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GT199700104AA - Procedimientos e intermedios para preparar derivados de cromanol sustituidos - Google Patents

Procedimientos e intermedios para preparar derivados de cromanol sustituidos

Info

Publication number
GT199700104AA
GT199700104AA GT199700104AK GT199700104K GT199700104AA GT 199700104A A GT199700104A A GT 199700104AA GT 199700104A K GT199700104A K GT 199700104AK GT 199700104 K GT199700104 K GT 199700104K GT 199700104A A GT199700104A A GT 199700104AA
Authority
GT
Guatemala
Prior art keywords
intermediates
procedures
chromanol derivatives
substituted chromanol
prepare substituted
Prior art date
Application number
GT199700104AK
Other languages
English (en)
Inventor
Anthony Piscopio
Joel M Hawkins
Stephane Caron
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT199700104AA publication Critical patent/GT199700104AA/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/40Halogenated unsaturated alcohols
    • C07C33/50Halogenated unsaturated alcohols containing six-membered aromatic rings and other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/22Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

ESTA INVENCION SE REFIERE A LA PREPARACION DE DERIVADOS DE CROMANOL SUSTITUIDOS Y A INTERMEDIOS UTILES EN DICHA PREPARACION. LOS DERIVADOS DE CROMANOL SUSTITUIDOS QUE SE PREPARAN DE ACUERDO CON LA PRESENTE INVENCION, INHIBEN LA ACCION DE LTB4. ESTOS COMPUESTOS TIENEN LA ESTRUCTURA QUIMICA(V), EN LA QUE X,R1,R2,Y, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE.
GT199700104AK 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos GT199700104AA (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US2637296P 1996-09-16 1996-09-16

Publications (1)

Publication Number Publication Date
GT199700104AA true GT199700104AA (es) 1999-03-28

Family

ID=21831429

Family Applications (3)

Application Number Title Priority Date Filing Date
GT199700104A GT199700104A (es) 1996-09-16 1997-09-08 Procedimientos e intermedios para preparar derivados de cromanol sustituidos.
GT199700104BL GT199700104BA (es) 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos
GT199700104AK GT199700104AA (es) 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos

Family Applications Before (2)

Application Number Title Priority Date Filing Date
GT199700104A GT199700104A (es) 1996-09-16 1997-09-08 Procedimientos e intermedios para preparar derivados de cromanol sustituidos.
GT199700104BL GT199700104BA (es) 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos

Country Status (39)

Country Link
US (4) US6096906A (es)
EP (1) EP0925292B1 (es)
JP (1) JP3117730B2 (es)
KR (1) KR100339164B1 (es)
CN (1) CN1108298C (es)
AP (1) AP726A (es)
AT (1) ATE249452T1 (es)
AU (1) AU713701B2 (es)
BG (1) BG63542B1 (es)
BR (1) BR9711482A (es)
CA (1) CA2265043C (es)
CO (1) CO4600635A1 (es)
DE (1) DE69724801T2 (es)
DK (1) DK0925292T3 (es)
DZ (1) DZ2308A1 (es)
EA (1) EA002204B1 (es)
ES (1) ES2206738T3 (es)
GT (3) GT199700104A (es)
HN (1) HN1997000127A (es)
HR (1) HRP970497B1 (es)
ID (1) ID19613A (es)
IL (1) IL128732A0 (es)
IS (1) IS4980A (es)
MA (1) MA24319A1 (es)
NO (1) NO991254L (es)
NZ (1) NZ334214A (es)
OA (1) OA10995A (es)
PA (1) PA8437901A1 (es)
PE (1) PE109798A1 (es)
PL (1) PL332351A1 (es)
PT (1) PT925292E (es)
SK (1) SK31399A3 (es)
TN (1) TNSN97155A1 (es)
TR (1) TR199900592T2 (es)
TW (1) TW449579B (es)
UA (1) UA58520C2 (es)
WO (1) WO1998011085A1 (es)
YU (1) YU13299A (es)
ZA (1) ZA978291B (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6436987B1 (en) * 2000-06-08 2002-08-20 Pfizer Inc. Crystalline forms of (3S-trans)-2-[3,4-dihydro-4-hydroxy-3-(phenylmethyl)-2H-1-benzopyran-7-yl]-4-(trifluoromethyl)-benzoic acid
WO2002060888A1 (en) * 2001-01-30 2002-08-08 Pfizer Products Inc. Processes for preparing chromanylbenzoic acids
AU4239302A (en) * 2001-06-28 2003-01-02 Pfizer Products Inc. Benzoic acid substituted benzopyrans for the treatment of atherosclerosis
JP2010534240A (ja) 2007-07-23 2010-11-04 ザ ボード オブ トラスティーズ オブ ザ ユニバーシティ オブ イリノイ ボロン酸の反応性の調節系
WO2010036921A2 (en) * 2008-09-26 2010-04-01 The Board Of Trustees Of The University Of Illinois Slow release of organoboronic acids in cross-coupling reactions
US20110218319A1 (en) * 2009-09-02 2011-09-08 E. I. Du Pont De Nemours And Company Polyaramid films comprising fluorovinylether functionalized aromatic moieties
CN102597060B (zh) * 2009-09-02 2014-05-07 纳幕尔杜邦公司 包含氟乙烯基醚官能化芳族部分的芳族聚酰胺
CN102612509A (zh) 2009-09-02 2012-07-25 纳幕尔杜邦公司 氟醚官能化的芳族二酯及其衍生物
KR20120092105A (ko) * 2009-09-02 2012-08-20 이 아이 듀폰 디 네모아 앤드 캄파니 개선된 발유성을 갖는 폴리에스테르 필름
US8293928B2 (en) * 2009-09-02 2012-10-23 E I Du Pont De Nemours And Company Fluorinated 4-oxo-chroman-7-carboxylates
IN2012DN01745A (es) * 2009-09-02 2015-06-05 Du Pont
WO2011103435A2 (en) * 2010-02-18 2011-08-25 The Board Of Trustees Of The University Of Illinois Methods for forming protected organoboronic acids
US10500178B2 (en) 2015-03-13 2019-12-10 The Board Of Trustees Of The Leland Stanford Junior University LTB4 inhibition to prevent and treat human lymphedema
KR102807066B1 (ko) * 2019-09-30 2025-05-15 주식회사 엘지화학 아민계 화합물 제조방법
CN117384617B (zh) * 2023-12-13 2024-03-29 中国石油大学(华东) 一种耐盐型胍胶压裂液交联剂水溶液及其制备方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9119920D0 (en) * 1991-09-18 1991-10-30 Glaxo Group Ltd Chemical compounds
MX9300312A (es) * 1992-01-23 1993-07-31 Pfizer Antagonistas benzopiranicos y relacionado de ltb.
ES2098547T3 (es) * 1992-01-23 1997-05-01 Pfizer Benzopirano y otros antagonistas de ltb4 relacionados.
CZ100895A3 (en) * 1992-10-21 1995-10-18 Pfizer Enantiomeric cis-3-(4,6-dihydroxychroman-3-ylmethyl)benzoic acids
RU95109929A (ru) * 1992-10-21 1997-03-20 Пфайзер Инк. (US) Сульфонамидные производные, фармацевтическая композиция и способ лечения млекопитающих
WO1996011920A1 (en) * 1994-10-13 1996-04-25 Pfizer Inc. Benzopyran and benzo-fused compounds, their preparation and their use as leukotriene b4 (ltb4) antagonists
CA2202056A1 (en) * 1994-10-13 1996-04-25 Mark A. Dombroski Benzopyran and benzo-fused compounds, their preparation and their use as leukotriene b4' (ltb4) antagonists
US5539128A (en) * 1994-11-30 1996-07-23 Pfizer Inc. Processes and intermediates for preparing cis(+)3-[4,6-dihydroxy chroman-3-ylmethyl]-4-methoxyaniline

Also Published As

Publication number Publication date
KR20000036136A (ko) 2000-06-26
OA10995A (en) 2001-11-06
TW449579B (en) 2001-08-11
US6096906A (en) 2000-08-01
EA002204B1 (ru) 2002-02-28
EA199900204A1 (ru) 1999-08-26
PE109798A1 (es) 1999-01-13
IS4980A (is) 1999-02-16
US6355825B1 (en) 2002-03-12
PL332351A1 (en) 1999-09-13
WO1998011085A1 (en) 1998-03-19
YU13299A (sh) 2001-03-07
PA8437901A1 (es) 2000-05-24
DE69724801T2 (de) 2004-06-17
US20020099227A1 (en) 2002-07-25
EP0925292B1 (en) 2003-09-10
PT925292E (pt) 2004-01-30
US20020042526A1 (en) 2002-04-11
HN1997000127A (es) 1997-12-20
DK0925292T3 (da) 2004-01-12
NO991254D0 (no) 1999-03-15
CA2265043A1 (en) 1998-03-19
AU713701B2 (en) 1999-12-09
DE69724801D1 (de) 2003-10-16
GT199700104A (es) 1999-03-02
TNSN97155A1 (fr) 2005-03-15
TR199900592T2 (xx) 1999-06-21
SK31399A3 (en) 2000-05-16
AP726A (en) 1999-01-29
DZ2308A1 (fr) 2002-12-28
UA58520C2 (uk) 2003-08-15
JP3117730B2 (ja) 2000-12-18
JP2000502726A (ja) 2000-03-07
CO4600635A1 (es) 1998-05-08
CN1108298C (zh) 2003-05-14
IL128732A0 (en) 2000-01-31
MA24319A1 (fr) 1998-04-01
NO991254L (no) 1999-05-14
ES2206738T3 (es) 2004-05-16
AU3781497A (en) 1998-04-02
CA2265043C (en) 2003-01-14
NZ334214A (en) 2000-09-29
HRP970497B1 (en) 2002-06-30
HRP970497A2 (en) 1998-08-31
US6288242B1 (en) 2001-09-11
ATE249452T1 (de) 2003-09-15
BG63542B1 (bg) 2002-04-30
ID19613A (id) 1998-07-23
KR100339164B1 (ko) 2002-06-01
AP9701083A0 (en) 1997-10-31
US6444826B1 (en) 2002-09-03
BR9711482A (pt) 1999-08-24
CN1230954A (zh) 1999-10-06
EP0925292A1 (en) 1999-06-30
BG103231A (en) 1999-12-30
ZA978291B (en) 1999-03-15
GT199700104BA (es) 1999-03-28

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