063236A1 (en) 2005-07-14
BRPI0407845A (pt) 2006-02-14
CY1105131T1 (el) 2009-11-04
HK1083596A1 (en) 2006-07-07
US20070191308A1 (en) 2007-08-16
AU2004308641A1 (en) 2005-07-14
CN100374112C (zh) 2008-03-12
EP1605932A1 (en) 2005-12-21
PT1605932E (pt) 2006-08-31
KR20060040578A (ko) 2006-05-10
EA200501159A1 (ru) 2006-02-24

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