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GT200000102A - Complejo farmaceutico. - Google Patents

Complejo farmaceutico.

Info

Publication number
GT200000102A
GT200000102A GT200000102A GT200000102A GT200000102A GT 200000102 A GT200000102 A GT 200000102A GT 200000102 A GT200000102 A GT 200000102A GT 200000102 A GT200000102 A GT 200000102A GT 200000102 A GT200000102 A GT 200000102A
Authority
GT
Guatemala
Prior art keywords
complex
eletriptan
formulation
same
sulfobutileter
Prior art date
Application number
GT200000102A
Other languages
English (en)
Inventor
Anne Billotte
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT200000102A publication Critical patent/GT200000102A/es

Links

Classifications

    • BPERFORMING OPERATIONS; TRANSPORTING
    • B82NANOTECHNOLOGY
    • B82YSPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/69Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit
    • A61K47/6949Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes
    • A61K47/6951Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes using cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Nanotechnology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Biophysics (AREA)
  • Biotechnology (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Molecular Biology (AREA)
  • Medical Informatics (AREA)
  • General Engineering & Computer Science (AREA)
  • Otolaryngology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Addiction (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

LA INVENCION SE REFIERE A UN COMPLEJO DE ELECTRIPAN (UNA METILPIRROLIDINA) Y A UNA SULFOBUTILETER BETA CICLODEXTRINA [MOSTRADO EN LA FIGURA I, DONDE "R" = OH O O(CH2)4) SO3 H], O A SALES FARMACEUTICAMENTE ACEPTABLES DE LOS MISMOS, Y A PROCEDIMIENTOS PARA LA PREPARACION DE TAL COMPLEJO, INCLUYENDO FORMULACIONES FARMACEUTICAS Y USOS DEL MISMO. EL ELETRIPTAN ES UN AGONISTA DEL RECEPTOR 5HT Y SE HA DEMOSTRADO ALTAMENTE EFICAZ PARA EL TRATAMIENTO DE LA MIGRAÑA, HIPERTENSION EMESIS, DEPRESION, DEPENDENCIA DE DROGAS. CON EL FIN DE ADMINISTRAR ELETRIPTAN, O UNA SAL DEL MISMO, POR VIA INTRANASAL, ES DESEABLE QUE LA FORMULACION NO PRODUZCA IRRITACION EN LA MUCOSA NASAL, CON ESE PROPOSITO SE LE HA AGREGADO EL COMPLEJO DE DEXTRINA, LOGRANDO UNA BUENA BIODISPONIBILIDAD Y UN COMIENZO DE ACCION RAPIDA; LA FORMULACION TAMBIEN INCLUYE COMPONENTES INDISPENSABLES COMO ANTIOXIDANTES Y EXCIPIENTES.
GT200000102A 1999-06-29 2000-06-22 Complejo farmaceutico. GT200000102A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9915231.6A GB9915231D0 (en) 1999-06-29 1999-06-29 Pharmaceutical complex

Publications (1)

Publication Number Publication Date
GT200000102A true GT200000102A (es) 2001-12-14

Family

ID=10856302

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200000102A GT200000102A (es) 1999-06-29 2000-06-22 Complejo farmaceutico.

Country Status (44)

Country Link
US (2) US6713461B1 (es)
EP (1) EP1189640B1 (es)
JP (2) JP4454900B2 (es)
KR (1) KR20020015067A (es)
CN (1) CN1198654C (es)
AP (1) AP2001002369A0 (es)
AR (1) AR033337A1 (es)
AT (1) ATE290884T1 (es)
AU (1) AU770169B2 (es)
BG (1) BG106151A (es)
BR (1) BR0011845A (es)
CA (1) CA2376847C (es)
CO (1) CO5170494A1 (es)
CZ (1) CZ20014572A3 (es)
DE (1) DE60018744T2 (es)
DZ (1) DZ3320A1 (es)
EA (1) EA003908B1 (es)
EC (1) ECSP003551A (es)
EE (1) EE200100697A (es)
ES (1) ES2235879T3 (es)
GB (1) GB9915231D0 (es)
GE (1) GEP20043377B (es)
GT (1) GT200000102A (es)
HR (1) HRP20010951A2 (es)
HU (1) HUP0201629A3 (es)
IL (1) IL146341A0 (es)
IS (1) IS6163A (es)
MA (1) MA26801A1 (es)
MX (1) MXPA01013274A (es)
NO (1) NO20016430L (es)
NZ (1) NZ515235A (es)
OA (1) OA11964A (es)
PA (1) PA8496801A1 (es)
PE (1) PE20010346A1 (es)
PL (1) PL352902A1 (es)
SK (1) SK18932001A3 (es)
SV (1) SV2002000112A (es)
TN (1) TNSN00142A1 (es)
TR (1) TR200103827T2 (es)
UA (1) UA66932C2 (es)
UY (1) UY26224A1 (es)
WO (1) WO2001000243A1 (es)
YU (1) YU87501A (es)
ZA (1) ZA200110454B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9915231D0 (en) * 1999-06-29 1999-09-01 Pfizer Ltd Pharmaceutical complex
HRP20050149B1 (hr) * 2002-08-20 2014-09-12 Otsuka Pharmaceutical Co., Ltd. Formulacija aripiprazol kompleksa i postupak
GB0329918D0 (en) * 2003-12-24 2004-01-28 West Pharm Serv Drug Res Ltd Intranasal compositions
CN1296391C (zh) * 2004-03-04 2007-01-24 中国人民解放军第二军医大学 氟代羧烷基环糊精醚类化合物及其制备方法和应用
GB0613925D0 (en) * 2006-07-13 2006-08-23 Unilever Plc Improvements relating to nanodispersions
CN101957330B (zh) * 2010-06-12 2013-10-09 南京巨环医药科技开发有限公司 磺丁基倍他环糊精含量的测定方法
WO2017122161A1 (en) * 2016-01-15 2017-07-20 Cadila Healthcare Limited An intranasal composition comprising 5ht1b/1d receptor agonists
WO2019143925A1 (en) * 2018-01-22 2019-07-25 Insys Development Company, Inc. Liquid rizatriptan compositions

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR0166088B1 (ko) * 1990-01-23 1999-01-15 . 수용해도가 증가된 시클로덱스트린 유도체 및 이의 용도
US5376645A (en) * 1990-01-23 1994-12-27 University Of Kansas Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof
HU210921B (en) 1990-03-28 1995-09-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing inclusion complexes of n-ethoxycarbonyl-3-morpholino-sydnonimine formed with cyclodextrines and pharmaceutical compositions containing them
HU212730B (en) 1990-03-28 1996-10-28 Chinoin Gyogyszer Es Vegyeszet Process for producing inclusion complexes of cyclodextrine or its derivative and 3-morpholino-sydnonimine or its salt or its tautomer and pharmaceutical compositions containing them
ES2104733T3 (es) 1990-10-15 1997-10-16 Pfizer Derivados de indol.
ZA941544B (en) 1993-03-05 1994-10-31 Hexal Pharma Gmbh Crystalline cyclodextrin complexes of ranitidine hydrochloride, process for their preparation and pharmaceutical compositions containing the same.
MX9504664A (es) 1994-03-07 1997-05-31 Dow Chemical Co Conjugados de dendrimeros bioactivos y/o dirigidos.
GB9417310D0 (en) 1994-08-27 1994-10-19 Pfizer Ltd Therapeutic agents
KR20000022239A (ko) 1996-07-11 2000-04-25 토마스 헤인 인돌 선택성 세로토닌 작용약을 함유한 내포 복합체
US5998462A (en) 1996-12-16 1999-12-07 Allelix Biopharmaceuticals Inc. 5-alkyl indole compounds
GB9704498D0 (en) 1997-03-05 1997-04-23 Glaxo Wellcome Spa Chemical compound
AU724728B2 (en) 1997-07-03 2000-09-28 Pfizer Inc. Pharmaceutical compositions containing eletriptan hemisulphate and caffeine
GB9816556D0 (en) * 1998-07-30 1998-09-30 Pfizer Ltd Therapy
GB9915231D0 (en) * 1999-06-29 1999-09-01 Pfizer Ltd Pharmaceutical complex

Also Published As

Publication number Publication date
US6713461B1 (en) 2004-03-30
AU770169B2 (en) 2004-02-12
GEP20043377B (en) 2004-04-13
PE20010346A1 (es) 2001-03-26
EP1189640A1 (en) 2002-03-27
CN1359303A (zh) 2002-07-17
TR200103827T2 (tr) 2002-05-21
JP4454900B2 (ja) 2010-04-21
CA2376847C (en) 2007-09-25
CO5170494A1 (es) 2002-06-27
NZ515235A (en) 2003-08-29
ES2235879T3 (es) 2005-07-16
CN1198654C (zh) 2005-04-27
YU87501A (sh) 2004-05-12
DZ3320A1 (fr) 2001-01-04
GB9915231D0 (en) 1999-09-01
OA11964A (en) 2006-04-17
WO2001000243A1 (en) 2001-01-04
ATE290884T1 (de) 2005-04-15
JP2006257091A (ja) 2006-09-28
HUP0201629A2 (hu) 2003-03-28
NO20016430L (no) 2002-02-26
UA66932C2 (en) 2004-06-15
PL352902A1 (en) 2003-09-22
MA26801A1 (fr) 2004-12-20
KR20020015067A (ko) 2002-02-27
UY26224A1 (es) 2001-01-31
DE60018744T2 (de) 2006-05-18
HUP0201629A3 (en) 2003-11-28
EP1189640B1 (en) 2005-03-16
BG106151A (en) 2002-05-31
SV2002000112A (es) 2002-02-05
ECSP003551A (es) 2002-01-25
AR033337A1 (es) 2003-12-17
JP2003503364A (ja) 2003-01-28
EA200101106A1 (ru) 2002-06-27
TNSN00142A1 (fr) 2005-11-10
HRP20010951A2 (en) 2005-04-30
AP2001002369A0 (en) 2001-12-31
ZA200110454B (en) 2002-12-20
US20040186076A1 (en) 2004-09-23
MXPA01013274A (es) 2002-06-04
NO20016430D0 (no) 2001-12-28
CZ20014572A3 (cs) 2002-08-14
DE60018744D1 (de) 2005-04-21
AU4774100A (en) 2001-01-31
EE200100697A (et) 2003-02-17
SK18932001A3 (sk) 2002-09-10
IS6163A (is) 2001-11-16
PA8496801A1 (es) 2002-02-21
IL146341A0 (en) 2002-07-25
EA003908B1 (ru) 2003-10-30
BR0011845A (pt) 2002-03-05
CA2376847A1 (en) 2001-01-04

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