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CO5261582A1 - Composiciones de valdecoxib - Google Patents

Composiciones de valdecoxib

Info

Publication number
CO5261582A1
CO5261582A1 CO00094074A CO00094074A CO5261582A1 CO 5261582 A1 CO5261582 A1 CO 5261582A1 CO 00094074 A CO00094074 A CO 00094074A CO 00094074 A CO00094074 A CO 00094074A CO 5261582 A1 CO5261582 A1 CO 5261582A1
Authority
CO
Colombia
Prior art keywords
valdecoxib
concentration
administration
time
maximum concentration
Prior art date
Application number
CO00094074A
Other languages
English (en)
Inventor
Nadkami Sreekant
Karkali Tugrul
Mark J Konthy
Desai Subhash
Original Assignee
Pharmacia Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27389729&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO5261582(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacia Corp filed Critical Pharmacia Corp
Publication of CO5261582A1 publication Critical patent/CO5261582A1/es

Links

Classifications

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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Abstract

Una composición farmacéutica que comprende valdecoxib particulado en una cantidad de alrededor de 1mg a alrededor de 100 mg por dosis y uno o más excipientes farmacéuticamente aceptables, donde una única dosis, ante administración oral a un sujeto rápido, proporciona un curso de tiempo de concentración de suero de sangre de valdecoxib que tiene por lo menos uno de(a) un tiempo para alcanzar concentración umbral por efecto terapéutico no mayor de alrededor de 0,5 h después de administración;(b) un tiempo para alcanzar máxima concentración (Tmax) no mayor de alrededor de 3 h después de administración, yicida líquido y quimicamente compatible conc) una máxima concentración (Cmax) no menor de alrededor de 100 ng/ml.<EMI FILE="00094074_1" ID="1" IMF=JPEG >
CO00094074A 1999-12-08 2000-12-11 Composiciones de valdecoxib CO5261582A1 (es)

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WO2001041761A2 (en) 2001-06-14
AU777402B2 (en) 2004-10-14
IL144763A0 (en) 2002-06-30
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HUP0200409A3 (en) 2004-07-28
AU1930301A (en) 2001-06-18
EP1165072A2 (en) 2002-01-02
EA003639B1 (ru) 2003-08-28
KR100664479B1 (ko) 2007-01-04
TWI265808B (en) 2006-11-11
HRP20010582A2 (en) 2002-08-31
CN1379669A (zh) 2002-11-13
CA2362816A1 (en) 2001-06-14
WO2001041762A2 (en) 2001-06-14
PE20010940A1 (es) 2001-09-12
EE200100414A (et) 2002-12-16
IS6040A (is) 2001-08-07
CN1203852C (zh) 2005-06-01
SK12692001A3 (sk) 2002-04-04
KR20020000760A (ko) 2002-01-05
NO20013858L (no) 2001-10-08
BR0008059A (pt) 2002-03-26
EA200100872A1 (ru) 2002-02-28
IL144763A (en) 2007-09-20
AR027896A1 (es) 2003-04-16
CA2362816C (en) 2007-02-06
HUP0200409A2 (en) 2002-06-29
CR6458A (es) 2004-05-19
TR200102297T1 (tr) 2002-03-21
KR20060019639A (ko) 2006-03-03
HK1041637A1 (zh) 2002-07-19
PL351069A1 (en) 2003-03-10
AU2005200015A1 (en) 2005-02-03
NO20013858D0 (no) 2001-08-08
BG105873A (bg) 2002-04-30
NZ513963A (en) 2003-10-31
CZ20013163A3 (cs) 2002-06-12
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