DE60308388D1 - 5-androsten-3-olsteroidzwischenprodukte und verfahren zu deren herstellung - Google Patents

5-androsten-3-olsteroidzwischenprodukte und verfahren zu deren herstellung

Info

Publication number: DE60308388D1
Authority: DE; Germany
Prior art keywords: androsten; olsteroid; production; intermediate products; 3beta
Prior art date: 2002-08-16
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired - Fee Related

Application number

DE60308388T

Other languages

English (en)

Other versions

DE60308388T2 (de

Inventor

J White

G Wuts

Doris Beck

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Pharmacia and Upjohn Co LLC

Original Assignee

Pharmacia and Upjohn Co LLC

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-08-16

Filing date

2003-03-21

Publication date

2006-10-26

2003-03-21 Application filed by Pharmacia and Upjohn Co LLC filed Critical Pharmacia and Upjohn Co LLC

2006-10-26 Application granted granted Critical

2006-10-26 Publication of DE60308388D1 publication Critical patent/DE60308388D1/de

2007-09-20 Publication of DE60308388T2 publication Critical patent/DE60308388T2/de

2023-03-22 Anticipated expiration legal-status Critical

Status Expired - Fee Related legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0003—Androstane derivatives
- C07J1/0011—Androstane derivatives substituted in position 17 by a keto group
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J21/001—Lactones
- C07J21/003—Lactones at position 17

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Steroid Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DE60308388T 2002-08-16 2003-03-21 5-Androsten-3beta-ol-Steroide und Verfahren für ihre Herstellung Expired - Fee Related DE60308388T2 (de)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
US40399002P	2002-08-16	2002-08-16
US403990P		2002-08-16
US41529302P	2002-10-01	2002-10-01
US415293P		2002-10-01
PCT/US2003/007791 WO2004016640A2 (en)	2002-08-16	2003-03-21	5 ANDROSTEN-3β-OL STEROID INTERMEDIATES AND PROCESSES FOR THEIR PREPARATION

Publications (2)

Publication Number	Publication Date
DE60308388D1 true DE60308388D1 (de)	2006-10-26
DE60308388T2 DE60308388T2 (de)	2007-09-20

Family

ID=31891414

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DE60308388T Expired - Fee Related DE60308388T2 (de)	2002-08-16	2003-03-21	5-Androsten-3beta-ol-Steroide und Verfahren für ihre Herstellung

Country Status (12)

Country	Link
US (2)	US20040034215A1 (de)
EP (1)	EP1534732B1 (de)
JP (1)	JP2006507369A (de)
AT (1)	ATE339437T1 (de)
AU (1)	AU2003285485A1 (de)
BR (1)	BR0313523A (de)
CA (1)	CA2495412A1 (de)
DE (1)	DE60308388T2 (de)
ES (1)	ES2271636T3 (de)
MX (1)	MXPA05001857A (de)
TW (1)	TW200406419A (de)
WO (1)	WO2004016640A2 (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ITMI20042338A1 (it) *	2004-12-06	2005-03-06	Ind Chimica Srl	Processo per la preparazione di drospirenone
US8084446B2 (en)	2005-04-26	2011-12-27	Eric Marchewitz	Use of DHEA derivatives for enhancing physical performance
ATE403668T1 (de)	2005-07-21	2008-08-15	Bayer Schering Pharma Ag	Verfahren zur herstellung von 3-oxo-pregn-4-en-21,17-carbolactonen durch die metallfreie oxidation von 17-(3-hydroxypropyl)-3,17- dihydroxyandrostanen
SI1910403T1 (sl) *	2005-07-21	2016-08-31	Bayer Pharma AG	Postopek za pripravo 3-okso-pregn-4-en-21,17-karbolaktonov z oksidacijo 17-(3-hidroksipropil)-3,17-dihidroksiandrostanov brez uporabe kovine
US7319154B2 (en) *	2005-07-21	2008-01-15	Bayer Schering Pharma Ag	Process for the production of 3-oxo-pregn-4-ene-21, 17-carbolactones by the metal free oxidation of 17-(3-hydroxypropyl)-3, 17-dihydroxyandrostanes
CN110331182A (zh) *	2019-08-06	2019-10-15	江苏远大仙乐药业有限公司	一种甾体中间体的生物转化制备方法
CN111057734A (zh) *	2019-12-24	2020-04-24	天津科技大学	一种甲基睾丸素高效转化生产11α-羟基-甲基睾丸素的方法
CN110885869A (zh) *	2019-12-24	2020-03-17	天津科技大学	一种利用微生物转化生产7α-羟基-脱氢表雄酮的方法

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3294646A (en) *	1963-10-23	1966-12-27	American Home Prod	Microbiological hydroxylation of norsteroids using aspergillus ochraceus
DE2349022A1 (de) *	1973-09-26	1975-04-10	Schering Ag	Neue d-homo-steroide
ES432106A1 (es) *	1973-11-30	1976-11-01	Schering Ag	Procedimiento para la preparacion de d-homo-20-cetopregna- nos.
US4031074A (en) *	1974-09-02	1977-06-21	Akzona Incorporated	Process for the preparation of 11β-hydroxy-18-alkyl-estrane compounds
IL48628A0 (en) *	1974-12-23	1976-02-29	Schering Ag	D-homo-20-keto-pregnanes and process for their manufactur
US4054563A (en) *	1975-04-25	1977-10-18	Ciba-Geigy Corporation	Process for the manufacture of spiro compounds of the steroid series
CH633562A5 (de) *	1976-12-10	1982-12-15	Schering Ag	Verfahren zur herstellung neuer kortikoide.
US4336332A (en) *	1979-02-20	1982-06-22	Hoffmann-La Roche, Inc.	Process for the manufacture of hydroxylated steroids
DE3042136A1 (de) *	1980-11-03	1982-06-09	Schering Ag, 1000 Berlin Und 4619 Bergkamen	Verfahren zur herstellung von 3 (beta), 7 (beta) -dihydroxy- (delta) (pfeil hoch)5(pfeil hoch) -steroiden
US4559332A (en) *	1983-04-13	1985-12-17	Ciba Geigy Corporation	20-Spiroxanes and analogues having an open ring E, processes for their manufacture, and pharmaceutical preparations thereof
AU7978794A (en) *	1993-10-13	1995-05-04	Neurocrine Biosciences, Inc.	3,17-dihydroxy-3,7,16 and/or 17-methyl-androst-5-ene compounds, derivatives thereof, and their use
CN100384866C (zh) *	1995-12-11	2008-04-30	G·D·瑟尔公司	制备7α-羧基9,11-环氧甾族化合物的方法和其中使用的中间体以及烯双键环氧化作用的一般方法
PT900283E (pt) *	1995-12-12	2002-09-30	Akzo Nobel Nv	11alfa-hidroxilacao microbiana de esteroides
FR2771105A1 (fr)	1997-11-20	1999-05-21	Vitasterol	Utilisation du fusarium monoliforme pour la preparation des derives 7alpha-hydroxyles de la dehydroepiandrosterone et de la pregnenolone

2003
- 2003-03-21 MX MXPA05001857A patent/MXPA05001857A/es unknown
- 2003-03-21 US US10/392,955 patent/US20040034215A1/en not_active Abandoned
- 2003-03-21 WO PCT/US2003/007791 patent/WO2004016640A2/en not_active Ceased
- 2003-03-21 DE DE60308388T patent/DE60308388T2/de not_active Expired - Fee Related
- 2003-03-21 JP JP2005502036A patent/JP2006507369A/ja not_active Abandoned
- 2003-03-21 AT AT03756776T patent/ATE339437T1/de not_active IP Right Cessation
- 2003-03-21 AU AU2003285485A patent/AU2003285485A1/en not_active Abandoned
- 2003-03-21 CA CA002495412A patent/CA2495412A1/en not_active Abandoned
- 2003-03-21 EP EP03756776A patent/EP1534732B1/de not_active Expired - Lifetime
- 2003-03-21 BR BR0313523-3A patent/BR0313523A/pt not_active IP Right Cessation
- 2003-03-21 ES ES03756776T patent/ES2271636T3/es not_active Expired - Lifetime
- 2003-03-21 TW TW092106331A patent/TW200406419A/zh unknown
2004
- 2004-06-01 US US10/858,177 patent/US7002028B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
WO2004016640A2 (en)	2004-02-26
JP2006507369A (ja)	2006-03-02
AU2003285485A1 (en)	2004-03-03
ATE339437T1 (de)	2006-10-15
DE60308388T2 (de)	2007-09-20
US7002028B2 (en)	2006-02-21
CA2495412A1 (en)	2004-02-26
US20040034215A1 (en)	2004-02-19
US20040220158A1 (en)	2004-11-04
EP1534732A2 (de)	2005-06-01
EP1534732B1 (de)	2006-09-13
ES2271636T3 (es)	2007-04-16
WO2004016640A3 (en)	2004-07-08
BR0313523A (pt)	2005-06-28
TW200406419A (en)	2004-05-01
MXPA05001857A (es)	2005-06-03

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Legal Events

Date	Code	Title	Description
2007-10-25	8364	No opposition during term of opposition
2009-01-22	8339	Ceased/non-payment of the annual fee