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HK1200371B - 以草酸酰胺作为脑啡肽酶抑制剂,其药物组合物及其制备方法 - Google Patents

以草酸酰胺作为脑啡肽酶抑制剂,其药物组合物及其制备方法 Download PDF

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Publication number
HK1200371B
HK1200371B HK15101114.2A HK15101114A HK1200371B HK 1200371 B HK1200371 B HK 1200371B HK 15101114 A HK15101114 A HK 15101114A HK 1200371 B HK1200371 B HK 1200371B
Authority
HK
Hong Kong
Prior art keywords
compound
alkyl
alkylene
chloro
mmol
Prior art date
Application number
HK15101114.2A
Other languages
German (de)
English (en)
French (fr)
Other versions
HK1200371A1 (zh
Inventor
Adam Hughes
Erik FENSTER
Melissa Fleury
Roland Gendron
Edmund J. Moran
Original Assignee
Theravance Biopharma R&D Ip, Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Theravance Biopharma R&D Ip, Llc filed Critical Theravance Biopharma R&D Ip, Llc
Priority claimed from PCT/US2012/063036 external-priority patent/WO2013067163A1/en
Publication of HK1200371A1 publication Critical patent/HK1200371A1/zh
Publication of HK1200371B publication Critical patent/HK1200371B/zh

Links

HK15101114.2A 2011-11-02 2012-11-01 以草酸酰胺作为脑啡肽酶抑制剂,其药物组合物及其制备方法 HK1200371B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161554625P 2011-11-02 2011-11-02
US61/554,625 2011-11-02
PCT/US2012/063036 WO2013067163A1 (en) 2011-11-02 2012-11-01 Neprilysin inhibitors

Publications (2)

Publication Number Publication Date
HK1200371A1 HK1200371A1 (zh) 2015-08-07
HK1200371B true HK1200371B (zh) 2018-04-13

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