ES500382A0 - Un procedimiento para la preparacion de derivados de triazo-lopiridazina - Google Patents
Un procedimiento para la preparacion de derivados de triazo-lopiridazinaInfo
- Publication number
- ES500382A0 ES500382A0 ES500382A ES500382A ES500382A0 ES 500382 A0 ES500382 A0 ES 500382A0 ES 500382 A ES500382 A ES 500382A ES 500382 A ES500382 A ES 500382A ES 500382 A0 ES500382 A0 ES 500382A0
- Authority
- ES
- Spain
- Prior art keywords
- lopiridazine
- triazo
- derivatives
- procedure
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D249/12—Oxygen or sulfur atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB7925576 | 1979-07-23 | ||
| GB8013203 | 1980-04-22 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8201580A1 ES8201580A1 (es) | 1982-01-01 |
| ES500382A0 true ES500382A0 (es) | 1982-01-01 |
Family
ID=26272284
Family Applications (5)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES493579A Expired ES8106306A1 (es) | 1979-07-23 | 1980-07-22 | Un procedimiento para la preparacion de derivados de triazo-lopiridazina |
| ES500383A Granted ES500383A0 (es) | 1979-07-23 | 1981-03-16 | Un procedimiento para la preparacion de derivados de triazo-lopiridazina |
| ES500382A Granted ES500382A0 (es) | 1979-07-23 | 1981-03-16 | Un procedimiento para la preparacion de derivados de triazo-lopiridazina |
| ES500384A Granted ES500384A0 (es) | 1979-07-23 | 1981-03-16 | Un procedimiento para la preparacion de derivados de triazo-lopiridazina |
| ES500385A Granted ES500385A0 (es) | 1979-07-23 | 1981-03-16 | Un procedimiento para la preparacion de derivados de triazo-lopiridazina |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES493579A Expired ES8106306A1 (es) | 1979-07-23 | 1980-07-22 | Un procedimiento para la preparacion de derivados de triazo-lopiridazina |
| ES500383A Granted ES500383A0 (es) | 1979-07-23 | 1981-03-16 | Un procedimiento para la preparacion de derivados de triazo-lopiridazina |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES500384A Granted ES500384A0 (es) | 1979-07-23 | 1981-03-16 | Un procedimiento para la preparacion de derivados de triazo-lopiridazina |
| ES500385A Granted ES500385A0 (es) | 1979-07-23 | 1981-03-16 | Un procedimiento para la preparacion de derivados de triazo-lopiridazina |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US4307094A (es) |
| EP (1) | EP0024309A3 (es) |
| AR (1) | AR229089A1 (es) |
| AU (1) | AU6044380A (es) |
| CA (1) | CA1137087A (es) |
| DK (1) | DK316480A (es) |
| ES (5) | ES8106306A1 (es) |
| FI (1) | FI802308A7 (es) |
| GR (1) | GR69719B (es) |
| HU (1) | HU180159B (es) |
| IL (1) | IL60617A0 (es) |
| MC (1) | MC1334A1 (es) |
| NO (1) | NO802206L (es) |
| PH (1) | PH16228A (es) |
| PT (1) | PT71587B (es) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0042100A1 (de) * | 1980-06-13 | 1981-12-23 | F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft | Pyrazolopyridazin-Derivate, Zwischenprodukte und Verfahren zu deren Herstellung, sowie diese enthaltende Arzneimittel |
| ZA833214B (en) * | 1982-05-12 | 1983-12-28 | Hoffmann La Roche | Bicyclic compounds |
| GB2128984B (en) * | 1982-05-12 | 1985-05-22 | Hoffmann La Roche | Diaza-bicyclic compounds |
| US4692438A (en) * | 1984-08-24 | 1987-09-08 | Hoffmann-La Roche Inc. | Pyridazo-diazepines, diazocines, and -triazepines having anti-hypertensive activity |
| US4619687A (en) * | 1984-09-27 | 1986-10-28 | Sumitomo Chemical Company, Limited | Triazolopyridazines and their use as herbicides |
| ZW11586A1 (en) * | 1985-07-01 | 1987-12-30 | Hoffmann La Roche | Bicyclic compounds |
| EP0440119A1 (en) * | 1990-01-31 | 1991-08-07 | Takeda Chemical Industries, Ltd. | Imidazopyridazine compounds, their production and use |
| AU1339092A (en) * | 1991-12-13 | 1993-07-19 | Corvas International, Inc. | Reagents for automated synthesis of peptide analogs |
| US6020331A (en) | 1995-03-24 | 2000-02-01 | Molecumetics, Ltd. | β-sheet mimetics and use thereof as protease inhibitors |
| US6699869B1 (en) * | 1995-03-24 | 2004-03-02 | Myriad Genetics Inc. | β-sheet mimetics and use thereof as inhibitors of biologically active peptides or proteins |
| US6245764B1 (en) | 1995-03-24 | 2001-06-12 | Molecumetics Ltd. | β-sheet mimetics and use thereof as inhibitors of biologically active peptides or proteins |
| US6117896A (en) * | 1997-02-10 | 2000-09-12 | Molecumetics Ltd. | Methods for regulating transcription factors |
| EP0915700B1 (en) * | 1996-08-05 | 2006-03-22 | Myriad Genetics, Inc. | Use of beta-sheet mimetics as protease and kinase inhibitors and as inhibitors of transcription factors |
| EP1661566A3 (en) * | 1996-08-05 | 2008-04-16 | Myriad Genetics, Inc. | Use of beta-sheet mimetics as protease and kinase inhibitors and as inhibitors of transcription factors |
| WO2000011005A1 (en) * | 1998-08-21 | 2000-03-02 | Axys Pharmaceuticals, Inc. | Process for the synthesis of triazolopyridazine compounds |
| CN1642550A (zh) | 2002-02-14 | 2005-07-20 | 美瑞德生物工程公司 | β-折叠模拟物和组合物及其有关方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3663564A (en) * | 1958-06-19 | 1972-05-16 | Knoll Pharmaceutical Co | Urazoles and their production |
| US3621099A (en) * | 1969-03-05 | 1971-11-16 | Charles R Jacobson | Therapeutic compositions and methods for stimulating the central nervous system |
| DE2526358A1 (de) | 1974-06-19 | 1976-01-08 | Mitsubishi Chem Ind | 1,2-alkylenurazolderivate, ihre herstellung und verwendung als herbizid |
-
1979
- 1979-07-17 IL IL60617A patent/IL60617A0/xx unknown
-
1980
- 1980-06-25 CA CA000354734A patent/CA1137087A/en not_active Expired
- 1980-07-16 AU AU60443/80A patent/AU6044380A/en not_active Abandoned
- 1980-07-17 US US06/169,571 patent/US4307094A/en not_active Expired - Lifetime
- 1980-07-21 GR GR62511A patent/GR69719B/el unknown
- 1980-07-22 EP EP80104300A patent/EP0024309A3/de not_active Withdrawn
- 1980-07-22 ES ES493579A patent/ES8106306A1/es not_active Expired
- 1980-07-22 PT PT71587A patent/PT71587B/pt unknown
- 1980-07-22 MC MC801459A patent/MC1334A1/fr unknown
- 1980-07-22 NO NO802206A patent/NO802206L/no unknown
- 1980-07-22 FI FI802308A patent/FI802308A7/fi not_active Application Discontinuation
- 1980-07-22 DK DK316480A patent/DK316480A/da not_active Application Discontinuation
- 1980-07-23 PH PH24329A patent/PH16228A/en unknown
- 1980-07-23 AR AR281879A patent/AR229089A1/es active
- 1980-07-23 HU HU80801837A patent/HU180159B/hu unknown
-
1981
- 1981-03-16 ES ES500383A patent/ES500383A0/es active Granted
- 1981-03-16 ES ES500382A patent/ES500382A0/es active Granted
- 1981-03-16 ES ES500384A patent/ES500384A0/es active Granted
- 1981-03-16 ES ES500385A patent/ES500385A0/es active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| CA1137087A (en) | 1982-12-07 |
| EP0024309A3 (de) | 1981-07-22 |
| ES8201582A1 (es) | 1982-01-01 |
| ES8201583A1 (es) | 1982-01-01 |
| IL60617A0 (en) | 1980-09-16 |
| ES493579A0 (es) | 1981-06-16 |
| AR229089A1 (es) | 1983-06-15 |
| PT71587A (en) | 1980-08-01 |
| AU6044380A (en) | 1981-01-29 |
| DK316480A (da) | 1981-01-24 |
| PH16228A (en) | 1983-08-09 |
| ES8201581A1 (es) | 1982-01-01 |
| FI802308A7 (fi) | 1981-01-01 |
| ES8201580A1 (es) | 1982-01-01 |
| ES500383A0 (es) | 1982-01-01 |
| PT71587B (en) | 1981-12-17 |
| NO802206L (no) | 1981-01-26 |
| ES8106306A1 (es) | 1981-06-16 |
| ES500385A0 (es) | 1982-01-01 |
| GR69719B (es) | 1982-07-09 |
| EP0024309A2 (de) | 1981-03-04 |
| US4307094A (en) | 1981-12-22 |
| ES500384A0 (es) | 1982-01-01 |
| MC1334A1 (fr) | 1981-04-21 |
| HU180159B (en) | 1983-02-28 |
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