IL153703A0 - 9-alpha-chloro-6-alpha-fluoro-17-alpha-hydroxy-16-methyl-17-beta-methoxycarbonyl-androst-1,4-dienes esterified in position 17-alpha by a cyclic acyl group - Google Patents

9-alpha-chloro-6-alpha-fluoro-17-alpha-hydroxy-16-methyl-17-beta-methoxycarbonyl-androst-1,4-dienes esterified in position 17-alpha by a cyclic acyl group

Info

Publication number: IL153703A0
Authority: IL; Israel
Prior art keywords: alpha; androst; dienes; methoxycarbonyl; esterified
Prior art date: 2000-06-28

Application number

IL15370301A

Other languages

English (en)

Original Assignee

Novartis Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-06-28

Filing date

2001-06-26

Publication date

2003-07-06

2001-06-26 Application filed by Novartis Ag filed Critical Novartis Ag

2003-07-06 Publication of IL153703A0 publication Critical patent/IL153703A0/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0038—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 with an androstane skeleton, including 18- or 19-substituted derivatives, 18-nor derivatives and also derivatives where position 17-beta is substituted by a carbon atom not directly bonded to a further carbon atom and not being part of an amide group
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
- C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0094—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 containing nitrile radicals, including thiocyanide radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes
- C07J71/0015—Oxiranes at position 9(11)

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pulmonology (AREA)
Toxicology (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Steroid Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)

IL15370301A 2000-06-28 2001-06-26 9-alpha-chloro-6-alpha-fluoro-17-alpha-hydroxy-16-methyl-17-beta-methoxycarbonyl-androst-1,4-dienes esterified in position 17-alpha by a cyclic acyl group IL153703A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GBGB0015876.6A GB0015876D0 (en)	2000-06-28	2000-06-28	Organic compounds
PCT/EP2001/007249 WO2002000679A2 (fr)	2000-06-28	2001-06-26	Composes organiques

Publications (1)

Publication Number	Publication Date
IL153703A0 true IL153703A0 (en)	2003-07-06

Family

ID=9894607

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
IL15370301A IL153703A0 (en)	2000-06-28	2001-06-26	9-alpha-chloro-6-alpha-fluoro-17-alpha-hydroxy-16-methyl-17-beta-methoxycarbonyl-androst-1,4-dienes esterified in position 17-alpha by a cyclic acyl group
IL153703A IL153703A (en)	2000-06-28	2002-12-26	9 - Alpha - Chloro - 6 - Alpha - Fluoro - 17 - Alpha - Hydroxy - 16 - Methyl - 17 - Beta - Methoxycarbonyl - Androst - 4,1 - Dianes that have been sterilized in position 17 - Alpha by a group of ring nobles

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
IL153703A IL153703A (en)	2000-06-28	2002-12-26	9 - Alpha - Chloro - 6 - Alpha - Fluoro - 17 - Alpha - Hydroxy - 16 - Methyl - 17 - Beta - Methoxycarbonyl - Androst - 4,1 - Dianes that have been sterilized in position 17 - Alpha by a group of ring nobles

Country Status (29)

Country	Link
US (1)	US6921757B2 (fr)
EP (1)	EP1299409B1 (fr)
JP (1)	JP4065399B2 (fr)
KR (1)	KR100483865B1 (fr)
CN (1)	CN1214038C (fr)
AR (1)	AR030707A1 (fr)
AT (1)	ATE292639T1 (fr)
AU (2)	AU8389101A (fr)
BR (1)	BR0112068A (fr)
CA (1)	CA2412541C (fr)
CZ (1)	CZ302513B6 (fr)
DE (1)	DE60109931T2 (fr)
EC (1)	ECSP014101A (fr)
ES (1)	ES2240499T3 (fr)
GB (1)	GB0015876D0 (fr)
HU (1)	HUP0300783A3 (fr)
IL (2)	IL153703A0 (fr)
MX (1)	MXPA02012830A (fr)
MY (1)	MY129523A (fr)
NO (1)	NO324055B1 (fr)
NZ (1)	NZ523194A (fr)
PE (1)	PE20020179A1 (fr)
PL (1)	PL207722B1 (fr)
PT (1)	PT1299409E (fr)
RU (1)	RU2277100C2 (fr)
SK (1)	SK286690B6 (fr)
TW (1)	TWI232868B (fr)
WO (1)	WO2002000679A2 (fr)
ZA (1)	ZA200300202B (fr)

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* Cited by examiner, † Cited by third party
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UA77656C2 (en)	2001-04-07	2007-01-15	Glaxo Group Ltd	S-fluoromethyl ester of 6-alpha, 9-alpha-difluoro-17-alpha-[(2-furanylcarbonyl)oxy]-11-beta-hydroxy-16- alpha-methyl-3-oxoandrosta-1,4-dien-17-beta-carbothioacid as anti-inflammatory agent
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AU2015294889B2 (en)	2014-07-31	2018-03-15	Novartis Ag	Combination therapy
EP3248123A1 (fr)	2015-01-20	2017-11-29	Novartis AG	Déverrouillage d'application au moyen d'un dispositif physique, et transfert de données entre ces éléments
PL3111978T3 (pl)	2015-07-03	2022-01-24	Novartis Ag	Inhalator przystosowany do odczytu informacji przechowywanych w środkach przechowywania danych pojemnika
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2000
- 2000-06-28 GB GBGB0015876.6A patent/GB0015876D0/en not_active Ceased
2001
- 2001-06-20 EC EC2001004101A patent/ECSP014101A/es unknown
- 2001-06-26 IL IL15370301A patent/IL153703A0/xx active IP Right Grant
- 2001-06-26 US US10/312,021 patent/US6921757B2/en not_active Expired - Fee Related
- 2001-06-26 KR KR10-2002-7017949A patent/KR100483865B1/ko not_active Expired - Fee Related
- 2001-06-26 PE PE2001000620A patent/PE20020179A1/es not_active Application Discontinuation
- 2001-06-26 PT PT01962783T patent/PT1299409E/pt unknown
- 2001-06-26 NZ NZ523194A patent/NZ523194A/en not_active IP Right Cessation
- 2001-06-26 RU RU2003100504/04A patent/RU2277100C2/ru not_active IP Right Cessation
- 2001-06-26 AT AT01962783T patent/ATE292639T1/de active
- 2001-06-26 ES ES01962783T patent/ES2240499T3/es not_active Expired - Lifetime
- 2001-06-26 CN CNB018117430A patent/CN1214038C/zh not_active Expired - Fee Related
- 2001-06-26 TW TW090115444A patent/TWI232868B/zh not_active IP Right Cessation
- 2001-06-26 HU HU0300783A patent/HUP0300783A3/hu unknown
- 2001-06-26 WO PCT/EP2001/007249 patent/WO2002000679A2/fr not_active Ceased
- 2001-06-26 AU AU8389101A patent/AU8389101A/xx active Pending
- 2001-06-26 BR BR0112068-9A patent/BR0112068A/pt not_active IP Right Cessation
- 2001-06-26 EP EP01962783A patent/EP1299409B1/fr not_active Expired - Lifetime
- 2001-06-26 SK SK1813-2002A patent/SK286690B6/sk not_active IP Right Cessation
- 2001-06-26 MX MXPA02012830A patent/MXPA02012830A/es active IP Right Grant
- 2001-06-26 CZ CZ20024203A patent/CZ302513B6/cs not_active IP Right Cessation
- 2001-06-26 CA CA002412541A patent/CA2412541C/fr not_active Expired - Fee Related
- 2001-06-26 JP JP2002505801A patent/JP4065399B2/ja not_active Expired - Fee Related
- 2001-06-26 AR ARP010103032A patent/AR030707A1/es active IP Right Grant
- 2001-06-26 PL PL358428A patent/PL207722B1/pl not_active IP Right Cessation
- 2001-06-26 AU AU2001283891A patent/AU2001283891B2/en not_active Ceased
- 2001-06-26 DE DE60109931T patent/DE60109931T2/de not_active Expired - Lifetime
- 2001-06-26 MY MYPI20013015A patent/MY129523A/en unknown
2002
- 2002-12-26 IL IL153703A patent/IL153703A/en not_active IP Right Cessation
- 2002-12-27 NO NO20026253A patent/NO324055B1/no not_active IP Right Cessation
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- 2003-01-08 ZA ZA200300202A patent/ZA200300202B/xx unknown

Also Published As

Publication number	Publication date
ECSP014101A (es)	2002-01-25
BR0112068A (pt)	2003-04-01
DE60109931D1 (de)	2005-05-12
MXPA02012830A (es)	2003-05-14
HUP0300783A3 (en)	2010-01-28
NO20026253D0 (no)	2002-12-27
NO20026253L (no)	2003-02-18
US6921757B2 (en)	2005-07-26
AU2001283891B2 (en)	2004-06-17
ZA200300202B (en)	2003-12-31
ES2240499T3 (es)	2005-10-16
HK1055974A1 (en)	2004-01-30
CN1439018A (zh)	2003-08-27
RU2277100C2 (ru)	2006-05-27
DE60109931T2 (de)	2006-02-02
AU8389101A (en)	2002-01-08
AR030707A1 (es)	2003-09-03
JP2004501930A (ja)	2004-01-22
NZ523194A (en)	2005-08-26
EP1299409B1 (fr)	2005-04-06
KR20030028768A (ko)	2003-04-10
WO2002000679A3 (fr)	2002-03-28
NO324055B1 (no)	2007-08-06
GB0015876D0 (en)	2000-08-23
ATE292639T1 (de)	2005-04-15
KR100483865B1 (ko)	2005-04-20
PL207722B1 (pl)	2011-01-31
CN1214038C (zh)	2005-08-10
PE20020179A1 (es)	2002-04-10
WO2002000679A2 (fr)	2002-01-03
SK18132002A3 (sk)	2003-08-05
CZ302513B6 (cs)	2011-06-29
CZ20024203A3 (cs)	2003-04-16
CA2412541A1 (fr)	2002-01-03
PL358428A1 (en)	2004-08-09
EP1299409A2 (fr)	2003-04-09
TWI232868B (en)	2005-05-21
CA2412541C (fr)	2009-01-06
JP4065399B2 (ja)	2008-03-26
US20030158163A1 (en)	2003-08-21
HUP0300783A2 (hu)	2003-07-28
SK286690B6 (sk)	2009-03-05
MY129523A (en)	2007-04-30
PT1299409E (pt)	2005-08-31
IL153703A (en)	2007-05-15

Publication	Publication Date	Title
IL153703A0 (en)	2003-07-06	9-alpha-chloro-6-alpha-fluoro-17-alpha-hydroxy-16-methyl-17-beta-methoxycarbonyl-androst-1,4-dienes esterified in position 17-alpha by a cyclic acyl group
GB0029531D0 (en)	2001-01-17	Speed govenor
AU8402601A (en)	2002-03-13	Selective cyclic peptides
GB0025244D0 (en)	2000-11-29	Turbine
GB0015207D0 (en)	2000-08-09	A turbine
AU9163801A (en)	2002-04-08	A conveyor
GB0023562D0 (en)	2000-11-08	An amusement machine
GB2381115B (en)	2004-10-20	Pusher amusement machine
GB0005989D0 (en)	2000-05-03	A rotor
PL357875A1 (en)	2004-07-26	Cyclic hexapeptide derivatives
AU2001282624A1 (en)	2002-03-22	Rankine cycle device
SI1299409T1 (en)	2005-10-31	9.alpha.-chloro-6.alpha.-fluoro-17.alpha.-hydroxy-16-methyl-17-beta-methoxycarbonyl-androst-1,4-dienes esterified in position 17.alpha. by a cyclic acyl group
GB2364719B (en)	2003-10-22	Post sock
GB2373028B (en)	2003-03-19	Turbines
TW441386U (en)	2001-06-16	Improved sandbag structure
GB9921415D0 (en)	1999-11-10	Variable position cycle
AU142477S (en)	2000-12-12	A doll
GB0026373D0 (en)	2000-12-13	A structure
GB0023271D0 (en)	2000-11-08	A toy having variable configuration
AU3409501A (en)	2001-08-27	Cyclic hexapeptide derivatives
GB2397426B (en)	2004-10-20	Pusher amusement machine
GB0012888D0 (en)	2000-07-19	Turbine
GB0007481D0 (en)	2000-05-17	A physical sefety barrier
AU4035301A (en)	2001-09-17	A toy
AU144611S (en)	2001-07-31	A toy

Legal Events

Date	Code	Title	Description
2007-10-31	FF	Patent granted
2008-01-06	KB	Patent renewed