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AR037255A1 - Composiciones farmaceuticas que contienen oxibutinina - Google Patents

Composiciones farmaceuticas que contienen oxibutinina

Info

Publication number
AR037255A1
AR037255A1 ARP020104230A ARP020104230A AR037255A1 AR 037255 A1 AR037255 A1 AR 037255A1 AR P020104230 A ARP020104230 A AR P020104230A AR P020104230 A ARP020104230 A AR P020104230A AR 037255 A1 AR037255 A1 AR 037255A1
Authority
AR
Argentina
Prior art keywords
drug
oxybutynin
dosage form
treatment
incontinence
Prior art date
Application number
ARP020104230A
Other languages
English (en)
Inventor
Juan Augusto Vergez
Marcelo Ricci
Original Assignee
Osmotica Argentina S A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25538393&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR037255(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Osmotica Argentina S A filed Critical Osmotica Argentina S A
Publication of AR037255A1 publication Critical patent/AR037255A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/216Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Urology & Nephrology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Se provee una composición farmacéutica y una forma de dosificación para el tratamiento de la incontinencia con oxibutinina y una segunda droga. La segunda droga puede ser cualquier droga para el tratamiento de la incontinencia. Dependiendo de la vía de administración, la forma de dosificación empleada, y la segunda droga que se utilice, la forma de dosificación puede incluir independientemente cantidades terapéuticas o subterapéuticas de oxibutinina y de la segunda droga. Realizaciones particulares incluyen una forma de dosificación que provee una liberación controlada de oxibutinina y de la segunda droga para mantener los niveles terapéuticos efectivos de oxibutinina y/o la segunda droga en un mamífero por un período de tiempo extendido. Se provee un dispositivo osmótico que comprende un núcleo bicapa. El dispositivo osmótico provee una liberación controlada dual de ambas drogas desde el núcleo. Se provee un método para el tratamiento de la incontinencia urinaria (por estrés o urgencia) con una composición farmacéutica y una forma de dosificación. Juntas, la oxibutinina y la segunda droga proveen un beneficio clínico general mejorado con relación a cualquiera de los agentes administrados solos y aproximadamente en la misma dosis.
ARP020104230A 2001-11-06 2002-11-06 Composiciones farmaceuticas que contienen oxibutinina AR037255A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US09/992,488 US20030185882A1 (en) 2001-11-06 2001-11-06 Pharmaceutical compositions containing oxybutynin

Publications (1)

Publication Number Publication Date
AR037255A1 true AR037255A1 (es) 2004-11-03

Family

ID=25538393

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP020104230A AR037255A1 (es) 2001-11-06 2002-11-06 Composiciones farmaceuticas que contienen oxibutinina
ARP020104231A AR037256A1 (es) 2001-11-06 2002-11-06 Forma de dosificacion de liberacion controlada dual

Family Applications After (1)

Application Number Title Priority Date Filing Date
ARP020104231A AR037256A1 (es) 2001-11-06 2002-11-06 Forma de dosificacion de liberacion controlada dual

Country Status (7)

Country Link
US (2) US20030185882A1 (es)
EP (1) EP1461018A2 (es)
AR (2) AR037255A1 (es)
AU (2) AU2002363361A1 (es)
BR (1) BR0213948A (es)
UY (2) UY27533A1 (es)
WO (2) WO2003039436A2 (es)

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Also Published As

Publication number Publication date
UY27533A1 (es) 2003-05-30
US8241667B2 (en) 2012-08-14
WO2003039436A2 (es) 2003-05-15
WO2003039519A3 (es) 2004-03-25
US20030185882A1 (en) 2003-10-02
US20060177510A1 (en) 2006-08-10
UY27532A1 (es) 2003-05-30
AR037256A1 (es) 2004-11-03
WO2003039436A3 (es) 2004-02-26
AU2002363360A1 (en) 2003-05-19
BR0213948A (pt) 2004-08-31
AU2002363361A1 (en) 2003-05-19
WO2003039519A2 (es) 2003-05-15
EP1461018A2 (en) 2004-09-29

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