CO6270303A2 - Producto de dispersion solida que contiene un compuesto a base de n-aril urea - Google Patents
Producto de dispersion solida que contiene un compuesto a base de n-aril ureaInfo
- Publication number
- CO6270303A2 CO6270303A2 CO10049270A CO10049270A CO6270303A2 CO 6270303 A2 CO6270303 A2 CO 6270303A2 CO 10049270 A CO10049270 A CO 10049270A CO 10049270 A CO10049270 A CO 10049270A CO 6270303 A2 CO6270303 A2 CO 6270303A2
- Authority
- CO
- Colombia
- Prior art keywords
- solid dispersion
- urea
- aril
- based compound
- product containing
- Prior art date
Links
- 239000007962 solid dispersion Substances 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 title 1
- 239000003795 chemical substances by application Substances 0.000 abstract 3
- 239000013543 active substance Substances 0.000 abstract 2
- 239000007788 liquid Substances 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 239000002904 solvent Substances 0.000 abstract 2
- 239000004202 carbamide Substances 0.000 abstract 1
- 239000011159 matrix material Substances 0.000 abstract 1
- 239000004094 surface-active agent Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
Landscapes
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Un producto que comprende al menos un agente farmacéuticamente activo a base de N-aril urea o un agente de estructura: relacionada que es obtenido mediante a) la preparacion de una mezcla liquida que contiene el al menos un agente activo, el al menos un agente formador de matriz aceptable para uso farmacéutico, el al menos un tensioactivo aceptable para uso farmacéutico y el al menos un solvente, y b) la eliminacion del o de los solventes de la mezcla liquida para obtener el producto de dispersion solida.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US99961307P | 2007-10-19 | 2007-10-19 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CO6270303A2 true CO6270303A2 (es) | 2011-04-20 |
Family
ID=40089072
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CO10049270A CO6270303A2 (es) | 2007-10-19 | 2010-04-27 | Producto de dispersion solida que contiene un compuesto a base de n-aril urea |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US20090143423A1 (es) |
| EP (1) | EP2197426A2 (es) |
| JP (1) | JP2011500647A (es) |
| KR (1) | KR20100090689A (es) |
| CN (1) | CN101827585A (es) |
| AR (1) | AR068916A1 (es) |
| AU (1) | AU2008313620A1 (es) |
| BR (1) | BRPI0818339A2 (es) |
| CA (1) | CA2699335A1 (es) |
| CL (1) | CL2008003092A1 (es) |
| CO (1) | CO6270303A2 (es) |
| CR (1) | CR11441A (es) |
| DO (1) | DOP2010000114A (es) |
| EC (1) | ECSP10010184A (es) |
| GT (1) | GT201000095A (es) |
| MX (1) | MX2010004292A (es) |
| PE (1) | PE20091041A1 (es) |
| RU (1) | RU2010119924A (es) |
| TW (1) | TW200922549A (es) |
| UA (1) | UA100866C2 (es) |
| UY (1) | UY31406A1 (es) |
| WO (1) | WO2009050289A2 (es) |
| ZA (1) | ZA201002130B (es) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2010045401A1 (en) * | 2008-10-17 | 2010-04-22 | Abbott Laboratories | Trpv1 antagonists |
| CA2737775A1 (en) * | 2008-10-17 | 2010-04-22 | Abbott Laboratories | Trpv1 antagonists |
| US20100210682A1 (en) * | 2009-02-19 | 2010-08-19 | Abbott Laboratories | Repeated Dosing of TRPV1 Antagonists |
| EP2477593A1 (de) * | 2009-09-18 | 2012-07-25 | Basf Se | Verfahren zur herstellung von zubereitungen von in wasser schwer löslichen substanzen |
| JP5903686B2 (ja) | 2010-12-23 | 2016-04-13 | アッヴィ・ドイチュラント・ゲー・エム・ベー・ハー・ウント・コー・カー・ゲー | 固体分散物を基にした固体徐放製剤 |
| CA2824066A1 (en) | 2011-01-10 | 2012-07-19 | Celgene Corporation | Oral dosage forms of cyclopropanecarboxylic acid {2-[(1s)-1-(3-ethoxy-4-methoxy-phenyl)-2-methanesulfonyl-ethyl]-3-oxo-2,3-dihydro-1h-isoindol-4-yl}-amide |
| CA2857339C (en) * | 2011-12-29 | 2015-11-17 | Abbvie Inc. | Solid compositions comprising an hcv inhibitor |
| US9034832B2 (en) | 2011-12-29 | 2015-05-19 | Abbvie Inc. | Solid compositions |
| TW201431570A (zh) | 2012-11-22 | 2014-08-16 | Ucb Pharma Gmbh | 用於經皮投服羅替戈汀(Rotigotine)之多天式貼片 |
| EP2950786B1 (en) | 2013-01-31 | 2019-11-27 | Gilead Pharmasset LLC | Combination formulation of two antiviral compounds |
| UA116237C2 (uk) | 2013-03-15 | 2018-02-26 | Бьорінгер Інгельхайм Інтернаціональ Гмбх | Тверда пероральна дозована композиція інгібітору нсv в аморфному стані |
| CN105358139B (zh) | 2013-07-03 | 2020-10-16 | Lts罗曼治疗方法有限公司 | 具有电子元件的经皮治疗系统 |
| NZ716840A (en) | 2013-08-27 | 2017-06-30 | Gilead Pharmasset Llc | Combination formulation of two antiviral compounds |
| JP6895755B2 (ja) | 2014-05-20 | 2021-06-30 | エルテーエス ローマン テラピー−ジステーメ アーゲー | 経皮送達システムにおける活性薬剤の放出を調節するための方法 |
| EP3145504B1 (en) | 2014-05-20 | 2023-07-26 | LTS Lohmann Therapie-Systeme AG | Transdermal delivery system including an interface mediator |
| EP3145502B1 (en) * | 2014-05-20 | 2022-07-06 | LTS Lohmann Therapie-Systeme AG | Transdermal delivery system containing rotigotine |
| US12133911B2 (en) | 2015-06-09 | 2024-11-05 | Capsugel Belgium Nv | Formulations to achieve rapid dissolution of drug from spray-dried dispersions in capsules |
| EP3393462B8 (en) * | 2015-12-22 | 2023-06-21 | Arizona Board of Regents on behalf of the University of Arizona | Compositions and methods for treatment, amelioration, and prevention of anesthesia-induced hypothermia |
| CA3117563A1 (en) * | 2018-10-30 | 2020-05-07 | Peloton Therapeutics, Inc. | Solid dispersions and pharmaceutical compositions comprising a substituted indane and methods for the preparation and use thereof |
| EP4019485B1 (en) | 2019-08-23 | 2024-08-07 | Mochida Pharmaceutical Co., Ltd. | Method for producing heterocyclidene acetamide derivatives |
| CA3150748A1 (en) | 2019-08-23 | 2021-03-04 | Mochida Pharmaceutical Co., Ltd. | Method for producing heterocyclidene acetamide derivative |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5362878A (en) * | 1991-03-21 | 1994-11-08 | Pfizer Inc. | Intermediates for making N-aryl and N-heteroarylamide and urea derivatives as inhibitors of acyl coenzyme A: cholesterol acyl transferase (ACAT) |
| CA2134359C (en) * | 1992-05-28 | 1997-07-01 | Ernest S. Hamanaka | New n-aryl and n-heteroarylurea derivatives as inhibitors of acyl coenzyme a: cholesterol acyl transferase (acat) |
| CN1273526A (zh) * | 1998-07-14 | 2000-11-15 | Em工业股份有限公司 | 微分散给药系统 |
| US7015233B2 (en) * | 2003-06-12 | 2006-03-21 | Abbott Laboratories | Fused compounds that inhibit vanilloid subtype 1 (VR1) receptor |
| AR049297A1 (es) * | 2004-06-08 | 2006-07-12 | Vertex Pharma | Una composicion farmaceutica y dispersiones solidas de vx-950 (inhibidor de la proteasa de hcv ns3/4a) y proceso de obtencion |
| CA2578442A1 (en) * | 2004-08-27 | 2006-03-09 | Bayer Pharmaceuticals Corporation | Pharmaceutical compositions comprising 4{4-[3-(4-chloro-3-trifluoromethylphenyl)-ureido]-phenoxy}-pyridine-2-carboxylic acid methyl amide for the treatment of cancer |
| JP2008536929A (ja) * | 2005-04-18 | 2008-09-11 | ルビコン・リサーチ・ピーヴィーティー・エルティーディー | 生体強化組成物 |
| KR100715355B1 (ko) * | 2005-09-30 | 2007-05-07 | 주식회사유한양행 | 프란루카스트를 함유하는 분무-건조 과립 및 그의 제조방법 |
| JP2009513642A (ja) * | 2005-10-25 | 2009-04-02 | アボット・ラボラトリーズ | 低水溶解度の薬剤を含む製剤およびそれの使用方法 |
| WO2007066189A2 (en) * | 2005-12-09 | 2007-06-14 | Pfizer Products Inc. | Salts, prodrugs and formulations of 1-[5-(4-amino-7-isopropyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-2-methoxy-phenyl]-3-(2,4-dichloro-phenyl)-urea |
| US7745448B2 (en) * | 2005-12-28 | 2010-06-29 | Abbott Laboratories Inc. | Crystalline N-(4-(4-aminothieno[2,3-d]pyrimidin-5-yl)phenyl)-N′-(2-fluoro-5-(trifluoromethyl)phenyl)urea ethanolate |
| CN103735515A (zh) * | 2006-02-09 | 2014-04-23 | 默沙东公司 | Cetp抑制剂的聚合物制剂 |
-
2008
- 2008-10-17 CN CN200880112161A patent/CN101827585A/zh active Pending
- 2008-10-17 JP JP2010529406A patent/JP2011500647A/ja active Pending
- 2008-10-17 UA UAA201006030A patent/UA100866C2/ru unknown
- 2008-10-17 BR BRPI0818339 patent/BRPI0818339A2/pt not_active IP Right Cessation
- 2008-10-17 KR KR1020107010874A patent/KR20100090689A/ko not_active Withdrawn
- 2008-10-17 TW TW097140229A patent/TW200922549A/zh unknown
- 2008-10-17 PE PE2008001785A patent/PE20091041A1/es not_active Application Discontinuation
- 2008-10-17 AU AU2008313620A patent/AU2008313620A1/en not_active Abandoned
- 2008-10-17 CL CL2008003092A patent/CL2008003092A1/es unknown
- 2008-10-17 CA CA2699335A patent/CA2699335A1/en not_active Abandoned
- 2008-10-17 EP EP08840773A patent/EP2197426A2/en not_active Withdrawn
- 2008-10-17 US US12/253,499 patent/US20090143423A1/en not_active Abandoned
- 2008-10-17 AR ARP080104542A patent/AR068916A1/es not_active Application Discontinuation
- 2008-10-17 WO PCT/EP2008/064073 patent/WO2009050289A2/en not_active Ceased
- 2008-10-17 UY UY31406A patent/UY31406A1/es not_active Application Discontinuation
- 2008-10-17 RU RU2010119924/15A patent/RU2010119924A/ru not_active Application Discontinuation
- 2008-10-17 MX MX2010004292A patent/MX2010004292A/es not_active Application Discontinuation
-
2010
- 2010-03-25 ZA ZA2010/02130A patent/ZA201002130B/en unknown
- 2010-04-15 GT GT201000095A patent/GT201000095A/es unknown
- 2010-04-16 DO DO2010000114A patent/DOP2010000114A/es unknown
- 2010-04-27 CO CO10049270A patent/CO6270303A2/es not_active Application Discontinuation
- 2010-05-17 EC EC2010010184A patent/ECSP10010184A/es unknown
- 2010-05-19 CR CR11441A patent/CR11441A/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| KR20100090689A (ko) | 2010-08-16 |
| AU2008313620A1 (en) | 2009-04-23 |
| AR068916A1 (es) | 2009-12-16 |
| TW200922549A (en) | 2009-06-01 |
| MX2010004292A (es) | 2010-08-02 |
| CR11441A (es) | 2010-10-25 |
| PE20091041A1 (es) | 2009-08-22 |
| CN101827585A (zh) | 2010-09-08 |
| WO2009050289A3 (en) | 2010-03-25 |
| ECSP10010184A (es) | 2010-06-29 |
| JP2011500647A (ja) | 2011-01-06 |
| UY31406A1 (es) | 2009-05-29 |
| DOP2010000114A (es) | 2010-05-15 |
| ZA201002130B (en) | 2011-11-30 |
| BRPI0818339A2 (pt) | 2015-04-22 |
| WO2009050289A2 (en) | 2009-04-23 |
| UA100866C2 (ru) | 2013-02-11 |
| GT201000095A (es) | 2012-04-03 |
| RU2010119924A (ru) | 2011-11-27 |
| CA2699335A1 (en) | 2009-04-23 |
| US20090143423A1 (en) | 2009-06-04 |
| CL2008003092A1 (es) | 2009-11-27 |
| EP2197426A2 (en) | 2010-06-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC | Application refused |