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GT200800123A - Compuestos mimeticos de lisina modificados - Google Patents

Compuestos mimeticos de lisina modificados

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Publication number
GT200800123A
GT200800123A GT200800123A GT200800123A GT200800123A GT 200800123 A GT200800123 A GT 200800123A GT 200800123 A GT200800123 A GT 200800123A GT 200800123 A GT200800123 A GT 200800123A GT 200800123 A GT200800123 A GT 200800123A
Authority
GT
Guatemala
Prior art keywords
lisine
modified
mimetic compounds
activity
mimetic
Prior art date
Application number
GT200800123A
Other languages
English (en)
Inventor
Bjarne Due Larsen
Jorgen Soberg Petersen
Ketil Jorgen Haugan
John A Butera
James K Hennan
Edward H Kerns
Evgueni Lvovich Piatnitski
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38110525&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GT200800123(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of GT200800123A publication Critical patent/GT200800123A/es

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    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00Carboxylic acid amides
    • C07C233/64Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/81Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
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    • C07C233/00Carboxylic acid amides
    • C07C233/01Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
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    • C07C233/31Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by doubly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
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    • C07C233/57Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of rings other than six-membered aromatic rings
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    • C07C233/82Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/83Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of an acyclic saturated carbon skeleton
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    • C07C237/20Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton containing six-membered aromatic rings
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Abstract

LA PRESENTE INVENCIÓN PRESENTA COMPUESTOS MIMÉTICOS DE LISINA QUE TIENEN ACTIVIDAD FARMACOLÓGICA ÚTIL TAL COMO ACTIVIDAD ANTIARRÍTMICA Y PROPIEDADES BENEFICIOSAS DE BIODISPONIBILIDAD. T2008
GT200800123A 2005-12-23 2008-06-20 Compuestos mimeticos de lisina modificados GT200800123A (es)

Applications Claiming Priority (1)

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US20120245106A1 (en) 2012-09-27
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ECSP088633A (es) 2008-09-29
CN102690221B (zh) 2014-12-03
RU2494095C2 (ru) 2013-09-27
US20070149460A1 (en) 2007-06-28
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NZ569293A (en) 2011-10-28
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WO2007078990A3 (en) 2007-11-22
IL192395A (en) 2015-09-24
UA96283C2 (uk) 2011-10-25
EP2386539A2 (en) 2011-11-16
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CA2634743C (en) 2014-07-29
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