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IS1822B - Glýkósamstæður, lyf sem innihalda þær, og notkun glýkósamstæðnanna við framleiðslu lyfja - Google Patents

Glýkósamstæður, lyf sem innihalda þær, og notkun glýkósamstæðnanna við framleiðslu lyfja

Info

Publication number
IS1822B
IS1822B IS4562A IS4562A IS1822B IS 1822 B IS1822 B IS 1822B IS 4562 A IS4562 A IS 4562A IS 4562 A IS4562 A IS 4562A IS 1822 B IS1822 B IS 1822B
Authority
IS
Iceland
Prior art keywords
glycosides
drugs
manufacture
drugs containing
cytostatics
Prior art date
Application number
IS4562A
Other languages
English (en)
Other versions
IS4562A (is
Inventor
Lerchen Hans-Georg
Von Dem Bruch Karsten
Petersen Uwe
Baumgarten Jörg
Piel Norbert
Antonicek Horst-Peter
Weichel Walter
Sperzel Michael
Dieter Bremm Klaus
Original Assignee
Bayer Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Aktiengesellschaft filed Critical Bayer Aktiengesellschaft
Publication of IS4562A publication Critical patent/IS4562A/is
Publication of IS1822B publication Critical patent/IS1822B/is

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/02Halogenated hydrocarbons
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/203Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/001Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence having less than 12 amino acids and not being part of a ring structure
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biotechnology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Medicinal Preparation (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Other Investigation Or Analysis Of Materials By Electrical Means (AREA)
  • Pyrane Compounds (AREA)
  • Steroid Compounds (AREA)
  • Peptides Or Proteins (AREA)
IS4562A 1995-04-04 1997-09-18 Glýkósamstæður, lyf sem innihalda þær, og notkun glýkósamstæðnanna við framleiðslu lyfja IS1822B (is)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19512484A DE19512484A1 (de) 1995-04-04 1995-04-04 Kohlenhydratmodifizierte Cytostatika
PCT/EP1996/001279 WO1996031532A1 (de) 1995-04-04 1996-03-22 Kohlenhydratmodifizierte cytostatika

Publications (2)

Publication Number Publication Date
IS4562A IS4562A (is) 1997-09-18
IS1822B true IS1822B (is) 2002-10-01

Family

ID=7758679

Family Applications (1)

Application Number Title Priority Date Filing Date
IS4562A IS1822B (is) 1995-04-04 1997-09-18 Glýkósamstæður, lyf sem innihalda þær, og notkun glýkósamstæðnanna við framleiðslu lyfja

Country Status (27)

Country Link
US (1) US6271342B1 (is)
EP (1) EP0819135B1 (is)
JP (1) JPH11502860A (is)
KR (1) KR19980703591A (is)
CN (1) CN1185786A (is)
AT (1) ATE186738T1 (is)
AU (1) AU713466B2 (is)
BG (1) BG63048B1 (is)
BR (1) BR9604825A (is)
CA (1) CA2217164A1 (is)
CZ (1) CZ291098B6 (is)
DE (2) DE19512484A1 (is)
DK (1) DK0819135T3 (is)
EE (1) EE03619B1 (is)
ES (1) ES2140078T3 (is)
GR (1) GR3032605T3 (is)
HU (1) HUP9800513A3 (is)
IS (1) IS1822B (is)
MX (1) MX9707613A (is)
NO (1) NO974564L (is)
NZ (1) NZ305855A (is)
PL (1) PL183574B1 (is)
RU (1) RU2170234C2 (is)
SK (1) SK281785B6 (is)
TW (1) TW384290B (is)
UA (1) UA61054C2 (is)
WO (1) WO1996031532A1 (is)

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CA2267328A1 (en) * 1996-09-30 1998-04-09 Bayer Aktiengesellschaft Glycoconjugates from modified camptothecin derivates (20-o-linkage)
DE19640970A1 (de) * 1996-10-04 1998-04-16 Bayer Ag Modifizierte Cytostatika
JP3101710B2 (ja) 1997-02-28 2000-10-23 工業技術院長 硫酸化オリゴ糖化合物
ID23424A (id) * 1997-05-14 2000-04-20 Bayer Ag Glikokonjugat dari 20(s)-kamptotesin
US6387928B1 (en) 1997-09-15 2002-05-14 The Procter & Gamble Co. Antimicrobial quinolones, their compositions and uses
AU735186B2 (en) 1997-09-15 2001-07-05 Warner Chilcott Company, Llc Antimicrobial quinolones, their compositions and uses
US6613879B1 (en) * 1999-05-14 2003-09-02 Boehringer Ingelheim Pharma Kg FAP-activated anti-tumour compounds
DE10005275A1 (de) * 2000-02-07 2001-08-09 Bayer Ag Neuartige Glycokonjugate
US7220824B1 (en) * 2000-08-28 2007-05-22 Bayer Aktiengesellschaft Integrin-mediated drug targeting
EP1219634A1 (en) * 2000-12-27 2002-07-03 Bayer Aktiengesellschaft Cytostatic-glycoconjugates having specifically cleavable peptidic linking units
EP1238678A1 (en) * 2001-03-08 2002-09-11 Bayer Aktiengesellschaft Enzyme-activated cytostatic conjugates with integrin ligands
US20050037423A1 (en) * 2001-11-09 2005-02-17 Bayer Healthcare Ag Isotopycally coded affinity marker 2
US7199149B2 (en) * 2003-10-01 2007-04-03 Bristol Myers Squibb Company Monocyclic and bicyclic lactams as factor Xa inhibitors
EP1718677B1 (en) 2003-12-19 2012-04-18 Genentech, Inc. Monovalent antibody fragments useful as therapeutics
EP1999125A2 (en) 2006-03-28 2008-12-10 The Procter and Gamble Company A coupling process for preparing quinolone intermediates
EP1999106B1 (en) 2006-03-28 2012-06-27 TaiGen Biotechnology Co., Ltd. A hydride reduction process for preparing quinolone intermediates
AU2007230630B2 (en) 2006-03-28 2012-12-20 Taigen Biotechnology Co., Ltd Malate salts, and polymorphs of (3S,5S)-7-[3-amino-5-methyl-piperidinyl]-1-cyclopropyl-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid
HK1245280A1 (zh) 2015-01-06 2018-08-24 Immunovaccine Technologies Inc. 脂质a模拟物、其制备方法和用途
SMT202400223T1 (it) 2015-11-25 2024-07-09 Ligachem Biosciences Inc Coniugati comprendenti gruppi autoimmolativi e metodi correlati ad essi
KR102847350B1 (ko) 2015-11-25 2025-08-19 주식회사 리가켐바이오사이언스 분지된 링커를 포함하는 항체-약물 접합체 및 이의 제조방법
JP7664680B2 (ja) 2017-03-29 2025-04-18 リガケム バイオサイエンシズ, インク. ピロロベンゾジアゼピン二量体前駆体及びそのリガンド-リンカーコンジュゲート化合物
SG11202010443WA (en) 2018-05-09 2020-11-27 Legochem Biosciences Inc Compositions and methods related to anti-cd19 antibody drug conjugates
KR20210028544A (ko) 2019-09-04 2021-03-12 주식회사 레고켐 바이오사이언스 인간 ror1에 대한 항체를 포함하는 항체 약물 접합체 및 이의 용도
JP2024537169A (ja) * 2021-10-06 2024-10-10 サムヤン コーポレイション 飽和フロジオキシン誘導体化合物及びその二次電池用添加剤としての使用

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Also Published As

Publication number Publication date
EE9700258A (et) 1998-04-15
EP0819135A1 (de) 1998-01-21
BR9604825A (pt) 1999-01-05
SK281785B6 (sk) 2001-07-10
IS4562A (is) 1997-09-18
UA61054C2 (en) 2003-11-17
PL322681A1 (en) 1998-02-16
BG63048B1 (bg) 2001-02-28
HUP9800513A2 (hu) 1998-06-29
AU5397696A (en) 1996-10-23
GR3032605T3 (en) 2000-05-31
RU2170234C2 (ru) 2001-07-10
DE59603678D1 (de) 1999-12-23
AU713466B2 (en) 1999-12-02
SK134597A3 (en) 1998-05-06
HUP9800513A3 (en) 1998-09-28
PL183574B1 (pl) 2002-06-28
MX9707613A (es) 1997-12-31
CZ314397A3 (cs) 1998-01-14
ES2140078T3 (es) 2000-02-16
US6271342B1 (en) 2001-08-07
CA2217164A1 (en) 1996-10-10
KR19980703591A (ko) 1998-11-05
NO974564D0 (no) 1997-10-02
NZ305855A (en) 1999-11-29
ATE186738T1 (de) 1999-12-15
DE19512484A1 (de) 1996-10-17
EE03619B1 (et) 2002-02-15
BG101892A (en) 1998-05-29
CN1185786A (zh) 1998-06-24
NO974564L (no) 1997-11-25
CZ291098B6 (cs) 2002-12-11
DK0819135T3 (da) 2000-05-08
WO1996031532A1 (de) 1996-10-10
JPH11502860A (ja) 1999-03-09
EP0819135B1 (de) 1999-11-17
TW384290B (en) 2000-03-11

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