AR229089A1 - Procedimiento para la preparacion de derivados de acido 2--(mercaptometil,-etil o-propil)-1,3-dioxo-1h-1,2,4-triazolo(1,2-a)piridazin-5-carboxilico - Google Patents
Procedimiento para la preparacion de derivados de acido 2--(mercaptometil,-etil o-propil)-1,3-dioxo-1h-1,2,4-triazolo(1,2-a)piridazin-5-carboxilicoInfo
- Publication number
- AR229089A1 AR229089A1 AR281879A AR28187980A AR229089A1 AR 229089 A1 AR229089 A1 AR 229089A1 AR 281879 A AR281879 A AR 281879A AR 28187980 A AR28187980 A AR 28187980A AR 229089 A1 AR229089 A1 AR 229089A1
- Authority
- AR
- Argentina
- Prior art keywords
- mercaptometil
- piridazin
- carboxilico
- propil
- etil
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D249/12—Oxygen or sulfur atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB7925576 | 1979-07-23 | ||
| GB8013203 | 1980-04-22 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR229089A1 true AR229089A1 (es) | 1983-06-15 |
Family
ID=26272284
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AR281879A AR229089A1 (es) | 1979-07-23 | 1980-07-23 | Procedimiento para la preparacion de derivados de acido 2--(mercaptometil,-etil o-propil)-1,3-dioxo-1h-1,2,4-triazolo(1,2-a)piridazin-5-carboxilico |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US4307094A (es) |
| EP (1) | EP0024309A3 (es) |
| AR (1) | AR229089A1 (es) |
| AU (1) | AU6044380A (es) |
| CA (1) | CA1137087A (es) |
| DK (1) | DK316480A (es) |
| ES (5) | ES493579A0 (es) |
| FI (1) | FI802308A7 (es) |
| GR (1) | GR69719B (es) |
| HU (1) | HU180159B (es) |
| IL (1) | IL60617A0 (es) |
| MC (1) | MC1334A1 (es) |
| NO (1) | NO802206L (es) |
| PH (1) | PH16228A (es) |
| PT (1) | PT71587B (es) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0042100A1 (de) * | 1980-06-13 | 1981-12-23 | F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft | Pyrazolopyridazin-Derivate, Zwischenprodukte und Verfahren zu deren Herstellung, sowie diese enthaltende Arzneimittel |
| NZ204130A (en) * | 1982-05-12 | 1986-03-14 | Hoffmann La Roche | Bicyclic heterocyclic compounds and pharmaceutical compositions |
| GB2128984B (en) * | 1982-05-12 | 1985-05-22 | Hoffmann La Roche | Diaza-bicyclic compounds |
| US4692438A (en) * | 1984-08-24 | 1987-09-08 | Hoffmann-La Roche Inc. | Pyridazo-diazepines, diazocines, and -triazepines having anti-hypertensive activity |
| US4619687A (en) * | 1984-09-27 | 1986-10-28 | Sumitomo Chemical Company, Limited | Triazolopyridazines and their use as herbicides |
| ZW11586A1 (en) * | 1985-07-01 | 1987-12-30 | Hoffmann La Roche | Bicyclic compounds |
| EP0440119A1 (en) * | 1990-01-31 | 1991-08-07 | Takeda Chemical Industries, Ltd. | Imidazopyridazine compounds, their production and use |
| WO1993012076A1 (en) * | 1991-12-13 | 1993-06-24 | Corvas International Inc. | Reagents for automated synthesis of peptide analogs |
| US6245764B1 (en) | 1995-03-24 | 2001-06-12 | Molecumetics Ltd. | β-sheet mimetics and use thereof as inhibitors of biologically active peptides or proteins |
| US6020331A (en) | 1995-03-24 | 2000-02-01 | Molecumetics, Ltd. | β-sheet mimetics and use thereof as protease inhibitors |
| US6699869B1 (en) | 1995-03-24 | 2004-03-02 | Myriad Genetics Inc. | β-sheet mimetics and use thereof as inhibitors of biologically active peptides or proteins |
| EP1661566A3 (en) * | 1996-08-05 | 2008-04-16 | Myriad Genetics, Inc. | Use of beta-sheet mimetics as protease and kinase inhibitors and as inhibitors of transcription factors |
| US6117896A (en) | 1997-02-10 | 2000-09-12 | Molecumetics Ltd. | Methods for regulating transcription factors |
| ATE320811T1 (de) * | 1996-08-05 | 2006-04-15 | Myriad Genetics Inc | Verwendung von beta-blatt mimetika als protease und kinase hemmer und alshemmer eines transkriptionsfaktors |
| AU5571099A (en) * | 1998-08-21 | 2000-03-14 | Axys Pharmaceuticals, Inc. | Process for the synthesis of triazolopyridazine compounds |
| JP2005526722A (ja) * | 2002-02-14 | 2005-09-08 | ミリアド・ジェネティックス・インコーポレイテッド | β−シートミメティックならびにそれに関連する組成物および方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3663564A (en) * | 1958-06-19 | 1972-05-16 | Knoll Pharmaceutical Co | Urazoles and their production |
| US3621099A (en) * | 1969-03-05 | 1971-11-16 | Charles R Jacobson | Therapeutic compositions and methods for stimulating the central nervous system |
| DE2526358A1 (de) * | 1974-06-19 | 1976-01-08 | Mitsubishi Chem Ind | 1,2-alkylenurazolderivate, ihre herstellung und verwendung als herbizid |
-
1979
- 1979-07-17 IL IL60617A patent/IL60617A0/xx unknown
-
1980
- 1980-06-25 CA CA000354734A patent/CA1137087A/en not_active Expired
- 1980-07-16 AU AU60443/80A patent/AU6044380A/en not_active Abandoned
- 1980-07-17 US US06/169,571 patent/US4307094A/en not_active Expired - Lifetime
- 1980-07-21 GR GR62511A patent/GR69719B/el unknown
- 1980-07-22 EP EP80104300A patent/EP0024309A3/de not_active Withdrawn
- 1980-07-22 FI FI802308A patent/FI802308A7/fi not_active Application Discontinuation
- 1980-07-22 DK DK316480A patent/DK316480A/da not_active Application Discontinuation
- 1980-07-22 NO NO802206A patent/NO802206L/no unknown
- 1980-07-22 MC MC801459A patent/MC1334A1/fr unknown
- 1980-07-22 ES ES493579A patent/ES493579A0/es active Granted
- 1980-07-22 PT PT71587A patent/PT71587B/pt unknown
- 1980-07-23 PH PH24329A patent/PH16228A/en unknown
- 1980-07-23 HU HU80801837A patent/HU180159B/hu unknown
- 1980-07-23 AR AR281879A patent/AR229089A1/es active
-
1981
- 1981-03-16 ES ES500383A patent/ES8201581A1/es not_active Expired
- 1981-03-16 ES ES500382A patent/ES8201580A1/es not_active Expired
- 1981-03-16 ES ES500384A patent/ES500384A0/es active Granted
- 1981-03-16 ES ES500385A patent/ES500385A0/es active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| NO802206L (no) | 1981-01-26 |
| HU180159B (en) | 1983-02-28 |
| PH16228A (en) | 1983-08-09 |
| ES8106306A1 (es) | 1981-06-16 |
| ES500382A0 (es) | 1982-01-01 |
| ES8201583A1 (es) | 1982-01-01 |
| ES8201582A1 (es) | 1982-01-01 |
| IL60617A0 (en) | 1980-09-16 |
| FI802308A7 (fi) | 1981-01-01 |
| AU6044380A (en) | 1981-01-29 |
| ES500384A0 (es) | 1982-01-01 |
| GR69719B (es) | 1982-07-09 |
| EP0024309A2 (de) | 1981-03-04 |
| CA1137087A (en) | 1982-12-07 |
| ES500383A0 (es) | 1982-01-01 |
| DK316480A (da) | 1981-01-24 |
| EP0024309A3 (de) | 1981-07-22 |
| US4307094A (en) | 1981-12-22 |
| MC1334A1 (fr) | 1981-04-21 |
| PT71587A (en) | 1980-08-01 |
| ES493579A0 (es) | 1981-06-16 |
| ES8201580A1 (es) | 1982-01-01 |
| ES500385A0 (es) | 1982-01-01 |
| PT71587B (en) | 1981-12-17 |
| ES8201581A1 (es) | 1982-01-01 |
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