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DK164669C - 2- eller 3-arylsubstituerede imidazooe1,2-aaapyridiner samt fremgangsmaader til fremstilling deraf - Google Patents

2- eller 3-arylsubstituerede imidazooe1,2-aaapyridiner samt fremgangsmaader til fremstilling deraf

Info

Publication number
DK164669C
DK164669C DK495287A DK495287A DK164669C DK 164669 C DK164669 C DK 164669C DK 495287 A DK495287 A DK 495287A DK 495287 A DK495287 A DK 495287A DK 164669 C DK164669 C DK 164669C
Authority
DK
Denmark
Prior art keywords
imidazooe1
aaapyridines
aryl
procedures
substituted
Prior art date
Application number
DK495287A
Other languages
English (en)
Other versions
DK495287A (da
DK164669B (da
DK495287D0 (da
Inventor
Jeffery B Press
Original Assignee
Ortho Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/909,648 external-priority patent/US4727145A/en
Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp
Publication of DK495287D0 publication Critical patent/DK495287D0/da
Publication of DK495287A publication Critical patent/DK495287A/da
Publication of DK164669B publication Critical patent/DK164669B/da
Application granted granted Critical
Publication of DK164669C publication Critical patent/DK164669C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK495287A 1986-09-22 1987-09-21 2- eller 3-arylsubstituerede imidazooe1,2-aaapyridiner samt fremgangsmaader til fremstilling deraf DK164669C (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US06/909,648 US4727145A (en) 1986-09-22 1986-09-22 2- Or 3- aryl substituted imidazo [1,2-a]pyridines
US90964886 1986-09-22
US07/090,111 US4791117A (en) 1986-09-22 1987-08-31 2- or 3-aryl substituted imidazo[1,2-a]pyridines and their use as calcium channel blockers
US9011187 1987-08-31

Publications (4)

Publication Number Publication Date
DK495287D0 DK495287D0 (da) 1987-09-21
DK495287A DK495287A (da) 1988-03-23
DK164669B DK164669B (da) 1992-07-27
DK164669C true DK164669C (da) 1992-12-21

Family

ID=26781926

Family Applications (1)

Application Number Title Priority Date Filing Date
DK495287A DK164669C (da) 1986-09-22 1987-09-21 2- eller 3-arylsubstituerede imidazooe1,2-aaapyridiner samt fremgangsmaader til fremstilling deraf

Country Status (5)

Country Link
US (1) US4791117A (da)
EP (1) EP0261912A3 (da)
AU (1) AU597108B2 (da)
DK (1) DK164669C (da)
IE (1) IE872541L (da)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2647451B1 (fr) * 1989-05-26 1994-08-05 Sanofi Sa Derives d'imidazo(1,2-a)pyridine, procede de preparation, compositions pharmaceutiques les contenant
DE4405378A1 (de) * 1994-02-19 1995-08-24 Merck Patent Gmbh Adhäsionsrezeptor-Antagonisten
US6541479B1 (en) * 1997-12-02 2003-04-01 Massachusetts College Of Pharmacy Calcium channel blockers
CA2311483A1 (en) 2000-06-12 2001-12-12 Gregory N Beatch IMIDAZO [1,2-A] PYRIDINIC ETHERS AND USES THEREOF
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
DE10117183A1 (de) * 2001-04-05 2002-10-10 Gruenenthal Gmbh Verwendung von substituierten Imidazo[1,2-a]-pyridinverbindungen als Arzneimittel
MY140561A (en) 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
DE10247271A1 (de) * 2002-10-10 2004-08-26 Grünenthal GmbH Substituierte C-Imidazo[1,2-a]pyridin-3-yle
HRP20050399B1 (hr) 2003-03-10 2013-09-30 Takeda Gmbh Novi postupci za dobivanje roflumilasta
US8663694B2 (en) 2005-03-16 2014-03-04 Takeda Gmbh Taste masked dosage form containing roflumilast
TW200803903A (en) * 2006-04-28 2008-01-16 Nihon Mediphysics Co Ltd Novel compound having affinity to amyloid
US8303935B2 (en) 2006-05-19 2012-11-06 Nihon Medi-Physics Co., Ltd. Alkoxy substituted imidazo[1,2-a]pyridines having affinity for amyloid
KR20090025282A (ko) * 2006-06-21 2009-03-10 니혼 메디피직스 가부시키가이샤 신규 아밀로이드 친화성 화합물
CA2669522A1 (en) * 2006-11-17 2008-05-22 Nihon Medi-Physics Co., Ltd. Novel compounds with affinity for amyloid
CA2670436A1 (en) 2006-11-30 2008-06-05 Nihon Medi-Physics Co., Ltd. Novel compound having affinity for amyloid
ES2421886T3 (es) 2007-02-13 2013-09-06 Nihon Mediphysics Co Ltd Método para producción de un agente de representación de imágenes de diagnóstico por radiación
CN101903381A (zh) * 2007-10-24 2010-12-01 日本医事物理股份有限公司 对淀粉样蛋白具有亲和性的新化合物
JP5313158B2 (ja) * 2007-10-26 2013-10-09 日本メジフィジックス株式会社 新規アミロイド親和性化合物
AU2008319985A1 (en) * 2007-10-30 2009-05-07 Nihon Medi-Physics Co., Ltd. Use of novel compound having affinity for amyloid, and process for production of the same
CN101909659A (zh) * 2007-10-30 2010-12-08 日本医事物理股份有限公司 对淀粉样蛋白具有亲和性的新化合物的应用及制备方法
EP2832234A1 (en) * 2013-07-30 2015-02-04 IMAX Discovery GmbH Imidazo[1,2-a]pyridine-ylmethyl-derivatives and their use as flavoring agents

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2937179A (en) * 1958-04-09 1960-05-17 Seymour L Shapiro Process for phenylimidazolino [1, 2-alpha]piperidines
GB1442707A (en) * 1973-07-07 1976-07-14 Yoshitomi Pharmaceutical Substituted phenylalkanoic acids and their derivatives and pharma ceutical compositions thereof
GB1473819A (en) * 1976-01-28 1977-05-18 Gallardo Antonio Sa Derivatives of imidazo 1,2-a pyridine
EP0068378B1 (en) * 1981-06-26 1986-03-05 Schering Corporation Novel imidazo(1,2-a)pyridines and pyrazines, processes for their preparation and pharmaceutical compositions containing them
GB8305245D0 (en) * 1983-02-25 1983-03-30 Fujisawa Pharmaceutical Co Imidazo-heterocyclic compounds
AU7928787A (en) * 1986-10-07 1988-04-14 Yamanouchi Pharmaceutical Co., Ltd. Imidazopyridine derivatives
US4831041A (en) * 1986-11-26 1989-05-16 Fujisawa Pharmaceutical Co., Ltd. Imidazopyridine compounds and processes for preparation thereof
DE3865073D1 (de) * 1987-03-27 1991-10-31 Synthelabo Imidazopyridinderivate, ihre herstellung und therapeutische verwendung.

Also Published As

Publication number Publication date
EP0261912A2 (en) 1988-03-30
DK495287A (da) 1988-03-23
AU7849387A (en) 1988-03-24
IE872541L (en) 1988-03-22
DK164669B (da) 1992-07-27
AU597108B2 (en) 1990-05-24
US4791117A (en) 1988-12-13
EP0261912A3 (en) 1989-09-20
DK495287D0 (da) 1987-09-21

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