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FI913800L - 3-(1,2-bensisoxazol-3-yl) -4-pyridinaminer och derivat daerav. - Google Patents

3-(1,2-bensisoxazol-3-yl) -4-pyridinaminer och derivat daerav. Download PDF

Info

Publication number
FI913800L
FI913800L FI913800A FI913800A FI913800L FI 913800 L FI913800 L FI 913800L FI 913800 A FI913800 A FI 913800A FI 913800 A FI913800 A FI 913800A FI 913800 L FI913800 L FI 913800L
Authority
FI
Finland
Prior art keywords
pyridinaminer
bensisoxazol
derivats
daerav
och
Prior art date
Application number
FI913800A
Other languages
English (en)
Other versions
FI103970B1 (fi
FI913800A0 (fi
FI103970B (fi
Inventor
Joseph Thomas Klein
Richard Charles Effland
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of FI913800A0 publication Critical patent/FI913800A0/fi
Publication of FI913800L publication Critical patent/FI913800L/fi
Application granted granted Critical
Publication of FI103970B1 publication Critical patent/FI103970B1/fi
Publication of FI103970B publication Critical patent/FI103970B/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
FI913800A 1990-08-13 1991-08-09 Menetelmä kivun lievittämiseen sekä ihotautien ja muistin toimintahäiriöiden hoitoon tarkoitettujen 3-(1,2-bentsisoksatsol-3-yyli)-4-pyridiiniamiinien ja näiden johdannaisten valmistamiseksi FI103970B (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/566,932 US5055476A (en) 1990-08-13 1990-08-13 3-(1,2-benzisoxazol-3-yl)-4-pyridinamines and derivatives
US56693290 1990-08-13

Publications (4)

Publication Number Publication Date
FI913800A0 FI913800A0 (fi) 1991-08-09
FI913800L true FI913800L (fi) 1992-02-14
FI103970B1 FI103970B1 (fi) 1999-10-29
FI103970B FI103970B (fi) 1999-10-29

Family

ID=24265033

Family Applications (1)

Application Number Title Priority Date Filing Date
FI913800A FI103970B (fi) 1990-08-13 1991-08-09 Menetelmä kivun lievittämiseen sekä ihotautien ja muistin toimintahäiriöiden hoitoon tarkoitettujen 3-(1,2-bentsisoksatsol-3-yyli)-4-pyridiiniamiinien ja näiden johdannaisten valmistamiseksi

Country Status (24)

Country Link
US (1) US5055476A (fi)
EP (1) EP0471297B1 (fi)
JP (1) JP3057829B2 (fi)
KR (1) KR100191386B1 (fi)
AT (1) ATE130004T1 (fi)
AU (1) AU633791B2 (fi)
CA (1) CA2048959C (fi)
CZ (1) CZ280568B6 (fi)
DE (1) DE69114405T2 (fi)
DK (1) DK0471297T3 (fi)
ES (1) ES2079531T3 (fi)
FI (1) FI103970B (fi)
GR (1) GR3018184T3 (fi)
HU (1) HU213201B (fi)
IE (1) IE70597B1 (fi)
IL (1) IL99166A (fi)
MX (1) MX9100639A (fi)
NO (1) NO179519C (fi)
NZ (1) NZ239326A (fi)
PT (1) PT98645B (fi)
RU (1) RU2012561C1 (fi)
TW (1) TW202446B (fi)
YU (1) YU140991A (fi)
ZA (1) ZA916342B (fi)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5308826A (en) * 1993-04-22 1994-05-03 Zeneca Limited Herbicidal 4-substituted pyridyl-3-carbinols
ZA953390B (en) * 1994-05-02 1996-01-12 Zeneca Ltd Herbicidal hydroxybenzyl-substituted heteroaryl compounds and derivatives thereof
US5595958A (en) * 1994-05-02 1997-01-21 Zeneca Limited 3-substituted pyridine compounds and derivatives thereof
EP0863897B1 (fr) * 1995-11-09 1999-06-16 Synthelabo Derives de 5-phenyl-3-(piperidin-4-yl)-1,3,4-oxadiazol-2(3h)-one, utiles comme ligands des recepteurs 5-ht4 ou h3
FR2762316B1 (fr) * 1997-04-18 1999-12-17 Sanofi Synthelabo Derives de 5-aryl-3-(8-azabicyclo[3.2.1] octan-3-yl)-1,3,4- oxadiazol-2(3h)-one, leur preparation et leur application en therapeutique
US9073947B2 (en) * 2011-06-10 2015-07-07 Merck Patent Gmbh Compositions and methods for the production of pyrimidine and pyridine compounds with BTK inhibitory activity
RU2626650C2 (ru) * 2015-08-31 2017-07-31 Федеральное государственное бюджетное образовательное учреждение высшего образования "Пермский государственный национальный исследовательский университет" 2-Арил-2,4-дигидрокси-2,5-дигидро-3-гетерил-5-оксо-1Н-пиррол-1-ил-4-метилбелзолсульфаниламиды, обладающие анальгетической активностью
WO2023083445A1 (en) 2021-11-10 2023-05-19 Symrise Ag Compositions comprising trpm8 agonistic cooling agents

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4355037A (en) * 1981-11-12 1982-10-19 Hoechst-Roussel Pharmaceuticals 3-(4-Piperidyl)-1,2-benzisoxales
IL66866A (en) * 1982-04-09 1987-08-31 Hoechst Roussel Pharma 1-(3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl)-4-(substituted)-piperazines and-piperidines,a process for the preparation thereof,and pharmaceutical compositions containing them
CA1335289C (en) * 1987-10-26 1995-04-18 Fujio Antoku Piperidinyl benzisoxazole derivatives, their production and pharmaceutical use
IE74711B1 (en) * 1990-07-27 1997-07-30 Ici Plc Fungicides

Also Published As

Publication number Publication date
HU912673D0 (en) 1992-01-28
DE69114405D1 (de) 1995-12-14
FI103970B1 (fi) 1999-10-29
PT98645A (pt) 1992-06-30
GR3018184T3 (en) 1996-02-29
NO179519B (no) 1996-07-15
NZ239326A (en) 1994-04-27
MX9100639A (es) 1992-04-01
KR100191386B1 (ko) 1999-06-15
US5055476A (en) 1991-10-08
HUT61755A (en) 1993-03-01
EP0471297B1 (en) 1995-11-08
IL99166A (en) 1995-12-08
TW202446B (fi) 1993-03-21
NO913142D0 (no) 1991-08-12
DK0471297T3 (da) 1996-03-04
RU2012561C1 (ru) 1994-05-15
IL99166A0 (en) 1992-07-15
IE70597B1 (en) 1996-12-11
FI913800A0 (fi) 1991-08-09
HU213201B (en) 1997-03-28
AU633791B2 (en) 1993-02-04
FI103970B (fi) 1999-10-29
AU8176591A (en) 1992-02-20
ATE130004T1 (de) 1995-11-15
CS248991A3 (en) 1992-03-18
CA2048959C (en) 2003-07-29
JPH05112562A (ja) 1993-05-07
IE912851A1 (en) 1992-02-26
PT98645B (pt) 1999-01-29
YU140991A (sh) 1995-01-31
JP3057829B2 (ja) 2000-07-04
CA2048959A1 (en) 1992-02-14
ZA916342B (en) 1992-04-29
NO913142L (no) 1992-02-14
KR920004383A (ko) 1992-03-27
NO179519C (no) 1996-10-23
DE69114405T2 (de) 1996-05-02
EP0471297A1 (en) 1992-02-19
ES2079531T3 (es) 1996-01-16
CZ280568B6 (cs) 1996-02-14

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Legal Events

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Owner name: HOECHST MARION ROUSSEL, INC.