GT199700104AA - Procedimientos e intermedios para preparar derivados de cromanol sustituidos - Google Patents
Procedimientos e intermedios para preparar derivados de cromanol sustituidosInfo
- Publication number
- GT199700104AA GT199700104AA GT199700104AK GT199700104K GT199700104AA GT 199700104A A GT199700104A A GT 199700104AA GT 199700104A K GT199700104A K GT 199700104AK GT 199700104 K GT199700104 K GT 199700104K GT 199700104A A GT199700104A A GT 199700104AA
- Authority
- GT
- Guatemala
- Prior art keywords
- intermediates
- procedures
- chromanol derivatives
- substituted chromanol
- prepare substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C33/00—Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
- C07C33/40—Halogenated unsaturated alcohols
- C07C33/50—Halogenated unsaturated alcohols containing six-membered aromatic rings and other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/22—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrane Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
ESTA INVENCION SE REFIERE A LA PREPARACION DE DERIVADOS DE CROMANOL SUSTITUIDOS Y A INTERMEDIOS UTILES EN DICHA PREPARACION. LOS DERIVADOS DE CROMANOL SUSTITUIDOS QUE SE PREPARAN DE ACUERDO CON LA PRESENTE INVENCION, INHIBEN LA ACCION DE LTB4. ESTOS COMPUESTOS TIENEN LA ESTRUCTURA QUIMICA(V), EN LA QUE X,R1,R2,Y, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2637296P | 1996-09-16 | 1996-09-16 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GT199700104AA true GT199700104AA (es) | 1999-03-28 |
Family
ID=21831429
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GT199700104A GT199700104A (es) | 1996-09-16 | 1997-09-08 | Procedimientos e intermedios para preparar derivados de cromanol sustituidos. |
| GT199700104BL GT199700104BA (es) | 1996-09-16 | 1997-10-04 | Procedimientos e intermedios para preparar derivados de cromanol sustituidos |
| GT199700104AK GT199700104AA (es) | 1996-09-16 | 1997-10-04 | Procedimientos e intermedios para preparar derivados de cromanol sustituidos |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GT199700104A GT199700104A (es) | 1996-09-16 | 1997-09-08 | Procedimientos e intermedios para preparar derivados de cromanol sustituidos. |
| GT199700104BL GT199700104BA (es) | 1996-09-16 | 1997-10-04 | Procedimientos e intermedios para preparar derivados de cromanol sustituidos |
Country Status (39)
| Country | Link |
|---|---|
| US (4) | US6096906A (es) |
| EP (1) | EP0925292B1 (es) |
| JP (1) | JP3117730B2 (es) |
| KR (1) | KR100339164B1 (es) |
| CN (1) | CN1108298C (es) |
| AP (1) | AP726A (es) |
| AT (1) | ATE249452T1 (es) |
| AU (1) | AU713701B2 (es) |
| BG (1) | BG63542B1 (es) |
| BR (1) | BR9711482A (es) |
| CA (1) | CA2265043C (es) |
| CO (1) | CO4600635A1 (es) |
| DE (1) | DE69724801T2 (es) |
| DK (1) | DK0925292T3 (es) |
| DZ (1) | DZ2308A1 (es) |
| EA (1) | EA002204B1 (es) |
| ES (1) | ES2206738T3 (es) |
| GT (3) | GT199700104A (es) |
| HN (1) | HN1997000127A (es) |
| HR (1) | HRP970497B1 (es) |
| ID (1) | ID19613A (es) |
| IL (1) | IL128732A0 (es) |
| IS (1) | IS4980A (es) |
| MA (1) | MA24319A1 (es) |
| NO (1) | NO991254L (es) |
| NZ (1) | NZ334214A (es) |
| OA (1) | OA10995A (es) |
| PA (1) | PA8437901A1 (es) |
| PE (1) | PE109798A1 (es) |
| PL (1) | PL332351A1 (es) |
| PT (1) | PT925292E (es) |
| SK (1) | SK31399A3 (es) |
| TN (1) | TNSN97155A1 (es) |
| TR (1) | TR199900592T2 (es) |
| TW (1) | TW449579B (es) |
| UA (1) | UA58520C2 (es) |
| WO (1) | WO1998011085A1 (es) |
| YU (1) | YU13299A (es) |
| ZA (1) | ZA978291B (es) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6436987B1 (en) * | 2000-06-08 | 2002-08-20 | Pfizer Inc. | Crystalline forms of (3S-trans)-2-[3,4-dihydro-4-hydroxy-3-(phenylmethyl)-2H-1-benzopyran-7-yl]-4-(trifluoromethyl)-benzoic acid |
| JP2004518685A (ja) * | 2001-01-30 | 2004-06-24 | ファイザー・プロダクツ・インク | クロマニル安息香酸の調製方法 |
| AU4239302A (en) * | 2001-06-28 | 2003-01-02 | Pfizer Products Inc. | Benzoic acid substituted benzopyrans for the treatment of atherosclerosis |
| CA2694068C (en) | 2007-07-23 | 2016-08-30 | The Board Of Trustees Of The University Of Illinois | System for controlling the reactivity of boronic acids |
| WO2010036921A2 (en) * | 2008-09-26 | 2010-04-01 | The Board Of Trustees Of The University Of Illinois | Slow release of organoboronic acids in cross-coupling reactions |
| WO2011028766A2 (en) * | 2009-09-02 | 2011-03-10 | E. I. Du Pont De Nemours And Company | Fluorinated 4-oxo-chroman-carboxylates |
| WO2011028767A2 (en) | 2009-09-02 | 2011-03-10 | E. I. Du Pont De Nemours And Company | Fluoroether functionalized aromatic diesters and derivatives thereof |
| TW201113311A (en) * | 2009-09-02 | 2011-04-16 | Du Pont | Polyaramid films comprising fluorovinylether functionalized aromatic moieties |
| BR112012004774A2 (pt) * | 2009-09-02 | 2017-05-30 | Du Pont | polímero e processo |
| US20110218319A1 (en) * | 2009-09-02 | 2011-09-08 | E. I. Du Pont De Nemours And Company | Polyaramid films comprising fluorovinylether functionalized aromatic moieties |
| AU2010289576B2 (en) * | 2009-09-02 | 2015-07-16 | E. I. Du Pont De Nemours And Company | Polyester films with improved oil repellency |
| WO2011103435A2 (en) | 2010-02-18 | 2011-08-25 | The Board Of Trustees Of The University Of Illinois | Methods for forming protected organoboronic acids |
| US10500178B2 (en) | 2015-03-13 | 2019-12-10 | The Board Of Trustees Of The Leland Stanford Junior University | LTB4 inhibition to prevent and treat human lymphedema |
| KR102807066B1 (ko) * | 2019-09-30 | 2025-05-15 | 주식회사 엘지화학 | 아민계 화합물 제조방법 |
| CN117384617B (zh) * | 2023-12-13 | 2024-03-29 | 中国石油大学(华东) | 一种耐盐型胍胶压裂液交联剂水溶液及其制备方法和应用 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9119920D0 (en) * | 1991-09-18 | 1991-10-30 | Glaxo Group Ltd | Chemical compounds |
| MX9300312A (es) * | 1992-01-23 | 1993-07-31 | Pfizer | Antagonistas benzopiranicos y relacionado de ltb. |
| CZ395492A3 (en) * | 1992-01-23 | 1994-03-16 | Pfizer | Benzopyran ltb4 antagonists and related compounds, process of their preparation, intermediates and use |
| CZ100895A3 (en) * | 1992-10-21 | 1995-10-18 | Pfizer | Enantiomeric cis-3-(4,6-dihydroxychroman-3-ylmethyl)benzoic acids |
| CZ100095A3 (en) * | 1992-10-21 | 1995-11-15 | Pfizer | Sulfonamide derivatives of hydroxy substituted alicyclic or heterocyclic compounds with condensed benzene nucleus and pharmaceutical preparations based thereon |
| CN1166834A (zh) * | 1994-10-13 | 1997-12-03 | 美国辉瑞有限公司 | 苯并吡喃和苯并稠合化合物,其制备方法和它们作为白三烯b4(ltb4)拮抗剂的用途 |
| CZ111797A3 (cs) * | 1994-10-13 | 1998-07-15 | Pfizer Inc. | Benzopyranové a jiné sloučeniny s přikondenzovaným benzenovým kruhem a farmaceutické prostředky na jejich bázi |
| US5539128A (en) * | 1994-11-30 | 1996-07-23 | Pfizer Inc. | Processes and intermediates for preparing cis(+)3-[4,6-dihydroxy chroman-3-ylmethyl]-4-methoxyaniline |
-
1997
- 1997-08-25 YU YU13299A patent/YU13299A/sh unknown
- 1997-08-25 PT PT97934679T patent/PT925292E/pt unknown
- 1997-08-25 SK SK313-99A patent/SK31399A3/sk unknown
- 1997-08-25 JP JP10513430A patent/JP3117730B2/ja not_active Expired - Fee Related
- 1997-08-25 UA UA99031394A patent/UA58520C2/uk unknown
- 1997-08-25 NZ NZ334214A patent/NZ334214A/xx unknown
- 1997-08-25 AT AT97934679T patent/ATE249452T1/de not_active IP Right Cessation
- 1997-08-25 KR KR1019997002175A patent/KR100339164B1/ko not_active Expired - Fee Related
- 1997-08-25 DK DK97934679T patent/DK0925292T3/da active
- 1997-08-25 PL PL97332351A patent/PL332351A1/xx unknown
- 1997-08-25 US US09/367,235 patent/US6096906A/en not_active Expired - Fee Related
- 1997-08-25 EA EA199900204A patent/EA002204B1/ru not_active IP Right Cessation
- 1997-08-25 ES ES97934679T patent/ES2206738T3/es not_active Expired - Lifetime
- 1997-08-25 TR TR1999/00592T patent/TR199900592T2/xx unknown
- 1997-08-25 BR BR9711482A patent/BR9711482A/pt not_active Application Discontinuation
- 1997-08-25 DE DE69724801T patent/DE69724801T2/de not_active Expired - Fee Related
- 1997-08-25 EP EP97934679A patent/EP0925292B1/en not_active Expired - Lifetime
- 1997-08-25 CA CA002265043A patent/CA2265043C/en not_active Expired - Fee Related
- 1997-08-25 AU AU37814/97A patent/AU713701B2/en not_active Ceased
- 1997-08-25 WO PCT/IB1997/001024 patent/WO1998011085A1/en not_active Ceased
- 1997-08-25 CN CN97197985A patent/CN1108298C/zh not_active Expired - Fee Related
- 1997-08-25 IL IL12873297A patent/IL128732A0/xx unknown
- 1997-08-29 HN HN1997000127A patent/HN1997000127A/es unknown
- 1997-09-04 CO CO97051475A patent/CO4600635A1/es unknown
- 1997-09-05 PA PA19978437901A patent/PA8437901A1/es unknown
- 1997-09-08 GT GT199700104A patent/GT199700104A/es unknown
- 1997-09-11 AP APAP/P/1997/001083A patent/AP726A/en active
- 1997-09-12 PE PE1997000813A patent/PE109798A1/es not_active Application Discontinuation
- 1997-09-12 TW TW086113297A patent/TW449579B/zh active
- 1997-09-15 ZA ZA978291A patent/ZA978291B/xx unknown
- 1997-09-15 MA MA24797A patent/MA24319A1/fr unknown
- 1997-09-15 TN TNTNSN97155A patent/TNSN97155A1/fr unknown
- 1997-09-15 ID IDP973183A patent/ID19613A/id unknown
- 1997-09-15 DZ DZ970158A patent/DZ2308A1/xx active
- 1997-09-16 HR HR970497A patent/HRP970497B1/xx not_active IP Right Cessation
- 1997-10-04 GT GT199700104BL patent/GT199700104BA/es unknown
- 1997-10-04 GT GT199700104AK patent/GT199700104AA/es unknown
-
1999
- 1999-02-16 IS IS4980A patent/IS4980A/is unknown
- 1999-03-09 BG BG103231A patent/BG63542B1/bg unknown
- 1999-03-12 OA OA9900056A patent/OA10995A/en unknown
- 1999-03-15 NO NO991254A patent/NO991254L/no not_active Application Discontinuation
-
2000
- 2000-02-23 US US09/511,475 patent/US6288242B1/en not_active Expired - Fee Related
-
2001
- 2001-03-21 US US09/813,546 patent/US6355825B1/en not_active Expired - Fee Related
- 2001-10-31 US US09/999,240 patent/US6444826B1/en not_active Expired - Fee Related
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