IL166405A0 - 3-z-Ä1-4-(n-((4-methyl-piperazin-1-yl)methylcarbonyl)-n-methyl-aminoanilo)-1-phenyl-methyleneÜ-6-methyxycarbonyl-2-indoline-monoethanesulphonate and the use thereof as a pharmaceutical composition - Google Patents

3-z-Ä1-4-(n-((4-methyl-piperazin-1-yl)methylcarbonyl)-n-methyl-aminoanilo)-1-phenyl-methyleneÜ-6-methyxycarbonyl-2-indoline-monoethanesulphonate and the use thereof as a pharmaceutical composition

Info

Publication number: IL166405A0
Authority: IL; Israel
Prior art keywords: methyl; methyxycarbonyl; methyleneü; aminoanilo; monoethanesulphonate
Prior art date: 2002-07-24

Application number

IL16640503A

Other languages

English (en)

Original Assignee

Boehringer Ingelheim Pharma

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-07-24

Filing date

2003-07-18

Publication date

2006-01-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=30469050&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL166405(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2003-07-18 Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma

2006-01-15 Publication of IL166405A0 publication Critical patent/IL166405A0/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/32—Oxygen atoms
- C07D209/34—Oxygen atoms in position 2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)
Hydrogenated Pyridines (AREA)

IL16640503A 2002-07-24 2003-07-18 3-z-Ä1-4-(n-((4-methyl-piperazin-1-yl)methylcarbonyl)-n-methyl-aminoanilo)-1-phenyl-methyleneÜ-6-methyxycarbonyl-2-indoline-monoethanesulphonate and the use thereof as a pharmaceutical composition IL166405A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE10233500A DE10233500A1 (de)	2002-07-24	2002-07-24	3-Z-[1-(4-(N-((4-Methyl-piperazin-1-yl)-methylcarbonyl)-N-methyl-amino)-anilino)-1-phenyl-methylen]-6-methoxycarbonyl-2-indolinon-Monoethansulfonat und dessen Verwendung als Arzneimittel
PCT/EP2003/007822 WO2004013099A1 (en)	2002-07-24	2003-07-18	3-z-[1-(4-(n-((4-methyl-piperazin-1-yl)-methylcarbonyl)-n-methyl-amino)-anilino)-1-phenyl-methylene]-6-methoxycarbonyl-2-indolinone-monoethanesulphonate and the use thereof as a pharmaceutical composition

Publications (1)

Publication Number	Publication Date
IL166405A0 true IL166405A0 (en)	2006-01-15

Family

ID=30469050

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
IL16640503A IL166405A0 (en)	2002-07-24	2003-07-18	3-z-Ä1-4-(n-((4-methyl-piperazin-1-yl)methylcarbonyl)-n-methyl-aminoanilo)-1-phenyl-methyleneÜ-6-methyxycarbonyl-2-indoline-monoethanesulphonate and the use thereof as a pharmaceutical composition
IL166405A IL166405A (en)	2002-07-24	2005-01-20	3 - z - [1 - 4 - (n - ((4 - methyl - piperazin - 1 - yl) - methylcarbonyl) - n - methyl - amino) anilino) - 1 -phenyl- methylene] - 6 - methyxycarbonyl - 2 - indolinone - monoethanesulphonate and the use thereof as a pharmaceutical composition

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
IL166405A IL166405A (en)	2002-07-24	2005-01-20	3 - z - [1 - 4 - (n - ((4 - methyl - piperazin - 1 - yl) - methylcarbonyl) - n - methyl - amino) anilino) - 1 -phenyl- methylene] - 6 - methyxycarbonyl - 2 - indolinone - monoethanesulphonate and the use thereof as a pharmaceutical composition

Country Status (35)

Country	Link
US (2)	US7119093B2 (no)
EP (2)	EP2386543A1 (no)
JP (1)	JP5039279B2 (no)
KR (1)	KR101145691B1 (no)
CN (1)	CN100351235C (no)
AR (2)	AR040662A1 (no)
AT (1)	ATE551322T1 (no)
AU (1)	AU2003254376B2 (no)
BR (1)	BRPI0312811B8 (no)
CA (1)	CA2493310C (no)
CY (1)	CY1112916T1 (no)
DE (1)	DE10233500A1 (no)
DK (1)	DK1527047T3 (no)
EA (1)	EA008684B1 (no)
EC (1)	ECSP055571A (no)
EG (1)	EG24562A (no)
ES (1)	ES2384968T3 (no)
HR (1)	HRP20050070B1 (no)
IL (2)	IL166405A0 (no)
ME (1)	ME00353B (no)
MX (1)	MXPA04012785A (no)
MY (1)	MY136883A (no)
NO (1)	NO330486B1 (no)
NZ (1)	NZ538367A (no)
PE (1)	PE20040704A1 (no)
PL (1)	PL223758B1 (no)
PT (1)	PT1527047E (no)
RS (1)	RS52283B (no)
SA (1)	SA03240446B1 (no)
SI (1)	SI1527047T1 (no)
TW (1)	TWI285635B (no)
UA (1)	UA78352C2 (no)
UY (1)	UY27904A1 (no)
WO (1)	WO2004013099A1 (no)
ZA (1)	ZA200409814B (no)

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2002
- 2002-07-24 DE DE10233500A patent/DE10233500A1/de not_active Withdrawn
2003
- 2003-07-18 NZ NZ538367A patent/NZ538367A/en not_active IP Right Cessation
- 2003-07-18 ES ES03766212T patent/ES2384968T3/es not_active Expired - Lifetime
- 2003-07-18 IL IL16640503A patent/IL166405A0/xx unknown
- 2003-07-18 EP EP11172210A patent/EP2386543A1/en not_active Withdrawn
- 2003-07-18 UA UAA200501637A patent/UA78352C2/uk unknown
- 2003-07-18 DK DK03766212.9T patent/DK1527047T3/da active
- 2003-07-18 WO PCT/EP2003/007822 patent/WO2004013099A1/en not_active Ceased
- 2003-07-18 EA EA200500146A patent/EA008684B1/ru active Protection Beyond IP Right Term
- 2003-07-18 AU AU2003254376A patent/AU2003254376B2/en active Active
- 2003-07-18 SI SI200332162T patent/SI1527047T1/sl unknown
- 2003-07-18 PT PT03766212T patent/PT1527047E/pt unknown
- 2003-07-18 AT AT03766212T patent/ATE551322T1/de active
- 2003-07-18 PL PL372996A patent/PL223758B1/pl unknown
- 2003-07-18 JP JP2004525239A patent/JP5039279B2/ja not_active Expired - Lifetime
- 2003-07-18 KR KR1020057001207A patent/KR101145691B1/ko not_active Expired - Lifetime
- 2003-07-18 ME MEP-2008-537A patent/ME00353B/me unknown
- 2003-07-18 CA CA2493310A patent/CA2493310C/en not_active Expired - Lifetime
- 2003-07-18 CN CNB038175304A patent/CN100351235C/zh not_active Ceased
- 2003-07-18 BR BRPI0312811A patent/BRPI0312811B8/pt active IP Right Grant
- 2003-07-18 EP EP03766212A patent/EP1527047B1/en not_active Expired - Lifetime
- 2003-07-18 MX MXPA04012785A patent/MXPA04012785A/es active IP Right Grant
- 2003-07-18 RS YU20050046A patent/RS52283B/sr unknown
- 2003-07-18 HR HRP20050070AA patent/HRP20050070B1/hr not_active IP Right Cessation
- 2003-07-21 US US10/623,971 patent/US7119093B2/en not_active Expired - Lifetime
- 2003-07-22 MY MYPI20032748A patent/MY136883A/en unknown
- 2003-07-22 EG EG2003070712A patent/EG24562A/xx active
- 2003-07-22 PE PE2003000728A patent/PE20040704A1/es active IP Right Grant
- 2003-07-23 TW TW092120101A patent/TWI285635B/zh active
- 2003-07-23 UY UY27904A patent/UY27904A1/es not_active Application Discontinuation
- 2003-07-23 AR AR20030102633A patent/AR040662A1/es not_active Application Discontinuation
- 2003-12-16 SA SA03240446A patent/SA03240446B1/ar unknown
2004
- 2004-12-03 ZA ZA200409814A patent/ZA200409814B/xx unknown
2005
- 2005-01-20 IL IL166405A patent/IL166405A/en active IP Right Grant
- 2005-01-24 EC EC2005005571A patent/ECSP055571A/es unknown
- 2005-02-23 NO NO20050985A patent/NO330486B1/no not_active IP Right Cessation
2006
- 2006-07-28 US US11/460,677 patent/US20060258681A1/en not_active Abandoned
2012
- 2012-06-13 CY CY20121100538T patent/CY1112916T1/el unknown
2013
- 2013-12-20 AR ARP130104954A patent/AR094217A2/es not_active Application Discontinuation

Also Published As

Publication number	Publication date
US20040176392A1 (en)	2004-09-09
EP2386543A1 (en)	2011-11-16
BRPI0312811A8 (pt)	2019-01-02
US7119093B2 (en)	2006-10-10
NO330486B1 (no)	2011-04-26
AU2003254376B2 (en)	2010-06-17
CN100351235C (zh)	2007-11-28
ME00353B (me)	2011-10-10
ES2384968T3 (es)	2012-07-16
AU2003254376A1 (en)	2004-02-23
JP5039279B2 (ja)	2012-10-03
PT1527047E (pt)	2012-06-28
NZ538367A (en)	2008-01-31
EP1527047B1 (en)	2012-03-28
BRPI0312811B1 (pt)	2019-03-12
SI1527047T1 (sl)	2012-07-31
HRP20050070B1 (hr)	2013-09-30
RS52283B (sr)	2012-10-31
CN1671660A (zh)	2005-09-21
ZA200409814B (en)	2006-02-22
DK1527047T3 (da)	2012-07-16
RS20050046A (sr)	2007-09-21
EP1527047A1 (en)	2005-05-04
AR094217A2 (es)	2015-07-15
EG24562A (en)	2009-10-25
NO20050985L (no)	2005-02-23
CY1112916T1 (el)	2016-04-13
PL223758B1 (pl)	2016-10-31
DE10233500A1 (de)	2004-02-19
UA78352C2 (uk)	2007-03-15
TW200409754A (en)	2004-06-16
TWI285635B (en)	2007-08-21
MY136883A (en)	2008-11-28
BRPI0312811B8 (pt)	2021-05-25
KR101145691B1 (ko)	2012-05-25
MXPA04012785A (es)	2005-06-08
HK1078851A1 (zh)	2006-03-24
IL166405A (en)	2009-11-18
KR20050042139A (ko)	2005-05-04
UY27904A1 (es)	2004-02-27
AR040662A1 (es)	2005-04-13
PE20040704A1 (es)	2004-11-29
EA200500146A1 (ru)	2005-08-25
WO2004013099A1 (en)	2004-02-12
MEP53708A (en)	2011-05-10
JP2005535684A (ja)	2005-11-24
ECSP055571A (es)	2005-04-18
HRP20050070A2 (en)	2005-12-31
BR0312811A (pt)	2005-04-19
CA2493310C (en)	2011-01-18
EA008684B1 (ru)	2007-06-29
SA03240446B1 (ar)	2007-07-31
ATE551322T1 (de)	2012-04-15
PL372996A1 (en)	2005-08-08
US20060258681A1 (en)	2006-11-16
CA2493310A1 (en)	2004-02-12

Publication	Publication Date	Title
IL166405A0 (en)	2006-01-15	3-z-Ä1-4-(n-((4-methyl-piperazin-1-yl)methylcarbonyl)-n-methyl-aminoanilo)-1-phenyl-methyleneÜ-6-methyxycarbonyl-2-indoline-monoethanesulphonate and the use thereof as a pharmaceutical composition
HUP0302845A3 (en)	2005-11-28	4-fluoro-n-indan-2-yl benzamide and its use as pharmaceutical
IL166129A0 (en)	2006-01-15	Pyrrolotriazine derivatives and pharmaceutical compositions containing the same
EP1550657A4 (en)	2009-12-30	AMINO COMPOUNDS AND THEIR USE
IL164987A (en)	2011-06-30	Proline derivatives and pharmaceutical compositions containing the same
IL166482A0 (en)	2006-01-15	Dihydropyrazolopyridine derivatives and pharmaceutical compositions containing the same
IL155196A0 (en)	2003-11-23	Benzamide derivatives and pharmaceutical compositions containing the same
PL378135A1 (pl)	2006-03-06	2-Cyjanopirolopirymidyny i ich zastosowania w farmaceutykach
IL166512A0 (en)	2006-01-15	Azaindoleoxoacetic piperazine derivatives and pharmaceutical compositions containing the same
EG25097A (en)	2011-08-17	Piprazinyl and diazapanyl benzamides and benzthioamides.
EP1586557A4 (en)	2006-06-28	4-NITRO-2- (4'-METHOXY) -PHENOXY \| -METHANESULFONANILIDE DERIVATIVES AND THEIR USE FOR PHARMACEUTICAL PURPOSES
GB0108470D0 (en)	2001-05-23	Pharmaceutical compositions and their use
GB0220214D0 (en)	2002-10-09	Compounds and their use
GB0615918D0 (en)	2006-09-20	Composition and its therapeutic use
AU2003298129A8 (en)	2004-06-15	Floor-furnace chimney and the use thereof
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AU2003258772A8 (en)	2003-12-02	Novel neutracetical and pharmaceutical compositions and their uses
GB0230134D0 (en)	2003-01-29	Compounds and their use
IL163627A0 (en)	2005-12-18	Aminoalcohol derivatives and pharmaceutical compositions containing the same
GB0218031D0 (en)	2002-09-11	Compounds and their use
GB0230281D0 (en)	2003-02-05	Compounds and their use
SI1543010T1 (sl)	2007-10-31	N-substituirani hidromorfoni in njihova uporaba
GB0220215D0 (en)	2002-10-09	Compounds and their use
EP1547593A4 (en)	2009-12-23	MEDICINAL COMPOSITION
AU2003242250A1 (en)	2003-12-31	Cyclic amine and medicinal composition containing the same