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FI971610L - Menetelmä syklisten depsipeptidien sulfonyloimiseksi, sulfenyloimiseksi, ja fosforyloimiseksi - Google Patents

Menetelmä syklisten depsipeptidien sulfonyloimiseksi, sulfenyloimiseksi, ja fosforyloimiseksi Download PDF

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Publication number
FI971610L
FI971610L FI971610A FI971610A FI971610L FI 971610 L FI971610 L FI 971610L FI 971610 A FI971610 A FI 971610A FI 971610 A FI971610 A FI 971610A FI 971610 L FI971610 L FI 971610L
Authority
FI
Finland
Prior art keywords
sulfenylation
sulfonylation
phosphorylation
cyclic depsipeptides
depsipeptides
Prior art date
Application number
FI971610A
Other languages
English (en)
Swedish (sv)
Other versions
FI971610A7 (fi
FI971610A0 (fi
Inventor
Juergen Scherkenbeck
Andrew Plant
Peter Jeschke
Achim Harder
Norbert Mencke
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of FI971610A7 publication Critical patent/FI971610A7/fi
Publication of FI971610A0 publication Critical patent/FI971610A0/fi
Publication of FI971610L publication Critical patent/FI971610L/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D273/00Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/26Sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6527Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and oxygen atoms as the only ring hetero atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI971610A 1994-10-18 1995-10-05 Menetelmä syklisten depsipeptidien sulfonyloimiseksi, sulfenyloimiseksi, ja fosforyloimiseksi FI971610L (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4437198A DE4437198A1 (de) 1994-10-18 1994-10-18 Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden
PCT/EP1995/003926 WO1996011945A2 (de) 1994-10-18 1995-10-05 Verfahren zur sulfonylierung, sulfenylierung und phosphorylierung von cyclischen depsipeptiden

Publications (3)

Publication Number Publication Date
FI971610A7 FI971610A7 (fi) 1997-04-16
FI971610A0 FI971610A0 (fi) 1997-04-16
FI971610L true FI971610L (fi) 1997-04-16

Family

ID=6531064

Family Applications (1)

Application Number Title Priority Date Filing Date
FI971610A FI971610L (fi) 1994-10-18 1995-10-05 Menetelmä syklisten depsipeptidien sulfonyloimiseksi, sulfenyloimiseksi, ja fosforyloimiseksi

Country Status (17)

Country Link
US (1) US5874530A (fi)
EP (1) EP0787141B1 (fi)
JP (1) JPH10511341A (fi)
AT (1) ATE195952T1 (fi)
AU (1) AU698898B2 (fi)
BR (1) BR9509377A (fi)
CA (1) CA2202751A1 (fi)
CZ (1) CZ112397A3 (fi)
DE (2) DE4437198A1 (fi)
DK (1) DK0787141T3 (fi)
ES (1) ES2149378T3 (fi)
FI (1) FI971610L (fi)
HU (1) HU218569B (fi)
NZ (1) NZ294843A (fi)
PL (1) PL319649A1 (fi)
SK (1) SK48697A3 (fi)
WO (1) WO1996011945A2 (fi)

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* Cited by examiner, † Cited by third party
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DE4437198A1 (de) * 1994-10-18 1996-04-25 Bayer Ag Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden
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DE19713626A1 (de) * 1997-04-02 1998-10-08 Bayer Ag Neue Thiodepsipeptide zur Bekämpfung von Endoparasiten und ein einfaches Verfahren zu ihrer Herstellung
US6136838A (en) * 1998-03-19 2000-10-24 Merck & Co., Inc. Sulfurpentafluorophenylpyrazoles for controlling ectoparasitic infestations
DE10031044A1 (de) * 2000-06-26 2002-01-03 Bayer Ag Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere
CA2560510C (en) 2004-03-18 2009-10-13 Pfizer Inc. N-(1-arylpyrazol-4yl) sulfonamides and their use as parasiticides
DE102004055316A1 (de) * 2004-11-16 2006-05-18 Bayer Healthcare Ag Verhinderung vertikaler Endoparasiten-Infektionen
DE102008022520A1 (de) 2008-05-07 2009-11-12 Bayer Animal Health Gmbh Feste Arzneimittelformulierung mit verzögerter Freisetzung
DE102008030764A1 (de) 2008-06-28 2009-12-31 Bayer Animal Health Gmbh Kombination von Amidin-Derivaten mit cyclischen Depsipeptiden
DE102008031283A1 (de) * 2008-07-02 2010-01-07 Bayer Schering Pharma Aktiengesellschaft Neue Bekämpfungsmöglichkeit von durch Trichomonadida hervorgerufenen Krankheiten
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CA2202751A1 (en) 1996-04-25
FI971610A7 (fi) 1997-04-16
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DK0787141T3 (da) 2000-12-11
HU218569B (hu) 2000-10-28
WO1996011945A3 (de) 1996-07-25
CZ112397A3 (en) 1997-07-16
DE59508691D1 (de) 2000-10-05
NZ294843A (en) 1998-11-25
FI971610A0 (fi) 1997-04-16
MX9702771A (es) 1997-07-31
US5874530A (en) 1999-02-23
SK48697A3 (en) 1997-11-05
AU698898B2 (en) 1998-11-12
WO1996011945A2 (de) 1996-04-25
PL319649A1 (en) 1997-08-18
ATE195952T1 (de) 2000-09-15
ES2149378T3 (es) 2000-11-01
EP0787141A2 (de) 1997-08-06
HUT77019A (hu) 1998-03-02
EP0787141B1 (de) 2000-08-30
BR9509377A (pt) 1997-11-18
DE4437198A1 (de) 1996-04-25
AU3803895A (en) 1996-05-06

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