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GT199700104AA - Procedimientos e intermedios para preparar derivados de cromanol sustituidos - Google Patents

Procedimientos e intermedios para preparar derivados de cromanol sustituidos

Info

Publication number
GT199700104AA
GT199700104AA GT199700104AK GT199700104K GT199700104AA GT 199700104A A GT199700104A A GT 199700104AA GT 199700104A K GT199700104A K GT 199700104AK GT 199700104 K GT199700104 K GT 199700104K GT 199700104A A GT199700104A A GT 199700104AA
Authority
GT
Guatemala
Prior art keywords
intermediates
procedures
chromanol derivatives
substituted chromanol
prepare substituted
Prior art date
Application number
GT199700104AK
Other languages
English (en)
Inventor
Anthony Piscopio
Joel M Hawkins
Stephane Caron
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT199700104AA publication Critical patent/GT199700104AA/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/40Halogenated unsaturated alcohols
    • C07C33/50Halogenated unsaturated alcohols containing six-membered aromatic rings and other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/22Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

ESTA INVENCION SE REFIERE A LA PREPARACION DE DERIVADOS DE CROMANOL SUSTITUIDOS Y A INTERMEDIOS UTILES EN DICHA PREPARACION. LOS DERIVADOS DE CROMANOL SUSTITUIDOS QUE SE PREPARAN DE ACUERDO CON LA PRESENTE INVENCION, INHIBEN LA ACCION DE LTB4. ESTOS COMPUESTOS TIENEN LA ESTRUCTURA QUIMICA(V), EN LA QUE X,R1,R2,Y, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE.
GT199700104AK 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos GT199700104AA (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US2637296P 1996-09-16 1996-09-16

Publications (1)

Publication Number Publication Date
GT199700104AA true GT199700104AA (es) 1999-03-28

Family

ID=21831429

Family Applications (3)

Application Number Title Priority Date Filing Date
GT199700104A GT199700104A (es) 1996-09-16 1997-09-08 Procedimientos e intermedios para preparar derivados de cromanol sustituidos.
GT199700104BL GT199700104BA (es) 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos
GT199700104AK GT199700104AA (es) 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos

Family Applications Before (2)

Application Number Title Priority Date Filing Date
GT199700104A GT199700104A (es) 1996-09-16 1997-09-08 Procedimientos e intermedios para preparar derivados de cromanol sustituidos.
GT199700104BL GT199700104BA (es) 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos

Country Status (39)

Country Link
US (4) US6096906A (es)
EP (1) EP0925292B1 (es)
JP (1) JP3117730B2 (es)
KR (1) KR100339164B1 (es)
CN (1) CN1108298C (es)
AP (1) AP726A (es)
AT (1) ATE249452T1 (es)
AU (1) AU713701B2 (es)
BG (1) BG63542B1 (es)
BR (1) BR9711482A (es)
CA (1) CA2265043C (es)
CO (1) CO4600635A1 (es)
DE (1) DE69724801T2 (es)
DK (1) DK0925292T3 (es)
DZ (1) DZ2308A1 (es)
EA (1) EA002204B1 (es)
ES (1) ES2206738T3 (es)
GT (3) GT199700104A (es)
HN (1) HN1997000127A (es)
HR (1) HRP970497B1 (es)
ID (1) ID19613A (es)
IL (1) IL128732A0 (es)
IS (1) IS4980A (es)
MA (1) MA24319A1 (es)
NO (1) NO991254L (es)
NZ (1) NZ334214A (es)
OA (1) OA10995A (es)
PA (1) PA8437901A1 (es)
PE (1) PE109798A1 (es)
PL (1) PL332351A1 (es)
PT (1) PT925292E (es)
SK (1) SK31399A3 (es)
TN (1) TNSN97155A1 (es)
TR (1) TR199900592T2 (es)
TW (1) TW449579B (es)
UA (1) UA58520C2 (es)
WO (1) WO1998011085A1 (es)
YU (1) YU13299A (es)
ZA (1) ZA978291B (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6436987B1 (en) * 2000-06-08 2002-08-20 Pfizer Inc. Crystalline forms of (3S-trans)-2-[3,4-dihydro-4-hydroxy-3-(phenylmethyl)-2H-1-benzopyran-7-yl]-4-(trifluoromethyl)-benzoic acid
JP2004518685A (ja) * 2001-01-30 2004-06-24 ファイザー・プロダクツ・インク クロマニル安息香酸の調製方法
AU4239302A (en) * 2001-06-28 2003-01-02 Pfizer Products Inc. Benzoic acid substituted benzopyrans for the treatment of atherosclerosis
CA2694068C (en) 2007-07-23 2016-08-30 The Board Of Trustees Of The University Of Illinois System for controlling the reactivity of boronic acids
WO2010036921A2 (en) * 2008-09-26 2010-04-01 The Board Of Trustees Of The University Of Illinois Slow release of organoboronic acids in cross-coupling reactions
WO2011028766A2 (en) * 2009-09-02 2011-03-10 E. I. Du Pont De Nemours And Company Fluorinated 4-oxo-chroman-carboxylates
WO2011028767A2 (en) 2009-09-02 2011-03-10 E. I. Du Pont De Nemours And Company Fluoroether functionalized aromatic diesters and derivatives thereof
TW201113311A (en) * 2009-09-02 2011-04-16 Du Pont Polyaramid films comprising fluorovinylether functionalized aromatic moieties
BR112012004774A2 (pt) * 2009-09-02 2017-05-30 Du Pont polímero e processo
US20110218319A1 (en) * 2009-09-02 2011-09-08 E. I. Du Pont De Nemours And Company Polyaramid films comprising fluorovinylether functionalized aromatic moieties
AU2010289576B2 (en) * 2009-09-02 2015-07-16 E. I. Du Pont De Nemours And Company Polyester films with improved oil repellency
WO2011103435A2 (en) 2010-02-18 2011-08-25 The Board Of Trustees Of The University Of Illinois Methods for forming protected organoboronic acids
US10500178B2 (en) 2015-03-13 2019-12-10 The Board Of Trustees Of The Leland Stanford Junior University LTB4 inhibition to prevent and treat human lymphedema
KR102807066B1 (ko) * 2019-09-30 2025-05-15 주식회사 엘지화학 아민계 화합물 제조방법
CN117384617B (zh) * 2023-12-13 2024-03-29 中国石油大学(华东) 一种耐盐型胍胶压裂液交联剂水溶液及其制备方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9119920D0 (en) * 1991-09-18 1991-10-30 Glaxo Group Ltd Chemical compounds
MX9300312A (es) * 1992-01-23 1993-07-31 Pfizer Antagonistas benzopiranicos y relacionado de ltb.
CZ395492A3 (en) * 1992-01-23 1994-03-16 Pfizer Benzopyran ltb4 antagonists and related compounds, process of their preparation, intermediates and use
CZ100895A3 (en) * 1992-10-21 1995-10-18 Pfizer Enantiomeric cis-3-(4,6-dihydroxychroman-3-ylmethyl)benzoic acids
CZ100095A3 (en) * 1992-10-21 1995-11-15 Pfizer Sulfonamide derivatives of hydroxy substituted alicyclic or heterocyclic compounds with condensed benzene nucleus and pharmaceutical preparations based thereon
CN1166834A (zh) * 1994-10-13 1997-12-03 美国辉瑞有限公司 苯并吡喃和苯并稠合化合物,其制备方法和它们作为白三烯b4(ltb4)拮抗剂的用途
CZ111797A3 (cs) * 1994-10-13 1998-07-15 Pfizer Inc. Benzopyranové a jiné sloučeniny s přikondenzovaným benzenovým kruhem a farmaceutické prostředky na jejich bázi
US5539128A (en) * 1994-11-30 1996-07-23 Pfizer Inc. Processes and intermediates for preparing cis(+)3-[4,6-dihydroxy chroman-3-ylmethyl]-4-methoxyaniline

Also Published As

Publication number Publication date
JP2000502726A (ja) 2000-03-07
OA10995A (en) 2001-11-06
NZ334214A (en) 2000-09-29
UA58520C2 (uk) 2003-08-15
AU713701B2 (en) 1999-12-09
US6288242B1 (en) 2001-09-11
EA199900204A1 (ru) 1999-08-26
BR9711482A (pt) 1999-08-24
ES2206738T3 (es) 2004-05-16
EP0925292B1 (en) 2003-09-10
US6444826B1 (en) 2002-09-03
EP0925292A1 (en) 1999-06-30
SK31399A3 (en) 2000-05-16
KR20000036136A (ko) 2000-06-26
BG63542B1 (bg) 2002-04-30
HRP970497B1 (en) 2002-06-30
TR199900592T2 (xx) 1999-06-21
TNSN97155A1 (fr) 2005-03-15
BG103231A (en) 1999-12-30
PE109798A1 (es) 1999-01-13
CA2265043C (en) 2003-01-14
ID19613A (id) 1998-07-23
HRP970497A2 (en) 1998-08-31
PT925292E (pt) 2004-01-30
CA2265043A1 (en) 1998-03-19
AU3781497A (en) 1998-04-02
AP9701083A0 (en) 1997-10-31
KR100339164B1 (ko) 2002-06-01
DE69724801D1 (de) 2003-10-16
IL128732A0 (en) 2000-01-31
GT199700104A (es) 1999-03-02
ATE249452T1 (de) 2003-09-15
US6355825B1 (en) 2002-03-12
ZA978291B (en) 1999-03-15
DK0925292T3 (da) 2004-01-12
PL332351A1 (en) 1999-09-13
JP3117730B2 (ja) 2000-12-18
GT199700104BA (es) 1999-03-28
US20020099227A1 (en) 2002-07-25
YU13299A (sh) 2001-03-07
CN1230954A (zh) 1999-10-06
US20020042526A1 (en) 2002-04-11
HN1997000127A (es) 1997-12-20
IS4980A (is) 1999-02-16
NO991254D0 (no) 1999-03-15
TW449579B (en) 2001-08-11
MA24319A1 (fr) 1998-04-01
DZ2308A1 (fr) 2002-12-28
EA002204B1 (ru) 2002-02-28
CO4600635A1 (es) 1998-05-08
AP726A (en) 1999-01-29
WO1998011085A1 (en) 1998-03-19
PA8437901A1 (es) 2000-05-24
NO991254L (no) 1999-05-14
US6096906A (en) 2000-08-01
DE69724801T2 (de) 2004-06-17
CN1108298C (zh) 2003-05-14

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