IS7733A - 1,2,4-Oxadíazól sem eru beinar fyrir hvatavirkjandi glútamatviðtaka-5 - Google Patents

1,2,4-Oxadíazól sem eru beinar fyrir hvatavirkjandi glútamatviðtaka-5

Info

Publication number: IS7733A
Authority: IS; Iceland
Prior art keywords: oxadiazole; direct; glutamate receptor; catalytic glutamate; catalytic
Prior art date: 2002-08-09

Application number

IS7733A

Other languages

English (en)

Inventor

Wensbo David

Xin Tao

Stefanac Tomislav

Arora Jalaj

Edwards Louise

Benjamin Isaac Methvin

Slassi Abdelmalik

M. Stormann Thomas

A. Mcleod Donald

Kers Annika

Malmberg Johan

Oscarsson Karin

Gyback Helena

Johansson Martin

Mindis Alexander

Waldman Magnus

Yngve Ulrika

Osterwall Christoffer

Original Assignee

Astrazeneca Ab

Nps Pharmaceuticals, Inc.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-08-09

Filing date

2005-03-09

Publication date

2005-03-09

2005-03-09 Application filed by Astrazeneca Ab, Nps Pharmaceuticals, Inc. filed Critical Astrazeneca Ab

2005-03-09 Publication of IS7733A publication Critical patent/IS7733A/is

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Psychiatry (AREA)
Physical Education & Sports Medicine (AREA)
Psychology (AREA)
Hospice & Palliative Care (AREA)
Cardiology (AREA)
Ophthalmology & Optometry (AREA)
Heart & Thoracic Surgery (AREA)
Toxicology (AREA)
Immunology (AREA)
Orthopedic Medicine & Surgery (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

IS7733A 2002-08-09 2005-03-09 1,2,4-Oxadíazól sem eru beinar fyrir hvatavirkjandi glútamatviðtaka-5 IS7733A (is)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US40204002P	2002-08-09	2002-08-09
PCT/US2003/024846 WO2004014881A2 (en)	2002-08-09	2003-08-08	'1,2,4'oxadiazoles as modulators of metabotropic glutamate receptor-5

Publications (1)

Publication Number	Publication Date
IS7733A true IS7733A (is)	2005-03-09

Family

ID=31715777

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IS7733A IS7733A (is)	2002-08-09	2005-03-09	1,2,4-Oxadíazól sem eru beinar fyrir hvatavirkjandi glútamatviðtaka-5

Country Status (20)

Country	Link
US (2)	US20040152699A1 (is)
EP (1)	EP1529045A2 (is)
JP (2)	JP4637578B2 (is)
KR (1)	KR20050033070A (is)
CN (2)	CN101723941A (is)
AR (1)	AR040847A1 (is)
AU (1)	AU2003259068B2 (is)
BR (1)	BR0313265A (is)
CA (1)	CA2494987C (is)
IL (1)	IL166510A0 (is)
IS (1)	IS7733A (is)
MX (1)	MXPA05001594A (is)
NO (1)	NO20051225L (is)
NZ (1)	NZ538225A (is)
PL (1)	PL375256A1 (is)
RU (1)	RU2352568C9 (is)
TW (1)	TWI341314B (is)
UA (1)	UA87653C2 (is)
WO (1)	WO2004014881A2 (is)
ZA (1)	ZA200500886B (is)

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2003
- 2003-08-08 JP JP2004527872A patent/JP4637578B2/ja not_active Expired - Fee Related
- 2003-08-08 AR AR20030102891A patent/AR040847A1/es unknown
- 2003-08-08 UA UAA200501100A patent/UA87653C2/ru unknown
- 2003-08-08 PL PL03375256A patent/PL375256A1/xx unknown
- 2003-08-08 AU AU2003259068A patent/AU2003259068B2/en not_active Ceased
- 2003-08-08 MX MXPA05001594A patent/MXPA05001594A/es active IP Right Grant
- 2003-08-08 NZ NZ538225A patent/NZ538225A/en not_active IP Right Cessation
- 2003-08-08 TW TW092121880A patent/TWI341314B/zh not_active IP Right Cessation
- 2003-08-08 US US10/637,012 patent/US20040152699A1/en not_active Abandoned
- 2003-08-08 CN CN200910208474A patent/CN101723941A/zh active Pending
- 2003-08-08 CN CNA038238454A patent/CN1894241A/zh active Pending
- 2003-08-08 KR KR1020057002101A patent/KR20050033070A/ko not_active Ceased
- 2003-08-08 RU RU2005106844/04A patent/RU2352568C9/ru not_active IP Right Cessation
- 2003-08-08 WO PCT/US2003/024846 patent/WO2004014881A2/en not_active Ceased
- 2003-08-08 EP EP03785036A patent/EP1529045A2/en not_active Withdrawn
- 2003-08-08 IL IL16651003A patent/IL166510A0/xx unknown
- 2003-08-08 BR BR0313265-0A patent/BR0313265A/pt not_active Application Discontinuation
- 2003-08-08 CA CA2494987A patent/CA2494987C/en not_active Expired - Fee Related
2005
- 2005-01-31 ZA ZA200500886A patent/ZA200500886B/en unknown
- 2005-03-09 NO NO20051225A patent/NO20051225L/no unknown
- 2005-03-09 IS IS7733A patent/IS7733A/is unknown
- 2005-11-14 US US11/274,611 patent/US7456200B2/en not_active Expired - Fee Related
2010
- 2010-06-14 JP JP2010135508A patent/JP2010248214A/ja active Pending

Also Published As

Publication number	Publication date
US20060122397A1 (en)	2006-06-08
IL166510A0 (en)	2006-01-15
AR040847A1 (es)	2005-04-20
RU2352568C9 (ru)	2009-06-27
AU2003259068B2 (en)	2009-07-02
CA2494987A1 (en)	2004-02-19
US7456200B2 (en)	2008-11-25
NZ538225A (en)	2008-05-30
JP2010248214A (ja)	2010-11-04
AU2003259068A1 (en)	2004-02-25
TW200413361A (en)	2004-08-01
RU2005106844A (ru)	2005-08-27
EP1529045A2 (en)	2005-05-11
JP2006503009A (ja)	2006-01-26
WO2004014881A2 (en)	2004-02-19
PL375256A1 (en)	2005-11-28
CN1894241A (zh)	2007-01-10
BR0313265A (pt)	2005-07-05
CA2494987C (en)	2012-04-17
UA87653C2 (en)	2009-08-10
ZA200500886B (en)	2006-07-26
MXPA05001594A (es)	2005-09-20
JP4637578B2 (ja)	2011-02-23
TWI341314B (en)	2011-05-01
RU2352568C2 (ru)	2009-04-20
KR20050033070A (ko)	2005-04-08
CN101723941A (zh)	2010-06-09
WO2004014881A3 (en)	2004-05-27
WO2004014881B1 (en)	2004-07-15
NO20051225L (no)	2005-05-09
US20040152699A1 (en)	2004-08-05

Publication	Publication Date	Title
IS7733A (is)	2005-03-09	1,2,4-Oxadíazól sem eru beinar fyrir hvatavirkjandi glútamatviðtaka-5
CY2014041I1 (el)	2016-07-27	2,3-διυδρο-6-νιτροϊμιδαζο 2,1 -b-οξαζολια
DK2308855T3 (da)	2013-01-28	2,4-Diaminopyrimidinderivater
NO20052993D0 (no)	2005-06-17	4,5-diaryltiazolderivater som CB-1 ligander.
DE60225341D1 (de)	2008-04-10	Neue 1,2,4-triazolverbindung
NO20053246D0 (no)	2005-07-01	Kondensert 1,3-dihydroimidazol-ringforbindelse.
ATE326467T1 (de)	2006-06-15	Imidazo 1,2-aöpyridine
DE60313440D1 (de)	2007-06-06	Gasversorgungsvorrichtung
MA27306A1 (fr)	2005-05-02	Ligands des recepteurs de la melanocortine.
ITBO20020284A1 (it)	2003-11-14	Macchina opercolatrice
IL165747A0 (en)	2006-01-15	Crystalline 2,5-dione-3-(1-methyl-1h-indol-3-yl)-4-Ä1-(pyridin-2-ylmethyl)piperidin-4-ylÜ-1h-indol-3-ylÜ-1h-pyrrole mono-hydrochloride
IS7609A (is)	2004-12-22	2,5-tvíútskipt 3-merkaptópentansýra
ITTO20020157A0 (it)	2002-02-25	Macchina depallettizzatrice.
NO20052975D0 (no)	2005-06-17	Nye 2',5'-oligoadenylsyreanaloger.
DE50304384D1 (de)	2006-09-07	Anordnung zum ansteuern von rückhaltemitteln
ITPD20020092A1 (it)	2003-10-13	Dispositivo di sicurezza a termocoppia, particolarmente per bruciatori a gas.
NO20044413L (no)	2004-10-18	1,2-Dihydropyrazol-3-oner som cytokinmediatorer
NO20044405L (no)	2004-10-15	Neurotensinaktive 2,3-diaryl-pyrazolidin derivater
FI20022023A7 (fi)	2004-05-14	Menetelmä kiinnirullaimen ohjaamiseksi
ITMI20032205A1 (it)	2004-05-28	Procedimento per l'esercizio di un motore termico.
NO20053110D0 (no)	2005-06-24	2-oksyamino-1-cyklopenten-1-nitriler som materialbeskyttelsesmidler.
EP1559708A4 (en)	2006-07-19	2,2-DISUBSTITUTED 1A, 25-DIHYDROXY-19-NORVITAMINE D DERIVATIVE
ES1051892Y (es)	2003-02-16	Bolsa termica.
LU90940B1 (de)	2004-02-02	Gasversorgungseinheit
ES1051900Y (es)	2003-02-16	Util para el tensado de alambre.