ES476232A1 - Procedimiento para la obtencion de derivados del fosfonilu- reidobenceno. - Google Patents
Procedimiento para la obtencion de derivados del fosfonilu- reidobenceno.Info
- Publication number
- ES476232A1 ES476232A1 ES476232A ES476232A ES476232A1 ES 476232 A1 ES476232 A1 ES 476232A1 ES 476232 A ES476232 A ES 476232A ES 476232 A ES476232 A ES 476232A ES 476232 A1 ES476232 A1 ES 476232A1
- Authority
- ES
- Spain
- Prior art keywords
- represent
- group
- compounds
- different
- phosphonyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 239000003814 drug Substances 0.000 title 1
- 229940079593 drug Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 4
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 125000000383 tetramethylene group Chemical group [H]C([H])([*:1])C([H])([H])C([H])([H])C([H])([H])[*:2] 0.000 abstract 2
- 125000003258 trimethylene group Chemical group [H]C([H])([*:2])C([H])([H])C([H])([H])[*:1] 0.000 abstract 2
- 241001466804 Carnivora Species 0.000 abstract 1
- 241001465754 Metazoa Species 0.000 abstract 1
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- -1 dimethylene group Chemical group 0.000 abstract 1
- 244000000013 helminth Species 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 125000004430 oxygen atom Chemical group O* 0.000 abstract 1
- 230000000590 parasiticidal effect Effects 0.000 abstract 1
- 239000002297 parasiticide Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000001984 thiazolidinyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6536—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and sulfur atoms with or without oxygen atoms, as the only ring hetero atoms
- C07F9/6539—Five-membered rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/06—Phosphorus compounds without P—C bonds
- C07F9/22—Amides of acids of phosphorus
- C07F9/24—Esteramides
- C07F9/2454—Esteramides the amide moiety containing a substituent or a structure which is considered as characteristic
- C07F9/2479—Compounds containing the structure P(=X)n-N-acyl, P(=X)n-N-heteroatom, P(=X)n-N-CN (X = O, S, Se; n = 0, 1)
- C07F9/2487—Compounds containing the structure P(=X)n-N-acyl, P(=X)n-N-heteroatom, P(=X)n-N-CN (X = O, S, Se; n = 0, 1) containing the structure P(=X)n-N-C(=X) (X = O, S, Se; n = 0, 1)
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/572—Five-membered rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6564—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms
- C07F9/6571—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and oxygen atoms as the only ring hetero atoms
- C07F9/657154—Cyclic esteramides of oxyacids of phosphorus
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Veterinary Medicine (AREA)
- Crystallography & Structural Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
Procedimiento para la obtención de derivados del fosfonilureidobenceno de fórmula general **formula** donde R1 y R2 pueden ser iguales o diferentes y significan alquilo, o R1 y R2 juntos están por un grupo dimetileno, un grupo trimetileno o un grupo tetrametileno, X e Y pueden ser iguales o diferentes, y significan un átomo de oxígeno o un átomo de azufre, R3 y R4 pueden ser iguales o diferentes y significan alquilo, o R3 y R4 juntos significan un grupo trimetileno o un grupo tetrametileno o R3 y R4 junto con el átomo de czarbono y de nitrógeno encerrado por ellos forma un sistema de anillo tiazolidina, asi como sus sales de adición de ácido fisiológicamente compatibles.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19772758005 DE2758005A1 (de) | 1977-12-24 | 1977-12-24 | Phosphonylureidobenzol-derivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES476232A1 true ES476232A1 (es) | 1979-04-16 |
Family
ID=6027282
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES476232A Expired ES476232A1 (es) | 1977-12-24 | 1978-12-21 | Procedimiento para la obtencion de derivados del fosfonilu- reidobenceno. |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US4247546A (es) |
| EP (1) | EP0002723B1 (es) |
| JP (1) | JPS5495549A (es) |
| AU (1) | AU520492B2 (es) |
| DE (2) | DE2758005A1 (es) |
| DK (1) | DK578878A (es) |
| ES (1) | ES476232A1 (es) |
| NZ (1) | NZ189265A (es) |
| TR (1) | TR20362A (es) |
| ZA (1) | ZA787230B (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5451437A (en) * | 1993-06-21 | 1995-09-19 | Minnesota Mining And Manufacturing Company | Method and article for protecting a container that holds a fluid |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2029299C3 (de) * | 1970-06-13 | 1980-08-21 | Bayer Ag, 5090 Leverkusen | Neue Aminophenylamidine, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel |
| DE2029298C3 (de) * | 1970-06-13 | 1980-04-17 | Bayer Ag, 5090 Leverkusen | Aminophenylamidine, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel |
| BE788743A (fr) | 1971-09-14 | 1973-03-13 | Bayer Ag | Nouveaux 2-(aminophenylimino)-3- aza-1-thia-cycloalcanes, leur procede de preparation et leur application comme |
| US4086336A (en) * | 1972-05-26 | 1978-04-25 | Rohm And Haas Company | Phosphonothioureide anthelmintics |
| US4076809A (en) * | 1975-10-28 | 1978-02-28 | Rohm And Haas Company | Phosphonoureide and phosphonothioureide anthelmintics |
| US4087521A (en) * | 1976-03-01 | 1978-05-02 | Rohm And Haas Company | Arthropodicidal and nematocidal phosphoramidates |
-
1977
- 1977-12-24 DE DE19772758005 patent/DE2758005A1/de not_active Withdrawn
-
1978
- 1978-12-06 US US05/967,035 patent/US4247546A/en not_active Expired - Lifetime
- 1978-12-13 DE DE7878101656T patent/DE2860364D1/de not_active Expired
- 1978-12-13 EP EP78101656A patent/EP0002723B1/de not_active Expired
- 1978-12-20 AU AU42750/78A patent/AU520492B2/en not_active Expired
- 1978-12-21 ZA ZA00787230A patent/ZA787230B/xx unknown
- 1978-12-21 ES ES476232A patent/ES476232A1/es not_active Expired
- 1978-12-21 TR TR20362A patent/TR20362A/xx unknown
- 1978-12-21 NZ NZ189265A patent/NZ189265A/en unknown
- 1978-12-22 DK DK578878A patent/DK578878A/da not_active Application Discontinuation
- 1978-12-22 JP JP15773178A patent/JPS5495549A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| NZ189265A (en) | 1984-04-27 |
| US4247546A (en) | 1981-01-27 |
| DK578878A (da) | 1979-06-25 |
| DE2860364D1 (en) | 1981-03-12 |
| AU4275078A (en) | 1979-06-28 |
| ZA787230B (en) | 1979-12-27 |
| EP0002723B1 (de) | 1981-01-21 |
| DE2758005A1 (de) | 1979-06-28 |
| TR20362A (tr) | 1981-04-21 |
| JPS5495549A (en) | 1979-07-28 |
| AU520492B2 (en) | 1982-02-04 |
| EP0002723A1 (de) | 1979-07-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19990405 |