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CN1362242A - Nano dark plum medicine and its preparation - Google Patents

Nano dark plum medicine and its preparation Download PDF

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Publication number
CN1362242A
CN1362242A CN 01100744 CN01100744A CN1362242A CN 1362242 A CN1362242 A CN 1362242A CN 01100744 CN01100744 CN 01100744 CN 01100744 A CN01100744 A CN 01100744A CN 1362242 A CN1362242 A CN 1362242A
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China
Prior art keywords
nano
nanometric
parts
chinese
dark plum
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CN 01100744
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Chinese (zh)
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杨孟君
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Individual
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Individual
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Priority to CN 01100744 priority Critical patent/CN1362242A/en
Publication of CN1362242A publication Critical patent/CN1362242A/en
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Abstract

The present invention discloses a nano mume preparation medicine. It is made up by using 9 Chinese medicinal materials of nano mume, nano asarum, nano dried ginger, nano tangkuei, nano aconite and othera as raw material through the processes of microwave extraction, reduced pressure concentration and supersonic jet spary drying. Its grain fineness is up to 1200-1500 meshes, grain size is 0.1-200 nm, in which most of grain size is less than 100 nm. Said medicine is high in biological utilization rate and obvious in therapeutic effect.

Description

Nano dark plum preparation medicine and preparation method thereof
The present invention relates to a kind of relieving pain by calming ascaris, the dirty nano dark plum preparation medicine of tonify deficiency temperature, the invention still further relates to the method for this medication preparation.
Wumei pills is a kind of classical Chinese patent medicine, mainly contain the anesthesia polypide, strengthen gallbladder and shrink, increase effects such as bile secretion, lax Oddi's sphincter, antibacterial, analgesia, being used for colic caused by ascaris, headache due to JUE YIN disorder, unhappy vomiting, time ends when sending out, must eat and then tell even do when vomiting ascaris, deadly cold hand and foot, stomachache.But traditional wumei pills absorbs not exclusively, and bioavailability is not high, slow curative effect.
The object of the present invention is to provide a kind of bioavailability height, solid dispersion is good, absorbs fully the nano dark plum preparation medicine of increase evident in efficacy.
Another object of the present invention provides the preparation method of this nano dark plum preparation medicine.
To achieve these goals, the present invention takes following technical scheme:
Medicine of the present invention is to make (consumption is a weight portion) by following component:
Nano dark plum 5-50 part nanometric Herbra Asarum 5-50 part nanometric ginger 5-50 part
Nano Chinese angelica 10-60 part nanometric Radix Aconiti Lateralis Preparata 5-50 part nanometric Zanthoxylum piperitum D.C. 5-50 part
Nano phellodendron bark 10-50 part nanometer coptis 10-50 part nano ginseng 5-50 part
The formula optimization weight proportion scope of medicine of the present invention is:
Nano dark plum 15-40 part nanometric Herbra Asarum 10-30 part nanometric ginger 10-30 part
Nano Chinese angelica 20-50 part nanometric Radix Aconiti Lateralis Preparata 10-30 part nanometric Zanthoxylum piperitum D.C. 15-40 part
Nano phellodendron bark 20-40 part nanometer coptis 18-40 part nano ginseng 10-30 part
The optimum weight proportioning of medicine of the present invention is:
18 parts of 20 parts of nanometric gingers of 25 parts of nanometric Herbra Asarums of nano dark plum
22 parts of 20 parts of nanometric Zanthoxylum piperitum D.C.s of 28 parts of nanometric Radix Aconiti Lateralis Preparatas of nano Chinese angelica
18 parts of 26 parts of nano ginsengs of 30 parts of nanometer coptis of nano phellodendron bark
Technical scheme of the present invention is based on the modern material technology.One of modern material Developing Trend in Technology is to develop to the more and more littler direction of yardstick.The granule of the past composition material, its size all are at micron or more than the millimeter magnitude, and have occurred the material to the nanoscale development now.Because extremely refinement of granule, the shared percentage by volume of crystal boundary increases, and makes some performance of material that outstanding variation take place.
The property of nano material is because the special construction of nano material---the particle size of material is less than the ultra-micro powder of 100nm, its body surface area is very big, the atom number ratio at crystal boundary place makes it to produce four big effects up to 15%-50%: i.e. small-size effect, quantum effect (containing macro quanta tunnel effect), skin effect and interfacial effect.Thereby has the not available physical and chemical performance of traditional material.Nanotechnology will bring a technological revolution of the field of Chinese medicines.
One of method of above-mentioned each component being made medicine of the present invention is:
1. divide and get the Chinese crude drug of respectively distinguishing the flavor of, add to concoct according to Chinese Pharmacopoeia one one of version in 2000 and be processed into the common Chinese decoction pieces
2. divide and get the common Chinese decoction pieces of respectively distinguishing the flavor of, be processed into the nanometer prepared slices of Chinese crude drugs, its method comprises the following steps:
1. the common Chinese decoction pieces is placed extraction pot, solubilizer also imports microwave extracting, makes its speed with 20-30 hundred million times/second do the change in polarity motion, and the temperature of its microwave extracting is 30 ℃-60 ℃, time 1-10 hour;
2. above-mentioned extract is carried out concentrating under reduced pressure, temperature is 30 ℃-60 ℃, and the time is 3-72 hour, collects volatile material in the Chinese medicine simultaneously in addition:
3. decompressed concentrate and volatile material merging are placed spray drying tower, use the supersonic jet technology, 330 meters-990 meter per seconds of effluxvelocity, 30 ℃ of-60 ℃ of temperature, under 0 to the 0.05MPa pressure,, promptly make the nanometer prepared slices of Chinese crude drugs with the instantaneous drying of hypersonic velocity.
3. the nanometer prepared slices of Chinese crude drugs (powder) are prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent standard, make pill, powder, tablet, suppository, granule, membrane, capsule, microcapsule, drop pill, aerosol, injection, unguentum, medicated wine, syrup, oral solution.
Two of medicine method for making of the present invention is:
1. be equipped with whole common Chinese decoction pieces in the proportioning ratio, place extraction pot, solubilizer also imports microwave extracting, makes its speed with 20-30 hundred million times/second do the change in polarity motion, and the temperature of its microwave extracting is 30 ℃-60 ℃, time 1-10 hour;
2. above-mentioned extract is carried out concentrating under reduced pressure, temperature is 30 ℃-60 ℃, and the time is 3-72 hour, collects volatile material in the Chinese medicine simultaneously in addition;
3. decompressed concentrate and volatile material merging are placed spray drying tower, use the supersonic jet technology, 330 meters-990 meter per seconds of effluxvelocity, 30 ℃ of-60 ℃ of temperature, under 0 to the 0.05MPa pressure,, get Fructus Mume preparation nano powder with the instantaneous drying of hypersonic velocity jet;
4. its nano powder is made aforementioned various preparation according to Chinese Pharmacopoeia version standard preparation in 2000.
The pharmacological effect that above-mentioned two kinds of methods are made the nano dark plum preparation medicine is identical.
A kind of important feature of the present invention is: the made drug material of the present invention has reached nanoscale, common wumei pills preparation material is micron or the above particle diameter of millimeter, can only cross the 80-120 mesh sieve, the drug material that the present invention is made, particle diameter is at 0.1-200nm, the overwhelming majority can be crossed the 1200-1500 mesh sieve less than 100nm.
Another important feature of the present invention is: solid preparation of the present invention disintegrate rapidly, and solid dispersion is good in water, absorb fully, the bioavailability height, the pharmacological action effect that mainly contains effective constituent is significantly higher than conventional formulation.
The pharmaceutical preparation that the present invention is made does not need to add any adjuvant, and is more favourable to human body.
The present invention has also created the new drug formulation that suppository, membrane, microcapsule, drop pill, aerosol, injection, medicated wine, syrup, oral solution of nano dark plum preparation medicine etc. is had no precedent in the past.
Pharmaceutical preparation of the present invention can be used for treatment of conditions such as ascariasis of biliary tract, bellyworm, schistosomicide and ancylostomiasis, diarrhoea, enteritis, irritable bowel syndrome, cholecystitis and cholelithiasis, nerve and spirit disease, ill antrum syndrome, leukorrhagia, metrorrhagia, dysmenorrhea, and clinical efficacy significantly is better than traditional wumei pills.
The present invention's added solvent in microwave extracting is water or ethanol.
The present invention carries out in the concentrating under reduced pressure step at extract, and its concentrating under reduced pressure is conventional scheme.
Embodiment 1:
Prepare nano raw material by preceding method:
18 parts of 20 parts of nanometric gingers of 25 parts of nanometric Herbra Asarums of nano dark plum
22 parts of 20 parts of nanometric Zanthoxylum piperitum D.C.s of 28 parts of nanometric Radix Aconiti Lateralis Preparatas of nano Chinese angelica
18 parts of 26 parts of nano ginsengs of 30 parts of nanometer coptis of nano phellodendron bark
Production method is as follows:
In the GMP cleaning shop, after the above-mentioned nanometer prepared slices of Chinese crude drugs or powder prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent capsules agent standard, do not add adjuvant, do not granulate, directly divide encapsulated with the fully-automatic capsule racking machine, make capsule, every capsules content of dispersion is a 0.1-0.6 gram, and the patient takes 1-4 time every day, every day the 1-5 grain.
Embodiment 2:
Prepare nano raw material by preceding method:
18 parts of 20 parts of nanometric gingers of 25 parts of nanometric Herbra Asarums of nano dark plum
22 parts of 20 parts of nanometric Zanthoxylum piperitum D.C.s of 28 parts of nanometric Radix Aconiti Lateralis Preparatas of nano Chinese angelica
18 parts of 26 parts of nano ginsengs of 30 parts of nanometer coptis of nano phellodendron bark
Production method is as follows:
In the GMP cleaning shop, after the above-mentioned nanometer prepared slices of Chinese crude drugs or powder prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent powder needle injection standard, do not add any adjuvant, make the nano dark plum powder needle injection, every injection content is the 5-20 milligram, and each consumption is that 1-2 props up, and use 1-3 every day.
Embodiment 3:
Prepare nano raw material by preceding method:
18 parts of 20 parts of nanometric gingers of 25 parts of nanometric Herbra Asarums of nano dark plum
22 parts of 20 parts of nanometric Zanthoxylum piperitum D.C.s of 28 parts of nanometric Radix Aconiti Lateralis Preparatas of nano Chinese angelica
18 parts of 26 parts of nano ginsengs of 30 parts of nanometer coptis of nano phellodendron bark
Production method is as follows:
In the GMP cleaning shop, after the above-mentioned nanometer prepared slices of Chinese crude drugs or powder prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent membrane standard, filmogen adopts polyvinyl alcohol, make the nano dark plum membrane, every membrane area size is the 2-100 square centimeter, and content of dispersion is the 1-50 gram, every medicine film pasted 1-7 days, pasted the medicine position: abdominal part.

Claims (6)

1, a kind of nano dark plum preparation medicine is characterized in that it is the medicament that the nano raw material of following weight proportioning is made:
Nano dark plum 5-50 part nanometric Herbra Asarum 5-50 part nanometric ginger 5-50 part
Nano Chinese angelica 10-60 part nanometric Radix Aconiti Lateralis Preparata 5-50 part nanometric Zanthoxylum piperitum D.C. 5-50 part
Nano phellodendron bark 10-50 part nanometer coptis 10-50 part nano ginseng 5-50 part
And adopt following method to make: to select the formula Chinese drug material to concoct and be processed into the prepared slices of Chinese crude drugs; Place extraction pot, solubilizer also imports microwave extracting, makes it do the change in polarity motion with hundred million times/second speed of 20--30, and the temperature of its microwave extracting is 30--60 ℃, time 1--10 hour; Above-mentioned extract is carried out concentrating under reduced pressure, and temperature is 30--60 ℃, and the time is 3--72 hour, collects volatile material in the Chinese medicine simultaneously in addition; Decompressed concentrate and volatile material merging are placed spray drying tower, use the Supersonic fluidics, 30--60 ℃ of temperature, under 0 to the 0.05MPa pressure, with hypersonic velocity instantaneous jet drying, wherein supersonic jet speed is 330 meters--990 meter per seconds, promptly make the nanometer prepared slices of Chinese crude drugs.
2, nano dark plum preparation medicine according to claim 1, wherein the weight proportion of each nano raw material is:
Nano dark plum 15-40 part nanometric Herbra Asarum 10-30 part nanometric ginger 10-30 part
Nano Chinese angelica 20-50 part nanometric Radix Aconiti Lateralis Preparata 10-30 part nanometric Zanthoxylum piperitum D.C. 15-40 part
Nano phellodendron bark 20-40 part nanometer coptis 18-40 part nano ginseng 10-30 part
3, nano dark plum preparation medicine according to claim 1, wherein the weight proportion of each nano raw material is:
18 parts of 20 parts of nanometric gingers of 25 parts of nanometric Herbra Asarums of nano dark plum
22 parts of 20 parts of nanometric Zanthoxylum piperitum D.C.s of 28 parts of nanometric Radix Aconiti Lateralis Preparatas of nano Chinese angelica
18 parts of 26 parts of nano ginsengs of 30 parts of nanometer coptis of nano phellodendron bark
4,, it is characterized in that said medicine is pill, powder, tablet, suppository, granule, membrane, capsule, microcapsule, drop pill, aerosol, injection, unguentum, medicated wine, syrup, oral solution according to claim 1 or 2 or 3 described nano dark plum preparation medicines.
5,, it is characterized in that this method comprises the steps: to select the formula Chinese drug material to concoct and is processed into the prepared slices of Chinese crude drugs according to the pharmaceutical methods of claim 1 or 2 or 3 described nano dark plum preparation medicines; Place extraction pot, solubilizer also imports microwave extracting, makes it do the change in polarity motion with hundred million times/second speed of 20--30, and the temperature of its microwave extracting is 30--60 ℃, time 1--10 hour; Above-mentioned extract is carried out concentrating under reduced pressure, and temperature is 30--60 ℃, and the time is 3--72 hour, collects volatile material in the Chinese medicine simultaneously in addition; Decompressed concentrate and volatile material merging are placed spray drying tower, use the Supersonic fluidics, 30--60 ℃ of temperature, under 0 to the 0.05MPa pressure, with hypersonic velocity instantaneous jet drying, wherein supersonic jet speed is 330 meters--990 meter per seconds, promptly make the nanometer prepared slices of Chinese crude drugs.
6, wherein respectively distinguish the flavor of Chinese medicine in the ratio of prescription or Chinese crude drug concoct be processed into the prepared slices of Chinese crude drugs after mixing, or after making the nanometer prepared slices of Chinese crude drugs mixing.
CN 01100744 2001-01-08 2001-01-08 Nano dark plum medicine and its preparation Pending CN1362242A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CN 01100744 CN1362242A (en) 2001-01-08 2001-01-08 Nano dark plum medicine and its preparation

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CN 01100744 CN1362242A (en) 2001-01-08 2001-01-08 Nano dark plum medicine and its preparation

Publications (1)

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CN1362242A true CN1362242A (en) 2002-08-07

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Family Applications (1)

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Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104940882A (en) * 2015-07-08 2015-09-30 河南中医学院 Traditional Chinese medicine for treating chronic diarrhea
CN106177344A (en) * 2016-08-31 2016-12-07 安徽新盛中药饮片有限公司 A kind of stomach invigorating removing toxic substances Fructus Mume micro-ferment decoction pieces and preparation method thereof

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104940882A (en) * 2015-07-08 2015-09-30 河南中医学院 Traditional Chinese medicine for treating chronic diarrhea
CN104940882B (en) * 2015-07-08 2018-05-01 河南中医学院 A kind of Chinese medicine for treating chronic diarrhea
CN106177344A (en) * 2016-08-31 2016-12-07 安徽新盛中药饮片有限公司 A kind of stomach invigorating removing toxic substances Fructus Mume micro-ferment decoction pieces and preparation method thereof

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