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EE05350B1 - Antiproliferatiivsete vahenditena kasutatavad bensoimidasooli derivaadid - Google Patents

Antiproliferatiivsete vahenditena kasutatavad bensoimidasooli derivaadid

Info

Publication number
EE05350B1
EE05350B1 EEP200200276A EEP200200276A EE05350B1 EE 05350 B1 EE05350 B1 EE 05350B1 EE P200200276 A EEP200200276 A EE P200200276A EE P200200276 A EEP200200276 A EE P200200276A EE 05350 B1 EE05350 B1 EE 05350B1
Authority
EE
Estonia
Prior art keywords
antiproliferative agents
derivatives used
benzoimidazole derivatives
benzoimidazole
antiproliferative
Prior art date
Application number
EEP200200276A
Other languages
English (en)
Inventor
Ernest Barth Wayne
Joseph Luzzio Michael
Peter Lyssikatos Joseph
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of EE200200276A publication Critical patent/EE200200276A/et
Publication of EE05350B1 publication Critical patent/EE05350B1/et

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P11/06Antiasthmatics
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    • A61P13/08Drugs for disorders of the urinary system of the prostate
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    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
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    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
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    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
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    • A61P17/04Antipruritics
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    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A61P9/00Drugs for disorders of the cardiovascular system
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10Spiro-condensed systems

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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Oncology (AREA)
  • Transplantation (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Ophthalmology & Optometry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
EEP200200276A 1999-11-30 2000-11-10 Antiproliferatiivsete vahenditena kasutatavad bensoimidasooli derivaadid EE05350B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US16821799P 1999-11-30 1999-11-30
PCT/IB2000/001636 WO2001040217A1 (en) 1999-11-30 2000-11-10 Novel benzoimidazole derivatives useful as antiproliferative agents

Publications (2)

Publication Number Publication Date
EE200200276A EE200200276A (et) 2003-06-16
EE05350B1 true EE05350B1 (et) 2010-10-15

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200200276A EE05350B1 (et) 1999-11-30 2000-11-10 Antiproliferatiivsete vahenditena kasutatavad bensoimidasooli derivaadid

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US (1) US7019147B1 (et)
EP (1) EP1235825B1 (et)
JP (2) JP4522635B2 (et)
KR (1) KR100479401B1 (et)
CN (2) CN1402721A (et)
AP (1) AP1895A (et)
AR (1) AR026633A1 (et)
AT (1) ATE316528T1 (et)
AU (1) AU782077B2 (et)
BG (1) BG65862B1 (et)
BR (1) BR0015911A (et)
CA (1) CA2392973C (et)
CO (1) CO5251455A1 (et)
CR (1) CR6643A (et)
CU (1) CU23132A3 (et)
CZ (1) CZ300789B6 (et)
DE (1) DE60025747T2 (et)
DK (1) DK1235825T3 (et)
DZ (1) DZ3327A1 (et)
EA (1) EA005407B1 (et)
EE (1) EE05350B1 (et)
EG (1) EG24433A (et)
ES (1) ES2256052T3 (et)
GE (1) GEP20033141B (et)
GT (1) GT200000198A (et)
HR (1) HRP20020475B1 (et)
HU (1) HU230829B1 (et)
IL (2) IL149841A0 (et)
IS (1) IS2209B (et)
MA (1) MA26847A1 (et)
MX (1) MXPA02005343A (et)
MY (1) MY128765A (et)
NO (1) NO324043B1 (et)
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PA (1) PA8507601A1 (et)
PE (1) PE20010899A1 (et)
PL (1) PL201784B1 (et)
RS (1) RS50800B (et)
SI (1) SI1235825T1 (et)
SK (1) SK286773B6 (et)
SV (1) SV2002000232A (et)
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UA (1) UA75055C2 (et)
WO (1) WO2001040217A1 (et)
ZA (1) ZA200204244B (et)

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