FI940530L - Quaternary ammonium derivatives of (-) and (+) 10-(1-azabicyclo(2.2.2.)oct-3-ylmethyl-10-phenothiazine, pharmaceutical compositions containing them and method of preparing them - Google Patents

Quaternary ammonium derivatives of (-) and (+) 10-(1-azabicyclo(2.2.2.)oct-3-ylmethyl-10-phenothiazine, pharmaceutical compositions containing them and method of preparing them Download PDF

Info

Publication number: FI940530L
Authority: FI; Finland
Prior art keywords: azabicyclo; phenothiazine; ylmethyl; oct; preparing
Prior art date: 1991-08-07

Application number

FI940530A

Other languages

Finnish (fi)

Swedish (sv)

Other versions

FI940530A0 (en

FI940530A7 (en

Inventor

Raffaello Giorgi

Alessandro Subissi

Luigi Turbanti

Original Assignee

Guidotti & C Spa Labor

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-08-07

Filing date

1992-08-03

Publication date

1994-02-04

1992-08-03 Application filed by Guidotti & C Spa Labor filed Critical Guidotti & C Spa Labor

1994-02-04 Publication of FI940530A0 publication Critical patent/FI940530A0/en

1994-02-04 Publication of FI940530L publication Critical patent/FI940530L/en

1994-02-04 Publication of FI940530A7 publication Critical patent/FI940530A7/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pulmonology (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Immunology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

FI940530A 1991-08-07 1992-08-03 Quaternary ammonium derivatives of (-) and (+) 10-(1-azabicyclo(2.2.2.)oct-3-ylmethyl-10-phenothiazine, pharmaceutical compositions containing them and method of preparing them FI940530A7 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
ITMI912225A IT1251161B (en)	1991-08-07	1991-08-07	QUATERNARY AMMONIUM DERIVATIVES OF (-) AND (+) - 3- (10 H-PHENOTHIAZIN-10-ILMETHYL) -L-AZABICYCLE (2.2.2.) OCT AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
PCT/EP1992/001759 WO1993003029A1 (en)	1991-08-07	1992-08-03	(-) and (+) 10-(1-azabicyclo[2.2.2.]oct-3-yl-methyl)-10 h-phenothiazine quaternary ammonium derivatives, pharmaceutical compositions containing them and process for their preparation

Publications (3)

Publication Number	Publication Date
FI940530A0 FI940530A0 (en)	1994-02-04
FI940530L true FI940530L (en)	1994-02-04
FI940530A7 FI940530A7 (en)	1994-02-04

Family

ID=11360550

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI940530A FI940530A7 (en)	1991-08-07	1992-08-03	Quaternary ammonium derivatives of (-) and (+) 10-(1-azabicyclo(2.2.2.)oct-3-ylmethyl-10-phenothiazine, pharmaceutical compositions containing them and method of preparing them

Country Status (19)

Country	Link
EP (1)	EP0599896A1 (en)
JP (1)	JPH06509570A (en)
CN (1)	CN1071667A (en)
AU (1)	AU2417392A (en)
BG (1)	BG98439A (en)
BR (1)	BR9206339A (en)
CA (1)	CA2114844A1 (en)
CZ (1)	CZ24894A3 (en)
EC (1)	ECSP920859A (en)
FI (1)	FI940530A7 (en)
HU (1)	HUT66570A (en)
IT (1)	IT1251161B (en)
MA (1)	MA22611A1 (en)
MX (1)	MX9204539A (en)
PT (1)	PT100765A (en)
SK (1)	SK11594A3 (en)
TN (1)	TNSN92073A1 (en)
WO (1)	WO1993003029A1 (en)
ZA (1)	ZA925852B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CN1216353C (en) *	1996-10-18	2005-08-24	雅马哈株式会社	Music teaching system, method and storing media for performing programme
WO2003105811A2 (en) *	2002-01-31	2003-12-24	Southwest Research Institute	Controlled release compositions and methods for using same
FR2910814B1 (en) *	2006-12-28	2011-06-17	Pf Medicament	USE OF 10- (R3) -1-AZABICYCLO2.2.2-OCT-3-YLMETHYL-10H-PHENOTHIAZINE FOR THE PREPARATION OF A MEDICAMENT EXERCISING SELECTIVE INHIBITION OF M1,2,3 MUSCARINIC RECEPTORS
FR2911606B1 (en) *	2007-01-18	2009-04-17	Pierre Fabre Medicament Sa	NEW QUINUCLIDINE DERIVATIVE USEFUL IN THE PREPARATION OF MEQUITAZINE
FR2924344B1 (en) *	2007-12-04	2010-04-16	Pf Medicament	USE OF MEQUITAZINE IN THE FORM OF RACEMATE OR ENANTIOMERS FOR THE PREPARATION OF A MEDICAMENT FOR THE TREATMENT OR PREVENTION OF PATHOLOGIES INVOLVING HISTAMIC RECEPTORS H4.
FR2970255B1 (en) *	2011-01-10	2013-09-06	Pf Medicament	VINYL QUINUCLIDINE USEFUL AS A SYNTHETIC INTERMEDIARY IN THE PREPARATION OF (R) -MEQUITAZINE
JP7599646B2 (en) *	2020-10-29	2024-12-16	国立大学法人金沢大学	Radioactive fluorine-labeled diagnostic imaging agents for measuring drug-metabolizing enzyme activities

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2522660A1 (en) *	1982-03-05	1983-09-09	Pharmuka Lab	MEQUITAZINE LEVOGYER ISOMER, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME
FR2526433B1 (en) *	1982-05-04	1985-10-18	Pharmuka Lab	DEXTROGYRIC ISOMERS OF AZA-1 BICYCLO (2,2,2) OCTANE DERIVATIVES, THEIR PREPARATION METHOD AND MEDICAMENTS CONTAINING THEM
IT1173445B (en) *	1984-03-16	1987-06-24	Guidotti & C Spa Labor	AGENTS WITH ANTIBRONCOSPASTIC ACTIVITY AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM

1991
- 1991-08-07 IT ITMI912225A patent/IT1251161B/en active IP Right Grant
1992
- 1992-08-03 AU AU24173/92A patent/AU2417392A/en not_active Abandoned
- 1992-08-03 MA MA22900A patent/MA22611A1/en unknown
- 1992-08-03 JP JP5503276A patent/JPH06509570A/en active Pending
- 1992-08-03 WO PCT/EP1992/001759 patent/WO1993003029A1/en not_active Ceased
- 1992-08-03 SK SK115-94A patent/SK11594A3/en unknown
- 1992-08-03 CZ CS94248A patent/CZ24894A3/en unknown
- 1992-08-03 EP EP92916942A patent/EP0599896A1/en not_active Ceased
- 1992-08-03 HU HU9400273A patent/HUT66570A/en unknown
- 1992-08-03 BR BR9206339A patent/BR9206339A/en not_active Application Discontinuation
- 1992-08-03 FI FI940530A patent/FI940530A7/en not_active Application Discontinuation
- 1992-08-03 CA CA002114844A patent/CA2114844A1/en not_active Abandoned
- 1992-08-04 ZA ZA925852A patent/ZA925852B/en unknown
- 1992-08-04 EC EC1992000859A patent/ECSP920859A/en unknown
- 1992-08-05 MX MX9204539A patent/MX9204539A/en unknown
- 1992-08-05 TN TNTNSN92073A patent/TNSN92073A1/en unknown
- 1992-08-06 CN CN92109021A patent/CN1071667A/en active Pending
- 1992-08-07 PT PT100765A patent/PT100765A/en not_active Application Discontinuation
1994
- 1994-02-07 BG BG98439A patent/BG98439A/en unknown

Also Published As

Publication number	Publication date
SK11594A3 (en)	1994-12-07
BR9206339A (en)	1994-11-08
HUT66570A (en)	1994-12-28
TNSN92073A1 (en)	1993-06-08
MX9204539A (en)	1993-02-01
BG98439A (en)	1994-09-30
ECSP920859A (en)	1993-08-03
ZA925852B (en)	1993-03-05
PT100765A (en)	1993-10-29
ITMI912225A1 (en)	1993-02-07
WO1993003029A1 (en)	1993-02-18
ITMI912225A0 (en)	1991-08-07
CA2114844A1 (en)	1993-02-18
MA22611A1 (en)	1993-04-01
FI940530A0 (en)	1994-02-04
CN1071667A (en)	1993-05-05
FI940530A7 (en)	1994-02-04
JPH06509570A (en)	1994-10-27
IT1251161B (en)	1995-05-04
AU2417392A (en)	1993-03-02
HU9400273D0 (en)	1994-05-30
CZ24894A3 (en)	1994-07-13
EP0599896A1 (en)	1994-06-08

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Legal Events

Date	Code	Title	Description
1997-02-28	FD	Application lapsed