FI923458L - 4,5-cykloalkano-3-benzazepin-7-ol- derivat och deras anvaendning. - Google Patents
4,5-cykloalkano-3-benzazepin-7-ol- derivat och deras anvaendning. Download PDFInfo
- Publication number
- FI923458L FI923458L FI923458A FI923458A FI923458L FI 923458 L FI923458 L FI 923458L FI 923458 A FI923458 A FI 923458A FI 923458 A FI923458 A FI 923458A FI 923458 L FI923458 L FI 923458L
- Authority
- FI
- Finland
- Prior art keywords
- derivats
- cycloalkano
- benzazepine
- och deras
- deras anvaendning
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D223/18—Dibenzazepines; Hydrogenated dibenzazepines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D223/32—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems containing carbocyclic rings other than six-membered
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Addiction (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US47442890A | 1990-02-02 | 1990-02-02 | |
| PCT/US1991/000503 WO1991011437A1 (en) | 1990-02-02 | 1991-01-31 | 4,5-cycloalkano-3-benzazepin-7-ol-derivatives and their use |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| FI923458L true FI923458L (fi) | 1992-07-31 |
| FI923458A0 FI923458A0 (fi) | 1992-07-31 |
| FI923458A7 FI923458A7 (fi) | 1992-07-31 |
Family
ID=23883493
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI923458A FI923458A7 (fi) | 1990-02-02 | 1991-01-31 | 4,5-sykloalkano-3-bentsatsepin-7-olijohdannaiset ja niiden käyttö |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US5362728A (fi) |
| EP (1) | EP0513174B1 (fi) |
| JP (1) | JPH0613474B2 (fi) |
| KR (1) | KR927003537A (fi) |
| AT (1) | ATE126511T1 (fi) |
| AU (1) | AU646432B2 (fi) |
| CA (1) | CA2075181C (fi) |
| DE (1) | DE69112201T2 (fi) |
| ES (1) | ES2075429T3 (fi) |
| FI (1) | FI923458A7 (fi) |
| OA (1) | OA09662A (fi) |
| WO (1) | WO1991011437A1 (fi) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2713641B1 (fr) * | 1993-12-09 | 1997-04-11 | Egyt Gyogyszervegyeszeti Gyar | Dérivés de l'épi-épibatidine. |
| DK0933993T3 (da) | 1996-06-14 | 2006-08-14 | Biocryst Pharm Inc | Substituerede cyclopentanforbindelser, der er egnede som neuraminidaseinhibitorer |
| AU728332B2 (en) * | 1997-06-23 | 2001-01-04 | Kioka Gaishi Kogyo Kabushiki Kaisha | Lock nut and attaching/removing tool for the same |
| EP1040094B9 (en) * | 1997-12-17 | 2015-09-09 | Biocryst Pharmaceuticals Inc. | Substituted cyclopentane and cyclopentene compounds useful as neuraminidase inhibitors |
| WO2000028328A1 (en) | 1998-11-05 | 2000-05-18 | Biocryst Pharmaceuticals, Inc. | New cyclopentane and cyclopentene compounds and use for detecting influenza virus |
| US7411093B2 (en) * | 2004-12-20 | 2008-08-12 | Hoffman-La Roche Inc. | Aminocycloalkanes as DPP-IV inhibitors |
| NZ565461A (en) * | 2005-08-30 | 2011-08-26 | Abbott Lab | Pharmaceutical compositions as inhibitors of dipeptidyl peptidase-IV (DPP-IV) |
| AU2008259841B2 (en) | 2007-05-31 | 2015-02-05 | Sunovion Pharmaceuticals Inc. | Phenyl substituted cycloalkylamines as monoamine reuptake inhibitors |
| SG10201506896RA (en) | 2010-09-01 | 2015-10-29 | Arena Pharm Inc | Administration of lorcaserin to individuals with renal impairment |
| US20130315994A1 (en) | 2010-09-01 | 2013-11-28 | Zezhi Jesse Shao | Modified-release dosage forms of 5-ht2c agonists useful for weight management |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3393192A (en) * | 1965-04-26 | 1968-07-16 | Schering Corp | Novel benzazepines |
| GB1118688A (en) * | 1967-02-17 | 1968-07-03 | Scherico Ltd | Novel benzazepines and process for making same |
| CH481110A (de) * | 1967-02-17 | 1969-11-15 | Geigy Ag J R | Verfahren zur Herstellung von 1,2,4,5-Tetrahydro-3-azepinen |
| US3609138A (en) * | 1967-12-22 | 1971-09-28 | Ciba Geigy Corp | 1-aryl-3-benzazepines |
| US3752892A (en) * | 1970-03-11 | 1973-08-14 | Ciba Geigy Corp | Anorexigenic tetrahydrobenzazepine derivative method and composition thereof |
| US4011319A (en) * | 1975-07-02 | 1977-03-08 | Smithkline Corporation | Pharmaceutical compositions and methods involving benzazepine derivatives |
| US4284555A (en) * | 1979-04-27 | 1981-08-18 | Schering Corporation | 7-Chloro-8(substituted amino carbonyloxy)-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepines |
| US4477378A (en) * | 1980-02-05 | 1984-10-16 | Schering Corp. | Esters of substituted 8-hydroxy-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepines |
| WO1987004430A2 (en) * | 1986-01-16 | 1987-07-30 | Schering Corporation | Fused benzazepines |
| US4973586A (en) * | 1986-01-16 | 1990-11-27 | Schering Corporation | Fused benzazepines, compositions of, and medical use thereof |
| ATE78467T1 (de) * | 1987-07-15 | 1992-08-15 | Schering Corp | Kondensierte benzazepine. |
-
1991
- 1991-01-31 JP JP3504442A patent/JPH0613474B2/ja not_active Expired - Fee Related
- 1991-01-31 FI FI923458A patent/FI923458A7/fi not_active Application Discontinuation
- 1991-01-31 ES ES91904114T patent/ES2075429T3/es not_active Expired - Lifetime
- 1991-01-31 AU AU72432/91A patent/AU646432B2/en not_active Ceased
- 1991-01-31 WO PCT/US1991/000503 patent/WO1991011437A1/en not_active Ceased
- 1991-01-31 DE DE69112201T patent/DE69112201T2/de not_active Expired - Fee Related
- 1991-01-31 US US07/915,710 patent/US5362728A/en not_active Expired - Lifetime
- 1991-01-31 EP EP91904114A patent/EP0513174B1/en not_active Expired - Lifetime
- 1991-01-31 CA CA002075181A patent/CA2075181C/en not_active Expired - Fee Related
- 1991-01-31 AT AT91904114T patent/ATE126511T1/de not_active IP Right Cessation
-
1992
- 1992-01-31 KR KR1019920701831A patent/KR927003537A/ko not_active Ceased
- 1992-07-31 OA OA60254A patent/OA09662A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES2075429T3 (es) | 1995-10-01 |
| OA09662A (en) | 1993-05-15 |
| KR927003537A (ko) | 1992-12-18 |
| ATE126511T1 (de) | 1995-09-15 |
| DE69112201D1 (de) | 1995-09-21 |
| JPH05504769A (ja) | 1993-07-22 |
| FI923458A0 (fi) | 1992-07-31 |
| US5362728A (en) | 1994-11-08 |
| EP0513174A1 (en) | 1992-11-19 |
| DE69112201T2 (de) | 1996-02-15 |
| CA2075181C (en) | 1997-12-09 |
| WO1991011437A1 (en) | 1991-08-08 |
| EP0513174B1 (en) | 1995-08-16 |
| AU7243291A (en) | 1991-08-21 |
| JPH0613474B2 (ja) | 1994-02-23 |
| FI923458A7 (fi) | 1992-07-31 |
| AU646432B2 (en) | 1994-02-24 |
| CA2075181A1 (en) | 1991-08-03 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD | Application lapsed |