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HN2000000045A - NEW PHARMACEUTICAL COMBINATIONS FOR INHIBITORS OF THE US. - Google Patents

NEW PHARMACEUTICAL COMBINATIONS FOR INHIBITORS OF THE US.

Info

Publication number
HN2000000045A
HN2000000045A HN2000000045A HN2000000045A HN2000000045A HN 2000000045 A HN2000000045 A HN 2000000045A HN 2000000045 A HN2000000045 A HN 2000000045A HN 2000000045 A HN2000000045 A HN 2000000045A HN 2000000045 A HN2000000045 A HN 2000000045A
Authority
HN
Honduras
Prior art keywords
inhibitors
new pharmaceutical
pharmaceutical combinations
present
new
Prior art date
Application number
HN2000000045A
Other languages
Spanish (es)
Inventor
Iii Mario David Saltarelli Joh
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of HN2000000045A publication Critical patent/HN2000000045A/en

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
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    • A61K31/15—Oximes (>C=N—O—); Hydrazines (>N—N<); Hydrazones (>N—N=) ; Imines (C—N=C)
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    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyridine Compounds (AREA)

Abstract

LA PRESENTE INVENCION SE REFIERE A NUEVOS USOS FARMACEUTICOS PARA COMPUESTOS QUE PRESENTAN ACTIVIDAD COMO INHIBIDORES DE LA OXIDO NITRICO SINTASA (NOS).THE PRESENT INVENTION REFERS TO NEW PHARMACEUTICAL USES FOR COMPOUNDS THAT PRESENT ACTIVITY AS INHIBITORS OF NITRICO SINTASA OXIDE (US).

HN2000000045A 1999-05-21 2000-04-04 NEW PHARMACEUTICAL COMBINATIONS FOR INHIBITORS OF THE US. HN2000000045A (en)

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AR (1) AR022640A1 (en)
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CA (1) CA2374668A1 (en)
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DZ (1) DZ3041A1 (en)
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DE10001785A1 (en) * 2000-01-18 2001-07-19 Boehringer Ingelheim Pharma Use of NK-1 receptor antagonists for treatment of restless legs syndrome
GB0019006D0 (en) * 2000-08-04 2000-09-20 Astrazeneca Ab Novel compounds
US20030045449A1 (en) * 2001-08-15 2003-03-06 Pfizer, Inc. Pharmaceutical combinations for the treatment of neurodegenerative diseases
DOP2002000467A (en) * 2001-10-10 2003-04-15 Pfizer Prod Inc 2-AMINO-6 (PHENYL REPLACED IN POSITIONS 2,4,5) -PIRIDINES
US6803470B2 (en) * 2001-10-10 2004-10-12 Pfizer Inc 2-amino-6-(2,4,5-substituted-phenyl)-pyridines
JP2009513491A (en) * 2003-06-24 2009-04-02 ノイロサーチ アクティーゼルスカブ Novel 8-aza-bicyclo [3.2.1] octane derivatives and their use as monoamine neurotransmitter reuptake inhibitors
EP1634598A1 (en) * 2004-09-07 2006-03-15 Laboratorios Del Dr. Esteve, S.A. Use of piperazine derivatives and analogues for the manufacture of a medicament for the prophylaxis and/or treatment of disorders of food ingestion
CN101678019B (en) 2007-06-08 2016-03-30 詹森药业有限公司 Piperidine/piperazine derivatives
JP5443342B2 (en) 2007-06-08 2014-03-19 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ Piperidine / piperazine derivatives
ES2483898T3 (en) 2007-06-08 2014-08-08 Janssen Pharmaceutica, N.V. Piperidine / Piperazine Derivatives
JO2972B1 (en) 2007-06-08 2016-03-15 جانسين فارماسوتيكا ان. في Piperidine/Piperazine derivatives
WO2009147170A2 (en) 2008-06-05 2009-12-10 Janssen Pharmaceutica Nv Drug combinations comprising a dgat inhibitor and a ppar-agonist
US8889674B2 (en) 2009-03-05 2014-11-18 Shionogi & Co., Ltd. Piperidine and pyrrolidine derivatives having NPY Y5 receptor antagonism
JP6440625B2 (en) 2012-11-14 2018-12-19 ザ・ジョンズ・ホプキンス・ユニバーシティー Methods and compositions for treating schizophrenia
WO2020252383A2 (en) * 2019-06-14 2020-12-17 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (pcsk9)
US12115154B2 (en) 2020-12-16 2024-10-15 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9)

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GT200000071A (en) 2001-11-08
PE20010157A1 (en) 2001-02-16
MA26732A1 (en) 2004-12-20
KR20020010916A (en) 2002-02-06
WO2000071107A8 (en) 2002-01-24
HUP0301287A3 (en) 2005-03-29
BR0010820A (en) 2002-03-05
JP2003523941A (en) 2003-08-12
NO20015651L (en) 2002-01-18
HRP20010862A2 (en) 2003-06-30
HUP0301287A2 (en) 2003-08-28
NO20015651D0 (en) 2001-11-20
DZ3041A1 (en) 2004-03-27
CA2374668A1 (en) 2000-11-30
OA11943A (en) 2006-04-12
PL358538A1 (en) 2004-08-09
ZA200109555B (en) 2004-04-07
TR200103351T2 (en) 2002-06-21
AU2935300A (en) 2000-12-12
IS6126A (en) 2001-10-26
PA8494601A1 (en) 2002-08-29
CO5160295A1 (en) 2002-05-30
EA200101110A1 (en) 2002-08-29
EP1178784A1 (en) 2002-02-13
IL145955A0 (en) 2002-07-25
WO2000071107A2 (en) 2000-11-30
TNSN00106A1 (en) 2005-11-10
CN1617743A (en) 2005-05-18
AP2001002326A0 (en) 2001-12-31
EE200100611A (en) 2003-02-17
BG106208A (en) 2002-09-30
AR022640A1 (en) 2002-09-04
MXPA01011978A (en) 2002-05-06
SK16602001A3 (en) 2003-03-04
UY26148A1 (en) 2000-12-29

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