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IL161915A0 - Salt forms of methoxy-N-(3-(4-(3-methyl-pyridin-3-yloxyl)-phenylamino)- quinazolin-6-yl)-allyl)-acetamide, its prepar - Google Patents

Salt forms of methoxy-N-(3-(4-(3-methyl-pyridin-3-yloxyl)-phenylamino)- quinazolin-6-yl)-allyl)-acetamide, its prepar

Info

Publication number
IL161915A0
IL161915A0 IL16191502A IL16191502A IL161915A0 IL 161915 A0 IL161915 A0 IL 161915A0 IL 16191502 A IL16191502 A IL 16191502A IL 16191502 A IL16191502 A IL 16191502A IL 161915 A0 IL161915 A0 IL 161915A0
Authority
IL
Israel
Prior art keywords
yloxyl
prepar
quinazolin
phenylamino
pyridin
Prior art date
Application number
IL16191502A
Other languages
English (en)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of IL161915A0 publication Critical patent/IL161915A0/xx

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Ophthalmology & Optometry (AREA)
  • Oncology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Reproductive Health (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL16191502A 2001-12-12 2002-11-11 Salt forms of methoxy-N-(3-(4-(3-methyl-pyridin-3-yloxyl)-phenylamino)- quinazolin-6-yl)-allyl)-acetamide, its prepar IL161915A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US34088501P 2001-12-12 2001-12-12
PCT/IB2002/004708 WO2003050108A1 (fr) 2001-12-12 2002-11-11 Formes salines de e-2-methoxy-n-(3-{4-[3-methl-4-(6-methylpyridin-3-yloxy)-phenylamino]-quinazolin-6-yl}-allyl)-acetamide

Publications (1)

Publication Number Publication Date
IL161915A0 true IL161915A0 (en) 2005-11-20

Family

ID=23335337

Family Applications (1)

Application Number Title Priority Date Filing Date
IL16191502A IL161915A0 (en) 2001-12-12 2002-11-11 Salt forms of methoxy-N-(3-(4-(3-methyl-pyridin-3-yloxyl)-phenylamino)- quinazolin-6-yl)-allyl)-acetamide, its prepar

Country Status (34)

Country Link
US (1) US6844349B2 (fr)
EP (1) EP1456199A1 (fr)
JP (1) JP4202926B2 (fr)
KR (1) KR20040065259A (fr)
CN (1) CN1608062A (fr)
AP (1) AP2004003059A0 (fr)
AR (1) AR037772A1 (fr)
AU (1) AU2002366581A1 (fr)
BR (1) BR0214876A (fr)
CA (1) CA2469889A1 (fr)
DO (1) DOP2002000544A (fr)
EA (1) EA007412B1 (fr)
EC (1) ECSP045148A (fr)
GE (1) GEP20063872B (fr)
GT (1) GT200200272A (fr)
HR (1) HRP20040530A2 (fr)
HU (1) HUP0402662A2 (fr)
IL (1) IL161915A0 (fr)
IS (1) IS7227A (fr)
MA (1) MA27095A1 (fr)
MX (1) MXPA04005678A (fr)
NO (1) NO20042925L (fr)
NZ (1) NZ532436A (fr)
OA (1) OA12735A (fr)
PA (1) PA8561401A1 (fr)
PE (1) PE20030716A1 (fr)
PL (1) PL370858A1 (fr)
RS (1) RS46404A (fr)
TN (1) TNSN04112A1 (fr)
TW (1) TW200301103A (fr)
UA (1) UA75482C2 (fr)
UY (1) UY27572A1 (fr)
WO (1) WO2003050108A1 (fr)
ZA (1) ZA200402995B (fr)

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EP1521747B1 (fr) 2002-07-15 2018-09-05 Symphony Evolution, Inc. Modulateurs de kinase de type recepteur et procedes d'utilisation
RU2005119172A (ru) * 2002-12-18 2006-01-20 Пфайзер Продактс Инк. (Us) Производные 4-анилинхиназолина для лечения патологического роста клеток
RU2005122659A (ru) * 2002-12-19 2006-01-20 Пфайзер Продактс Инк. (Us) Комплексы е-2-метокси-n-(3-{4-[3-метил-4-(6-метилпиридин-3-илокси) фениламино] хиназолин-6-ил} аллил) ацетамида, способ получения и применения указанных комплексов
US7429565B2 (en) 2003-04-25 2008-09-30 Gilead Sciences, Inc. Antiviral phosphonate analogs
KR20060037447A (ko) * 2003-08-18 2006-05-03 화이자 프로덕츠 인크. erbB2 항암제에 대한 투약 스케쥴
ES2925655T3 (es) 2003-09-26 2022-10-19 Exelixis Inc Moduladores c-Met y métodos de uso
CA2543201C (fr) * 2003-10-27 2010-12-21 Merck & Co., Inc. Sel de succinate de ((ir, 3s)-3-isopropyl-3-{ [3-(trifluoromethyl)-7, 8-dihydro-1, 6-naphthyridin-6 (5h)- yl] carbonyl} cyclopentyl) [(3s, 4s)-3-methoxytetrahydro-2h-pyran-4-yl] amine, sa composition et son utilisation dans le traitemetn des maladies inflammatoires
US20050192298A1 (en) * 2004-02-27 2005-09-01 Pfizer Inc Crystal forms of E-2-Methoxy-N-(3-{4-[3-methyl-4-(6-methyl-pyridin-3-yloxy)-phenylamino]-quinazolin-6-yl}-allyl)-acetamide
WO2005121124A1 (fr) * 2004-06-07 2005-12-22 Pfizer Products Inc. Complexes de e-2-methoxy-n-(3-{4-[3-methyl-pyridin-3-yloxy)-phenylamino]-quinazolin-6-yl}-allyl)-acetamide et procedes de preparation de ces derniers
HRP20070078A2 (hr) 2004-07-27 2007-05-31 Gilead Sciences Fosfonatni analozi spojeva koji inhibiraju hiv
EP1896451A2 (fr) * 2005-06-03 2008-03-12 Pfizer Products Incorporated Derives bicycliques pour le traitement de croissance cellulaire anormale
CA2610661A1 (fr) * 2005-06-03 2006-12-07 Pfizer Products Inc. Combinaisons d'inhibiteurs d'erbb2 avec d'autres agents therapeutiques dans le traitement du cancer
PT2020996E (pt) * 2006-05-16 2012-02-20 Gilead Sciences Inc Método e composições para tratar neoplasias malignas hematológicas
CA2673097A1 (fr) 2006-12-12 2008-06-19 Takeda Pharmaceutical Company Limited Compose heterocyclique condense
CN101611029B (zh) * 2006-12-21 2014-09-10 辉瑞产品公司 2-((4-(1-甲基-4-(吡啶-4-基)-1h-吡唑-3-基)苯氧基)甲基)喹啉的琥珀酸盐
WO2008124824A1 (fr) * 2007-04-10 2008-10-16 Myriad Genetics, Inc. Doses et méthodes de traitement du cancer
TW200944528A (en) 2008-03-12 2009-11-01 Takeda Pharmaceutical Fused heterocyclic compound
PT2307435E (pt) * 2008-07-08 2012-09-19 Gilead Sciences Inc Sais de compostos inibidores de vih
KR20250123237A (ko) 2009-01-16 2025-08-14 엑셀리시스, 인코포레이티드 암의 치료를 위한 n-(4-{〔6,7-비스(메틸옥시)퀴놀린-4-일〕옥시}페닐)-n'-(4-플루오로페닐)사이클로프로판-1,1-디카르복사미드의 말산염 및 그 결정형
UA108618C2 (uk) 2009-08-07 2015-05-25 Застосування c-met-модуляторів в комбінації з темозоломідом та/або променевою терапією для лікування раку
WO2011153050A1 (fr) 2010-06-02 2011-12-08 The Trustees Of The University Of Pennsylvania Méthodes et utilisation de composés qui se lient au complexe du récepteur her2/neu
US8993634B2 (en) 2010-06-02 2015-03-31 The Trustees Of The University Of Pennsylvania Methods and use of compounds that bind to Her2/neu receptor complex
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WO2019027920A1 (fr) 2017-08-01 2019-02-07 Gilead Sciences, Inc. Formes cristallines d'éthyl ((s)-((((2r,5r)-5-(6-amino-9h-purin-9-yl)-4-fluoro-2,5-dihydrofuran-2-yl)oxy)méthyl)(phénoxy)phosphoryl)-l-alaninate (gs-9131) pour le traitement d'infections virales
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JP4044839B2 (ja) * 2000-06-22 2008-02-06 ファイザー・プロダクツ・インク 異常細胞増殖を治療するための置換2環式誘導体

Also Published As

Publication number Publication date
EA200400674A1 (ru) 2004-10-28
DOP2002000544A (es) 2003-06-16
UA75482C2 (en) 2006-04-17
OA12735A (en) 2006-06-29
TNSN04112A1 (fr) 2006-06-01
US20030158217A1 (en) 2003-08-21
NO20042925L (no) 2004-09-07
MA27095A1 (fr) 2004-12-20
HUP0402662A2 (hu) 2005-05-30
MXPA04005678A (es) 2004-12-06
JP4202926B2 (ja) 2008-12-24
PA8561401A1 (es) 2005-02-04
AU2002366581A1 (en) 2003-06-23
GEP20063872B (en) 2006-07-10
WO2003050108A8 (fr) 2003-12-18
RS46404A (sr) 2006-10-27
EA007412B1 (ru) 2006-10-27
BR0214876A (pt) 2004-12-28
PL370858A1 (en) 2005-05-30
PE20030716A1 (es) 2003-08-29
KR20040065259A (ko) 2004-07-21
AR037772A1 (es) 2004-12-01
UY27572A1 (es) 2003-07-31
CN1608062A (zh) 2005-04-20
ZA200402995B (en) 2005-04-20
GT200200272A (es) 2003-12-12
WO2003050108A1 (fr) 2003-06-19
HRP20040530A2 (en) 2004-10-31
AP2004003059A0 (en) 2004-06-30
US6844349B2 (en) 2005-01-18
IS7227A (is) 2004-04-19
JP2005511744A (ja) 2005-04-28
NZ532436A (en) 2006-01-27
ECSP045148A (es) 2004-07-23
TW200301103A (en) 2003-07-01
EP1456199A1 (fr) 2004-09-15
CA2469889A1 (fr) 2003-06-19

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