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EE200300567A - Meetod amorfse naatrium-tsilastatiini valmistamiseks - Google Patents

Meetod amorfse naatrium-tsilastatiini valmistamiseks

Info

Publication number
EE200300567A
EE200300567A EEP200300567A EEP200300567A EE200300567A EE 200300567 A EE200300567 A EE 200300567A EE P200300567 A EEP200300567 A EE P200300567A EE P200300567 A EEP200300567 A EE P200300567A EE 200300567 A EE200300567 A EE 200300567A
Authority
EE
Estonia
Prior art keywords
preparation
cilastatin sodium
amorphous
amorphous cilastatin
sodium
Prior art date
Application number
EEP200300567A
Other languages
English (en)
Inventor
Kumar Yatendra
Dutt Tyagi Om
Rohtagi Amit
Original Assignee
Ranbaxy Laboratories Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ranbaxy Laboratories Limited filed Critical Ranbaxy Laboratories Limited
Publication of EE200300567A publication Critical patent/EE200300567A/et

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C31/00Saturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C31/02Monohydroxylic acyclic alcohols
    • C07C31/04Methanol
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/26Separation; Purification; Stabilisation; Use of additives
    • C07C319/28Separation; Purification
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12NMICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
    • C12N9/00Enzymes; Proenzymes; Compositions thereof; Processes for preparing, activating, inhibiting, separating or purifying enzymes
    • C12N9/14Hydrolases (3)
    • C12N9/48Hydrolases (3) acting on peptide bonds (3.4)

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Zoology (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Microbiology (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Biochemistry (AREA)
  • General Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Steroid Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Cephalosporin Compounds (AREA)
EEP200300567A 2001-05-18 2002-05-17 Meetod amorfse naatrium-tsilastatiini valmistamiseks EE200300567A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN593DE2001 2001-05-18
PCT/IB2002/001696 WO2002094742A1 (en) 2001-05-18 2002-05-17 Process for the preparation of amorphous cilastatin sodium

Publications (1)

Publication Number Publication Date
EE200300567A true EE200300567A (et) 2004-04-15

Family

ID=11097060

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200300567A EE200300567A (et) 2001-05-18 2002-05-17 Meetod amorfse naatrium-tsilastatiini valmistamiseks

Country Status (24)

Country Link
US (1) US20040152780A1 (et)
EP (1) EP1395530A4 (et)
JP (1) JP2004526805A (et)
KR (1) KR20040044409A (et)
CN (1) CN1522235A (et)
AP (2) AP1511A (et)
AR (1) AR036017A1 (et)
BG (1) BG108447A (et)
BR (1) BR0209843A (et)
CA (1) CA2447788A1 (et)
CZ (1) CZ20033352A3 (et)
EA (1) EA005947B1 (et)
EE (1) EE200300567A (et)
HR (1) HRP20031052A2 (et)
HU (1) HUP0400825A2 (et)
IL (1) IL158945A0 (et)
MX (1) MXPA03010547A (et)
NO (1) NO20035138D0 (et)
NZ (1) NZ529625A (et)
OA (1) OA12607A (et)
PL (1) PL367937A1 (et)
SK (1) SK15082003A3 (et)
WO (1) WO2002094742A1 (et)
ZA (1) ZA200309287B (et)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2431275T3 (es) 2005-11-09 2013-11-25 Orchid Chemicals&Pharmaceuticals Limited Un procedimiento mejorado para la preparación de cilastatina ácida
WO2011080648A1 (en) * 2010-01-01 2011-07-07 Orchid Chemicals And Pharmaceuticals Limited An improved process for the preparation of cilastatin sodium
CN102675175B (zh) * 2011-03-08 2014-02-19 深圳市海滨制药有限公司 一种西司他丁的分离纯化方法
WO2018091679A1 (en) * 2016-11-18 2018-05-24 Universitat De Barcelona Combined cd6 and imipenem therapy for treatment of infectious diseases and related inflammatory processes

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5147868A (en) * 1978-07-24 1992-09-15 Merck & Co., Inc. Thienamycin renal peptidase inhibitors
US4292436A (en) * 1980-06-25 1981-09-29 Merck & Co., Inc. Process for the preparation of N-protected N-formimidoyl 2-aminoethanethiol
US5202467A (en) * 1990-02-08 1993-04-13 Sumitomo Chemical Company, Limited Process for preparing haloketo acid derivatives
US5166417A (en) * 1990-09-04 1992-11-24 Lonza Ltd. Process for resolution of racemates of 2,2-dimethylcyclopropanecarboxylic acid
CA2056840A1 (en) * 1990-12-17 1992-06-18 Thomas Meul Process for the production of dimethylcyclopropanecarboxylic acid
EP0524604B1 (de) * 1991-07-26 1998-10-14 Lonza A.G. Gentechnologisches Verfahren zur Herstellung von S-(+)-2,2-Dimethylcyclopropancarboxamid mittels Mikroorganismen
US5245069A (en) * 1992-10-27 1993-09-14 Merck & Co., Inc. Process for the preparation of bis(aryl)-phosphorohalidates
IN191798B (et) * 2000-11-03 2004-01-03 Ranbaxy Lab Ltd

Also Published As

Publication number Publication date
WO2002094742A1 (en) 2002-11-28
BR0209843A (pt) 2004-08-24
IL158945A0 (en) 2004-05-12
EA200301225A1 (ru) 2004-06-24
HUP0400825A2 (hu) 2004-08-30
AP2003002912A0 (en) 2002-05-17
NZ529625A (en) 2006-02-24
BG108447A (en) 2005-03-31
EA005947B1 (ru) 2005-08-25
OA12607A (en) 2006-06-08
CN1522235A (zh) 2004-08-18
SK15082003A3 (sk) 2004-06-08
ZA200309287B (en) 2004-07-22
AP2003002913A0 (en) 2003-12-31
CA2447788A1 (en) 2002-11-28
KR20040044409A (ko) 2004-05-28
HRP20031052A2 (en) 2004-06-30
CZ20033352A3 (en) 2004-06-16
AR036017A1 (es) 2004-08-04
AP1511A (en) 2005-12-20
JP2004526805A (ja) 2004-09-02
EP1395530A1 (en) 2004-03-10
MXPA03010547A (es) 2004-05-27
EP1395530A4 (en) 2006-01-18
US20040152780A1 (en) 2004-08-05
PL367937A1 (en) 2005-03-07
NO20035138D0 (no) 2003-11-18

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